MXPA03004534A - Compuestos novedosos para su uso como inhibidores de la proteasa del virus de inmunodeficiencia humana (vih). - Google Patents
Compuestos novedosos para su uso como inhibidores de la proteasa del virus de inmunodeficiencia humana (vih).Info
- Publication number
- MXPA03004534A MXPA03004534A MXPA03004534A MXPA03004534A MXPA03004534A MX PA03004534 A MXPA03004534 A MX PA03004534A MX PA03004534 A MXPA03004534 A MX PA03004534A MX PA03004534 A MXPA03004534 A MX PA03004534A MX PA03004534 A MXPA03004534 A MX PA03004534A
- Authority
- MX
- Mexico
- Prior art keywords
- protease inhibitors
- novel compounds
- hiv protease
- hiv
- inhibitors
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0028483.6A GB0028483D0 (en) | 2000-11-22 | 2000-11-22 | Hydroxyethylamine HIV protease inhibitors |
| PCT/EP2001/013068 WO2002042277A1 (en) | 2000-11-22 | 2001-11-12 | Novel compounds for use as hiv protease inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA03004534A true MXPA03004534A (es) | 2003-09-10 |
Family
ID=9903670
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA03004534A MXPA03004534A (es) | 2000-11-22 | 2001-11-12 | Compuestos novedosos para su uso como inhibidores de la proteasa del virus de inmunodeficiencia humana (vih). |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US6472404B1 (es) |
| EP (1) | EP1339692A1 (es) |
| JP (1) | JP2004520283A (es) |
| KR (1) | KR20030060953A (es) |
| CN (1) | CN1476436A (es) |
| AR (1) | AR031763A1 (es) |
| AU (2) | AU2002229546B2 (es) |
| BG (1) | BG107839A (es) |
| BR (1) | BR0115566A (es) |
| CA (1) | CA2428459A1 (es) |
| CZ (1) | CZ20031667A3 (es) |
| EC (1) | ECSP034618A (es) |
| GB (1) | GB0028483D0 (es) |
| GT (1) | GT200100233A (es) |
| HU (1) | HUP0303007A2 (es) |
| IL (1) | IL155573A0 (es) |
| MA (1) | MA26966A1 (es) |
| MX (1) | MXPA03004534A (es) |
| NO (1) | NO20032290D0 (es) |
| NZ (1) | NZ525550A (es) |
| PA (1) | PA8533401A1 (es) |
| PE (1) | PE20020610A1 (es) |
| PL (1) | PL366704A1 (es) |
| RU (1) | RU2265016C2 (es) |
| SK (1) | SK7602003A3 (es) |
| UY (1) | UY27033A1 (es) |
| WO (1) | WO2002042277A1 (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7550463B2 (en) * | 2004-09-15 | 2009-06-23 | Shionogi & Co., Ltd. | Carbamoylpyridone derivatives having inhibitory activity against HIV integrase |
| UA87884C2 (uk) * | 2004-12-03 | 2009-08-25 | Мерк Энд Ко., Инк. | Безводна кристалічна калієва сіль інгібітора віл-інтегрази |
| WO2009119534A1 (ja) * | 2008-03-26 | 2009-10-01 | 第一三共株式会社 | 新規テトラヒドロイソキノリン誘導体 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8927913D0 (en) | 1989-12-11 | 1990-02-14 | Hoffmann La Roche | Amino acid derivatives |
| MX9308016A (es) * | 1992-12-22 | 1994-08-31 | Lilly Co Eli | Compuestos inhibidores de la proteasa del virus de la inmunodeficiencia humana, procedimiento para su preparacion y formulacion farmaceutica que los contiene. |
-
2000
- 2000-11-22 GB GBGB0028483.6A patent/GB0028483D0/en not_active Ceased
-
2001
- 2001-11-12 SK SK760-2003A patent/SK7602003A3/sk unknown
- 2001-11-12 HU HU0303007A patent/HUP0303007A2/hu unknown
- 2001-11-12 KR KR10-2003-7006907A patent/KR20030060953A/ko not_active Application Discontinuation
- 2001-11-12 NZ NZ525550A patent/NZ525550A/en unknown
- 2001-11-12 MX MXPA03004534A patent/MXPA03004534A/es active IP Right Grant
- 2001-11-12 CZ CZ20031667A patent/CZ20031667A3/cs unknown
- 2001-11-12 RU RU2003117468/04A patent/RU2265016C2/ru not_active IP Right Cessation
- 2001-11-12 AU AU2002229546A patent/AU2002229546B2/en not_active Ceased
- 2001-11-12 CA CA002428459A patent/CA2428459A1/en not_active Abandoned
- 2001-11-12 BR BR0115566-0A patent/BR0115566A/pt not_active IP Right Cessation
- 2001-11-12 EP EP01990405A patent/EP1339692A1/en not_active Withdrawn
- 2001-11-12 PL PL01366704A patent/PL366704A1/xx not_active Application Discontinuation
- 2001-11-12 WO PCT/EP2001/013068 patent/WO2002042277A1/en active IP Right Grant
- 2001-11-12 CN CNA018192890A patent/CN1476436A/zh active Pending
- 2001-11-12 IL IL15557301A patent/IL155573A0/xx unknown
- 2001-11-12 JP JP2002544412A patent/JP2004520283A/ja active Pending
- 2001-11-12 AU AU2954602A patent/AU2954602A/xx active Pending
- 2001-11-20 US US09/999,082 patent/US6472404B1/en not_active Expired - Fee Related
- 2001-11-21 GT GT200100233A patent/GT200100233A/es unknown
- 2001-11-21 AR ARP010105431A patent/AR031763A1/es unknown
- 2001-11-21 PA PA20018533401A patent/PA8533401A1/es unknown
- 2001-11-21 UY UY27033A patent/UY27033A1/es not_active Application Discontinuation
- 2001-11-22 PE PE2001001170A patent/PE20020610A1/es not_active Application Discontinuation
-
2003
- 2003-05-21 EC EC2003004618A patent/ECSP034618A/es unknown
- 2003-05-21 NO NO20032290A patent/NO20032290D0/no unknown
- 2003-05-22 BG BG107839A patent/BG107839A/bg unknown
- 2003-05-22 MA MA27172A patent/MA26966A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20030060953A (ko) | 2003-07-16 |
| AR031763A1 (es) | 2003-10-01 |
| NO20032290L (no) | 2003-05-21 |
| PL366704A1 (en) | 2005-02-07 |
| US6472404B1 (en) | 2002-10-29 |
| BR0115566A (pt) | 2003-09-30 |
| UY27033A1 (es) | 2002-06-20 |
| PE20020610A1 (es) | 2002-07-13 |
| RU2003117468A (ru) | 2005-01-27 |
| AU2002229546B2 (en) | 2006-05-04 |
| GB0028483D0 (en) | 2001-01-10 |
| BG107839A (bg) | 2004-06-30 |
| AU2954602A (en) | 2002-06-03 |
| CA2428459A1 (en) | 2002-05-30 |
| ECSP034618A (es) | 2003-06-25 |
| SK7602003A3 (en) | 2004-01-08 |
| WO2002042277A1 (en) | 2002-05-30 |
| NO20032290D0 (no) | 2003-05-21 |
| MA26966A1 (fr) | 2004-12-20 |
| RU2265016C2 (ru) | 2005-11-27 |
| EP1339692A1 (en) | 2003-09-03 |
| CN1476436A (zh) | 2004-02-18 |
| HUP0303007A2 (hu) | 2003-12-29 |
| PA8533401A1 (es) | 2002-10-31 |
| NZ525550A (en) | 2004-11-26 |
| GT200100233A (es) | 2002-07-04 |
| JP2004520283A (ja) | 2004-07-08 |
| IL155573A0 (en) | 2003-11-23 |
| CZ20031667A3 (cs) | 2004-01-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MXPA03005838A (es) | Inhibidores de antigenos de aparicion muy tardia-4. | |
| ZA200109890B (en) | Metalloprotease inhibitors. | |
| IL150964A0 (en) | Protease inhibitors | |
| IL155202A0 (en) | Biaryl compounds as serine protease inhibitors | |
| ZA200204397B (en) | Nitrile derivatives as cathepsin K inhibitors. | |
| ZA992447B (en) | Quinoxalinones as serine protease inhibitors. | |
| HK1054034A1 (en) | Substituted pyrrolopyridinone derivatives useful as phosphodiesterase inhibitors. | |
| MXPA03007310A (es) | Derivados de ftalazinona piperidino como inhibidores pde4. | |
| ZA992448B (en) | Quinoxalinones as serine protease inhibitors. | |
| AP2003002856A0 (en) | Broadspectrum 2-(substitutted-amino)-benzothiazolesulphonamide HIV protease inhibitors. | |
| MXPA03009361A (es) | Compuestos de urea utilies como agentes anti-inflamatorios. | |
| AU2001247589A1 (en) | Non-amidine containing protease inhibitors | |
| MXPA03005673A (es) | Inhibidores de 8-arilquinolin-fosfodiesterasa-4-substituidos. | |
| AU6989501A (en) | Hiv integrase inhibitors | |
| PL360508A1 (en) | Protease inhibitors | |
| IL151087A0 (en) | Protease inhibitors | |
| MXPA03004534A (es) | Compuestos novedosos para su uso como inhibidores de la proteasa del virus de inmunodeficiencia humana (vih). | |
| AU2001268303A1 (en) | Hepatitis c protease exosite for inhibitor design | |
| EP1401453A4 (en) | PROTEASE INHIBITORS | |
| MXPA03004542A (es) | Inhibidores de proteasa. | |
| AU2003287325A8 (en) | N-cycloalkylglycines as hiv protease inhibitors | |
| ZA200207478B (en) | Protease inhibitors. | |
| AU2002255485A8 (en) | Hiv/fiv protease inhibitors | |
| AU2001228648A1 (en) | Clavams as protease inhibitors | |
| ZA200003398B (en) | Inhibitors. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |