NO20043726L - Heteroarylforbindelser anvendelige som inhibitorer av GSK-3 - Google Patents
Heteroarylforbindelser anvendelige som inhibitorer av GSK-3Info
- Publication number
- NO20043726L NO20043726L NO20043726A NO20043726A NO20043726L NO 20043726 L NO20043726 L NO 20043726L NO 20043726 A NO20043726 A NO 20043726A NO 20043726 A NO20043726 A NO 20043726A NO 20043726 L NO20043726 L NO 20043726L
- Authority
- NO
- Norway
- Prior art keywords
- gsk
- inhibitors
- compounds useful
- heteroaryl compounds
- heteroaryl
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4245—Oxadiazoles
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A—HUMAN NECESSITIES
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US35484302P | 2002-02-06 | 2002-02-06 | |
PCT/US2003/003655 WO2003066629A2 (en) | 2002-02-06 | 2003-02-06 | Heteroaryl compounds useful as inhibitors of gsk-3 |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20043726L true NO20043726L (no) | 2004-11-08 |
Family
ID=27734431
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20043726A NO20043726L (no) | 2002-02-06 | 2004-09-06 | Heteroarylforbindelser anvendelige som inhibitorer av GSK-3 |
Country Status (13)
Country | Link |
---|---|
US (2) | US20040034037A1 (es) |
EP (2) | EP1472245A2 (es) |
JP (2) | JP4656838B2 (es) |
KR (1) | KR20040084896A (es) |
AU (1) | AU2003215087B2 (es) |
CA (1) | CA2475633C (es) |
ES (1) | ES2437391T3 (es) |
MX (1) | MXPA04007697A (es) |
NO (1) | NO20043726L (es) |
PL (1) | PL372198A1 (es) |
RU (1) | RU2004126671A (es) |
SG (1) | SG159380A1 (es) |
WO (1) | WO2003066629A2 (es) |
Families Citing this family (116)
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ATE294797T1 (de) * | 2000-09-15 | 2005-05-15 | Vertex Pharma | Pyrazolverbindungen als protein-kinasehemmer |
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GB0206860D0 (en) * | 2002-03-22 | 2002-05-01 | Glaxo Group Ltd | Compounds |
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2003
- 2003-02-06 AU AU2003215087A patent/AU2003215087B2/en not_active Ceased
- 2003-02-06 JP JP2003566002A patent/JP4656838B2/ja not_active Expired - Fee Related
- 2003-02-06 RU RU2004126671/04A patent/RU2004126671A/ru not_active Application Discontinuation
- 2003-02-06 PL PL03372198A patent/PL372198A1/xx not_active Application Discontinuation
- 2003-02-06 EP EP03710903A patent/EP1472245A2/en not_active Withdrawn
- 2003-02-06 MX MXPA04007697A patent/MXPA04007697A/es not_active Application Discontinuation
- 2003-02-06 KR KR10-2004-7012258A patent/KR20040084896A/ko not_active Application Discontinuation
- 2003-02-06 CA CA2475633A patent/CA2475633C/en not_active Expired - Fee Related
- 2003-02-06 WO PCT/US2003/003655 patent/WO2003066629A2/en active Application Filing
- 2003-02-06 ES ES10180554.7T patent/ES2437391T3/es not_active Expired - Lifetime
- 2003-02-06 SG SG200605228-6A patent/SG159380A1/en unknown
- 2003-02-06 EP EP10180554.7A patent/EP2322521B1/en not_active Expired - Lifetime
- 2003-02-06 US US10/360,535 patent/US20040034037A1/en not_active Abandoned
-
2004
- 2004-09-06 NO NO20043726A patent/NO20043726L/no unknown
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2007
- 2007-07-12 US US11/776,756 patent/US20070270420A1/en not_active Abandoned
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2010
- 2010-02-26 JP JP2010043557A patent/JP2010132697A/ja active Pending
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WO2003066629A3 (en) | 2003-10-30 |
EP2322521A1 (en) | 2011-05-18 |
KR20040084896A (ko) | 2004-10-06 |
CA2475633C (en) | 2013-04-02 |
JP4656838B2 (ja) | 2011-03-23 |
PL372198A1 (en) | 2005-07-11 |
SG159380A1 (en) | 2010-03-30 |
WO2003066629A2 (en) | 2003-08-14 |
EP1472245A2 (en) | 2004-11-03 |
US20040034037A1 (en) | 2004-02-19 |
ES2437391T3 (es) | 2014-01-10 |
AU2003215087B2 (en) | 2009-07-16 |
CA2475633A1 (en) | 2003-08-14 |
MXPA04007697A (es) | 2004-11-10 |
AU2003215087A1 (en) | 2003-09-02 |
US20070270420A1 (en) | 2007-11-22 |
JP2005526028A (ja) | 2005-09-02 |
EP2322521B1 (en) | 2013-09-04 |
RU2004126671A (ru) | 2005-04-10 |
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