NO20075647L - Kjemiske forbindelser - Google Patents
Kjemiske forbindelserInfo
- Publication number
- NO20075647L NO20075647L NO20075647A NO20075647A NO20075647L NO 20075647 L NO20075647 L NO 20075647L NO 20075647 A NO20075647 A NO 20075647A NO 20075647 A NO20075647 A NO 20075647A NO 20075647 L NO20075647 L NO 20075647L
- Authority
- NO
- Norway
- Prior art keywords
- chemical connections
- connections
- chemical
- cancer
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US68151505P | 2005-05-16 | 2005-05-16 | |
US72228205P | 2005-09-30 | 2005-09-30 | |
PCT/GB2006/001760 WO2006123113A2 (en) | 2005-05-16 | 2006-05-12 | Pyrazolylaminopyrimidine derivatives useful as tyrosine kinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20075647L true NO20075647L (no) | 2007-12-13 |
Family
ID=37087720
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20075647A NO20075647L (no) | 2005-05-16 | 2007-11-06 | Kjemiske forbindelser |
Country Status (15)
Country | Link |
---|---|
US (2) | US20080287437A1 (de) |
EP (1) | EP1899323A2 (de) |
JP (1) | JP2008540622A (de) |
KR (1) | KR20080015409A (de) |
AR (1) | AR056354A1 (de) |
AU (1) | AU2006248780B2 (de) |
BR (1) | BRPI0610184A2 (de) |
CA (1) | CA2608009A1 (de) |
IL (1) | IL186845A0 (de) |
MX (1) | MX2007014328A (de) |
NO (1) | NO20075647L (de) |
NZ (1) | NZ564317A (de) |
TW (1) | TW200716606A (de) |
UY (1) | UY29530A1 (de) |
WO (1) | WO2006123113A2 (de) |
Families Citing this family (71)
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ATE407132T1 (de) * | 2000-12-05 | 2008-09-15 | Vertex Pharma | Inhibitoren von c-jun n-terminalen kinasen (jnk) und anderen proteinkinasen |
PT1846394E (pt) * | 2005-02-04 | 2012-01-05 | Astrazeneca Ab | Derivados de pirazolilaminopiridina úteis como inibidores da quinase |
BRPI0607455A2 (pt) | 2005-02-16 | 2009-09-01 | Astrazeneca Ab | composto, processo para a preparação do mesmo, uso de um composto, e composição farmacêutica |
EP1899323A2 (de) * | 2005-05-16 | 2008-03-19 | AstraZeneca AB | Als tyrosinkinaseinhibitoren geeignete pyrazolylaminopyrimidinderivate |
PT1945631E (pt) * | 2005-10-28 | 2012-10-15 | Astrazeneca Ab | Derivados de 4-(3-aminopirazole)pirimidina para utilização como inibidores da tirosina-cinase no tratamento do cancro |
TW200823196A (en) * | 2006-11-01 | 2008-06-01 | Astrazeneca Ab | New use |
WO2008117050A1 (en) * | 2007-03-27 | 2008-10-02 | Astrazeneca Ab | Pyrazolyl-amino-substituted pyrazines and their use for the treatment of cancer |
US20100204246A1 (en) * | 2007-04-18 | 2010-08-12 | Astrazeneca Ab | 5-aminopyrazol-3-yl-3h-imidazo (4,5-b) pyridine derivatives and their use for the treatment of cancer |
TW200846344A (en) * | 2007-04-25 | 2008-12-01 | Astrazeneca Ab | Chemical compounds |
UA99459C2 (en) * | 2007-05-04 | 2012-08-27 | Астразенека Аб | 9-(pyrazol-3-yl)- 9h-purine-2-amine and 3-(pyraz0l-3-yl)-3h-imidazo[4,5-b]pyridin-5-amine derivatives and their use for the treatment of cancer |
ATE521609T1 (de) * | 2007-05-04 | 2011-09-15 | Astrazeneca Ab | Aminothiazolylpyrimidinderivate und ihre verwendung bei der behandlung von krebs |
WO2009007753A2 (en) * | 2007-07-11 | 2009-01-15 | Astrazeneca Ab | 4- (3-aminopyrazole) -pyrimidine derivativee and their use as tyrosine kinase inhibitors for the treatment of cancer |
WO2009013545A2 (en) * | 2007-07-26 | 2009-01-29 | Astrazeneca Ab | Chemical compounds |
TW200906818A (en) * | 2007-07-31 | 2009-02-16 | Astrazeneca Ab | Chemical compounds |
WO2009027736A2 (en) * | 2007-08-27 | 2009-03-05 | Astrazeneca Ab | 2,4 diaminopyrimid'lnes for the treatment of myeloproliferative disorders and cancer |
WO2009056886A1 (en) * | 2007-11-01 | 2009-05-07 | Astrazeneca Ab | Pyrimidine derivatives and their use as modulators of fgfr activity |
WO2009095712A2 (en) * | 2008-01-29 | 2009-08-06 | Astrazeneca Ab | Chemical compounds |
CN102119157A (zh) * | 2008-06-11 | 2011-07-06 | 阿斯利康(瑞典)有限公司 | 用于治疗癌症和骨髓增生性疾病的三环2,4-二氨基-l,3,5-三嗪衍生物 |
ES2464461T3 (es) | 2008-09-22 | 2014-06-02 | Array Biopharma, Inc. | Compuestos de imidazo[1,2B]piridazina sustituidos como inhibidores de la TRK cinasa |
TW201018693A (en) * | 2008-09-30 | 2010-05-16 | Astrazeneca Ab | Chemical compounds 496-1p |
TWI577680B (zh) | 2008-10-22 | 2017-04-11 | 亞雷生物製藥股份有限公司 | 作為TRK激酶抑制劑之經取代吡唑并〔1,5-a〕嘧啶化合物 |
EP2181980A1 (de) * | 2008-10-28 | 2010-05-05 | Chemo Ibérica, S.A. | Verfahren zur Herstellung von (R)-1-Aminoindanen |
AR077468A1 (es) | 2009-07-09 | 2011-08-31 | Array Biopharma Inc | Compuestos de pirazolo (1,5 -a) pirimidina sustituidos como inhibidores de trk- quinasa |
NZ604708A (en) | 2010-05-20 | 2015-05-29 | Array Biopharma Inc | Macrocyclic compounds as trk kinase inhibitors |
JP2012102088A (ja) * | 2010-10-14 | 2012-05-31 | Sumitomo Chemical Co Ltd | ヘテロ芳香環化合物およびその有害生物防除用途 |
EP2731439A4 (de) | 2011-07-12 | 2014-12-03 | Merck Sharp & Dohme | Trka-kinase-hemmer, zusammensetzungen daraus und verfahren dafür |
EP2554544A1 (de) | 2011-08-01 | 2013-02-06 | Almirall, S.A. | Pyridin-2(1H-)-on-Derivate als JAK-Inhibitoren |
KR20140062079A (ko) | 2011-08-25 | 2014-05-22 | 에프. 호프만-라 로슈 아게 | 세린/트레오닌 pak1 억제제 |
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EP2858501A4 (de) | 2012-05-22 | 2015-12-09 | Merck Sharp & Dohme | Trka-kinase-hemmer, zusammensetzungen daraus und verfahren dafür |
US10407509B2 (en) | 2013-07-30 | 2019-09-10 | Blueprint Medicines Corporation | NTRK2 fusions |
WO2015039334A1 (en) | 2013-09-22 | 2015-03-26 | Merck Sharp & Dohme Corp. | TrkA KINASE INHIBITORS, COMPOSITIONS AND METHODS THEREOF |
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JP7061068B2 (ja) | 2015-12-18 | 2022-04-27 | イグナイタ インコーポレイテッド | 癌治療のための併用薬 |
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PT1846394E (pt) * | 2005-02-04 | 2012-01-05 | Astrazeneca Ab | Derivados de pirazolilaminopiridina úteis como inibidores da quinase |
BRPI0607455A2 (pt) | 2005-02-16 | 2009-09-01 | Astrazeneca Ab | composto, processo para a preparação do mesmo, uso de um composto, e composição farmacêutica |
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TW200826937A (en) | 2006-11-01 | 2008-07-01 | Astrazeneca Ab | New use |
TW200823196A (en) | 2006-11-01 | 2008-06-01 | Astrazeneca Ab | New use |
-
2006
- 2006-05-12 EP EP06727105A patent/EP1899323A2/de not_active Withdrawn
- 2006-05-12 WO PCT/GB2006/001760 patent/WO2006123113A2/en active Application Filing
- 2006-05-12 CA CA002608009A patent/CA2608009A1/en not_active Abandoned
- 2006-05-12 AU AU2006248780A patent/AU2006248780B2/en not_active Ceased
- 2006-05-12 BR BRPI0610184-4A patent/BRPI0610184A2/pt not_active IP Right Cessation
- 2006-05-12 MX MX2007014328A patent/MX2007014328A/es unknown
- 2006-05-12 KR KR1020077026987A patent/KR20080015409A/ko not_active Application Discontinuation
- 2006-05-12 NZ NZ564317A patent/NZ564317A/en not_active IP Right Cessation
- 2006-05-12 JP JP2008511776A patent/JP2008540622A/ja active Pending
- 2006-05-12 US US11/914,492 patent/US20080287437A1/en not_active Abandoned
- 2006-05-15 UY UY29530A patent/UY29530A1/es unknown
- 2006-05-16 AR ARP060101974A patent/AR056354A1/es not_active Application Discontinuation
- 2006-05-16 TW TW095117309A patent/TW200716606A/zh unknown
-
2007
- 2007-10-22 IL IL186845A patent/IL186845A0/en unknown
- 2007-11-06 NO NO20075647A patent/NO20075647L/no not_active Application Discontinuation
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2010
- 2010-02-26 US US12/713,777 patent/US8114989B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
MX2007014328A (es) | 2008-02-12 |
AU2006248780A1 (en) | 2006-11-23 |
BRPI0610184A2 (pt) | 2012-09-25 |
IL186845A0 (en) | 2008-02-09 |
JP2008540622A (ja) | 2008-11-20 |
US8114989B2 (en) | 2012-02-14 |
NZ564317A (en) | 2011-01-28 |
AR056354A1 (es) | 2007-10-03 |
CA2608009A1 (en) | 2006-11-23 |
US20080287437A1 (en) | 2008-11-20 |
WO2006123113A3 (en) | 2007-01-04 |
US20100210648A1 (en) | 2010-08-19 |
WO2006123113A2 (en) | 2006-11-23 |
EP1899323A2 (de) | 2008-03-19 |
TW200716606A (en) | 2007-05-01 |
UY29530A1 (es) | 2006-12-29 |
KR20080015409A (ko) | 2008-02-19 |
AU2006248780B2 (en) | 2010-06-03 |
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