MA52218A - Traitement de cancers associés à trk - Google Patents

Traitement de cancers associés à trk

Info

Publication number
MA52218A
MA52218A MA052218A MA52218A MA52218A MA 52218 A MA52218 A MA 52218A MA 052218 A MA052218 A MA 052218A MA 52218 A MA52218 A MA 52218A MA 52218 A MA52218 A MA 52218A
Authority
MA
Morocco
Prior art keywords
trk
treatment
cancers associated
cancers
Prior art date
Application number
MA052218A
Other languages
English (en)
Inventor
Joshua H Bilenker
Nisha Nanda
Naarden Jacob Van
Original Assignee
Loxo Oncology Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Loxo Oncology Inc filed Critical Loxo Oncology Inc
Publication of MA52218A publication Critical patent/MA52218A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MA052218A 2018-03-29 2019-03-29 Traitement de cancers associés à trk MA52218A (fr)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201862650255P 2018-03-29 2018-03-29
US201862679426P 2018-06-01 2018-06-01
US201862683821P 2018-06-12 2018-06-12
US201862686524P 2018-06-18 2018-06-18
US201862721269P 2018-08-22 2018-08-22
US201962795422P 2019-01-22 2019-01-22
US201962804617P 2019-02-12 2019-02-12

Publications (1)

Publication Number Publication Date
MA52218A true MA52218A (fr) 2021-02-17

Family

ID=66429531

Family Applications (1)

Application Number Title Priority Date Filing Date
MA052218A MA52218A (fr) 2018-03-29 2019-03-29 Traitement de cancers associés à trk

Country Status (5)

Country Link
US (1) US20210023086A1 (fr)
EP (1) EP3773725A1 (fr)
CA (1) CA3095366A1 (fr)
MA (1) MA52218A (fr)
WO (1) WO2019191659A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI577680B (zh) 2008-10-22 2017-04-11 亞雷生物製藥股份有限公司 作為TRK激酶抑制劑之經取代吡唑并〔1,5-a〕嘧啶化合物
CR20180501A (es) 2016-04-04 2019-04-05 Loxo Oncology Inc Formulaciones liquidas de (s)-n-(5-((r)-2(2,5-difluorofenil)-pirrolidin-1-il)-pirazolo[1,5-a] pirimidin-3-il)-3-hidroxipirrolidina-1-carboxamida
US10045991B2 (en) 2016-04-04 2018-08-14 Loxo Oncology, Inc. Methods of treating pediatric cancers
SI3458456T1 (sl) 2016-05-18 2021-04-30 Loxo Oncology, Inc. Priprava (S)-N-(5-((R)-2-(2,5-difluorofenil) pirolidin-1-il) pirazolo (1,5-A) pirimidin-3-il)-3-hidroksipirolidin-1-karboksamida
JOP20190092A1 (ar) 2016-10-26 2019-04-25 Array Biopharma Inc عملية لتحضير مركبات بيرازولو[1، 5-a]بيريميدين وأملاح منها
BR112021007679A2 (pt) 2018-10-22 2021-07-27 Esker Therapeutics, Inc inibidores de tyk2 e seus usos
EP4180428A1 (fr) 2021-11-12 2023-05-17 Genzyme Corporation Composé cristallin d'imidazo[4,5-b]pyridine, compositions pharmaceutiques et leur utilisation dans le traitement d'états médicaux

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Also Published As

Publication number Publication date
CA3095366A1 (fr) 2019-10-03
WO2019191659A1 (fr) 2019-10-03
US20210023086A1 (en) 2021-01-28
EP3773725A1 (fr) 2021-02-17

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