NO20032290L - Nye forbindelser for anvendelse som HIV-protease-inhibitorer - Google Patents

Nye forbindelser for anvendelse som HIV-protease-inhibitorer

Info

Publication number
NO20032290L
NO20032290L NO20032290A NO20032290A NO20032290L NO 20032290 L NO20032290 L NO 20032290L NO 20032290 A NO20032290 A NO 20032290A NO 20032290 A NO20032290 A NO 20032290A NO 20032290 L NO20032290 L NO 20032290L
Authority
NO
Norway
Prior art keywords
protease inhibitors
new compounds
hiv protease
hiv
compounds
Prior art date
Application number
NO20032290A
Other languages
English (en)
Norwegian (no)
Other versions
NO20032290D0 (no
Inventor
Joseph Armstrong Martin
Sally Redshaw
Steven Swallow
Gareth John Thomas
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO20032290D0 publication Critical patent/NO20032290D0/no
Publication of NO20032290L publication Critical patent/NO20032290L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20032290A 2000-11-22 2003-05-21 Nye forbindelser for anvendelse som HIV-protease-inhibitorer NO20032290L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0028483.6A GB0028483D0 (en) 2000-11-22 2000-11-22 Hydroxyethylamine HIV protease inhibitors
PCT/EP2001/013068 WO2002042277A1 (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors

Publications (2)

Publication Number Publication Date
NO20032290D0 NO20032290D0 (no) 2003-05-21
NO20032290L true NO20032290L (no) 2003-05-21

Family

ID=9903670

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20032290A NO20032290L (no) 2000-11-22 2003-05-21 Nye forbindelser for anvendelse som HIV-protease-inhibitorer

Country Status (27)

Country Link
US (1) US6472404B1 (cs)
EP (1) EP1339692A1 (cs)
JP (1) JP2004520283A (cs)
KR (1) KR20030060953A (cs)
CN (1) CN1476436A (cs)
AR (1) AR031763A1 (cs)
AU (2) AU2954602A (cs)
BG (1) BG107839A (cs)
BR (1) BR0115566A (cs)
CA (1) CA2428459A1 (cs)
CZ (1) CZ20031667A3 (cs)
EC (1) ECSP034618A (cs)
GB (1) GB0028483D0 (cs)
GT (1) GT200100233A (cs)
HU (1) HUP0303007A2 (cs)
IL (1) IL155573A0 (cs)
MA (1) MA26966A1 (cs)
MX (1) MXPA03004534A (cs)
NO (1) NO20032290L (cs)
NZ (1) NZ525550A (cs)
PA (1) PA8533401A1 (cs)
PE (1) PE20020610A1 (cs)
PL (1) PL366704A1 (cs)
RU (1) RU2265016C2 (cs)
SK (1) SK7602003A3 (cs)
UY (1) UY27033A1 (cs)
WO (1) WO2002042277A1 (cs)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4953297B2 (ja) * 2004-09-15 2012-06-13 塩野義製薬株式会社 Hivインテグラーゼ阻害活性を有するカルバモイルピリドン誘導体
UA87884C2 (uk) * 2004-12-03 2009-08-25 Мерк Энд Ко., Инк. Безводна кристалічна калієва сіль інгібітора віл-інтегрази
CN101981012A (zh) * 2008-03-26 2011-02-23 第一三共株式会社 新的四氢异喹啉衍生物
US12083099B2 (en) 2020-10-28 2024-09-10 Accencio LLC Methods of treating symptoms of coronavirus infection with viral protease inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8927913D0 (en) 1989-12-11 1990-02-14 Hoffmann La Roche Amino acid derivatives
US5484926A (en) * 1993-10-07 1996-01-16 Agouron Pharmaceuticals, Inc. HIV protease inhibitors
MX9308016A (es) * 1992-12-22 1994-08-31 Lilly Co Eli Compuestos inhibidores de la proteasa del virus de la inmunodeficiencia humana, procedimiento para su preparacion y formulacion farmaceutica que los contiene.

Also Published As

Publication number Publication date
ECSP034618A (es) 2003-06-25
NO20032290D0 (no) 2003-05-21
PL366704A1 (en) 2005-02-07
BR0115566A (pt) 2003-09-30
IL155573A0 (en) 2003-11-23
EP1339692A1 (en) 2003-09-03
BG107839A (bg) 2004-06-30
WO2002042277A1 (en) 2002-05-30
PA8533401A1 (es) 2002-10-31
US6472404B1 (en) 2002-10-29
RU2003117468A (ru) 2005-01-27
UY27033A1 (es) 2002-06-20
NZ525550A (en) 2004-11-26
SK7602003A3 (en) 2004-01-08
GT200100233A (es) 2002-07-04
MA26966A1 (fr) 2004-12-20
AU2002229546B2 (en) 2006-05-04
HUP0303007A2 (hu) 2003-12-29
MXPA03004534A (es) 2003-09-10
CN1476436A (zh) 2004-02-18
CZ20031667A3 (cs) 2004-01-14
RU2265016C2 (ru) 2005-11-27
CA2428459A1 (en) 2002-05-30
PE20020610A1 (es) 2002-07-13
JP2004520283A (ja) 2004-07-08
KR20030060953A (ko) 2003-07-16
GB0028483D0 (en) 2001-01-10
AU2954602A (en) 2002-06-03
AR031763A1 (es) 2003-10-01

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