NO20084627L - Pyrrolo- og tiazolpyridinforbindelser og fremgangsmater for anvendelse derav - Google Patents
Pyrrolo- og tiazolpyridinforbindelser og fremgangsmater for anvendelse deravInfo
- Publication number
- NO20084627L NO20084627L NO20084627A NO20084627A NO20084627L NO 20084627 L NO20084627 L NO 20084627L NO 20084627 A NO20084627 A NO 20084627A NO 20084627 A NO20084627 A NO 20084627A NO 20084627 L NO20084627 L NO 20084627L
- Authority
- NO
- Norway
- Prior art keywords
- pyrrolo
- methods
- pyridine compounds
- thiazole pyridine
- thiazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Gastroenterology & Hepatology (AREA)
- Obesity (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Endocrinology (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Foreliggende oppfinnelse angår nye forbindelser i stand til å modulere stabiliteten og/eller aktiviteten til hypoksiinduserbar faktor (HIF).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US78931006P | 2006-04-04 | 2006-04-04 | |
PCT/US2007/065987 WO2007115315A2 (en) | 2006-04-04 | 2007-04-04 | Pyrrolo- and thiazolo-pyridine compounds as hif modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20084627L true NO20084627L (no) | 2008-11-26 |
Family
ID=38477095
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20084627A NO20084627L (no) | 2006-04-04 | 2008-11-03 | Pyrrolo- og tiazolpyridinforbindelser og fremgangsmater for anvendelse derav |
Country Status (15)
Country | Link |
---|---|
US (1) | US7696223B2 (no) |
EP (2) | EP3124489B1 (no) |
JP (1) | JP5111491B2 (no) |
KR (1) | KR101084635B1 (no) |
CN (2) | CN101460497A (no) |
AU (1) | AU2007234408B2 (no) |
BR (1) | BRPI0710527B8 (no) |
CA (1) | CA2647596C (no) |
HK (1) | HK1127046A1 (no) |
IL (1) | IL194311A (no) |
MX (1) | MX2008012734A (no) |
NO (1) | NO20084627L (no) |
RU (1) | RU2461557C2 (no) |
WO (1) | WO2007115315A2 (no) |
ZA (1) | ZA200808410B (no) |
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BRPI0411055B1 (pt) | 2003-06-06 | 2018-08-21 | Fibrogen, Inc | Compostos de heteroarilas contendo nitrogênio. seus usos no aumento da eritropoietina endógena, composição farmacêutica que os compreende e método in vitro de inibição da atividade da enzima hidrolase |
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MX2008012734A (es) | 2006-04-04 | 2009-01-29 | Fibrogen Inc | Compuestos pirrolo- y tiazolo-piridina como moduladores del factor inducible de hipoxia (hif). |
US8962530B2 (en) * | 2007-06-27 | 2015-02-24 | Regents Of The University Of Colorado | Inflammatory bowel disease therapies |
US20100227846A1 (en) * | 2007-08-30 | 2010-09-09 | Takeda Pharmaceutical Company Limited | Substituted pyrazole derivative |
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2007
- 2007-04-04 MX MX2008012734A patent/MX2008012734A/es active IP Right Grant
- 2007-04-04 CN CNA200780011561XA patent/CN101460497A/zh active Pending
- 2007-04-04 US US11/696,549 patent/US7696223B2/en active Active
- 2007-04-04 EP EP16174358.8A patent/EP3124489B1/en active Active
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- 2007-04-04 CN CN201310337398.3A patent/CN103497184A/zh active Pending
- 2007-04-04 EP EP07760122.7A patent/EP2016078B1/en active Active
- 2007-04-04 WO PCT/US2007/065987 patent/WO2007115315A2/en active Application Filing
- 2007-04-04 BR BRPI0710527A patent/BRPI0710527B8/pt active IP Right Grant
- 2007-04-04 AU AU2007234408A patent/AU2007234408B2/en not_active Ceased
- 2007-04-04 RU RU2008143564/04A patent/RU2461557C2/ru active
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Also Published As
Publication number | Publication date |
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AU2007234408B2 (en) | 2011-05-19 |
BRPI0710527A2 (pt) | 2012-06-05 |
CN101460497A (zh) | 2009-06-17 |
WO2007115315A3 (en) | 2007-12-06 |
JP5111491B2 (ja) | 2013-01-09 |
MX2008012734A (es) | 2009-01-29 |
IL194311A0 (en) | 2009-08-03 |
RU2461557C2 (ru) | 2012-09-20 |
EP2016078A2 (en) | 2009-01-21 |
CN103497184A (zh) | 2014-01-08 |
JP2009532502A (ja) | 2009-09-10 |
US20080004309A1 (en) | 2008-01-03 |
KR20080112350A (ko) | 2008-12-24 |
EP2016078B1 (en) | 2016-06-15 |
EP3124489A1 (en) | 2017-02-01 |
HK1127046A1 (zh) | 2009-10-02 |
CA2647596C (en) | 2012-06-12 |
IL194311A (en) | 2015-09-24 |
ZA200808410B (en) | 2009-12-30 |
US7696223B2 (en) | 2010-04-13 |
KR101084635B1 (ko) | 2011-11-18 |
WO2007115315A2 (en) | 2007-10-11 |
CA2647596A1 (en) | 2007-10-11 |
BRPI0710527B1 (pt) | 2019-09-03 |
EP3124489B1 (en) | 2020-07-15 |
RU2008143564A (ru) | 2010-05-10 |
AU2007234408A1 (en) | 2007-10-11 |
BRPI0710527B8 (pt) | 2021-05-25 |
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