GB0028483D0 - Hydroxyethylamine HIV protease inhibitors - Google Patents

Hydroxyethylamine HIV protease inhibitors

Info

Publication number
GB0028483D0
GB0028483D0 GBGB0028483.6A GB0028483A GB0028483D0 GB 0028483 D0 GB0028483 D0 GB 0028483D0 GB 0028483 A GB0028483 A GB 0028483A GB 0028483 D0 GB0028483 D0 GB 0028483D0
Authority
GB
United Kingdom
Prior art keywords
hydroxyethylamine
protease inhibitors
hiv protease
hiv
inhibitors
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB0028483.6A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Priority to GBGB0028483.6A priority Critical patent/GB0028483D0/en
Publication of GB0028483D0 publication Critical patent/GB0028483D0/en
Priority to CZ20031667A priority patent/CZ20031667A3/cs
Priority to AU2954602A priority patent/AU2954602A/xx
Priority to KR10-2003-7006907A priority patent/KR20030060953A/ko
Priority to HU0303007A priority patent/HUP0303007A2/hu
Priority to CA002428459A priority patent/CA2428459A1/en
Priority to EP01990405A priority patent/EP1339692A1/en
Priority to IL15557301A priority patent/IL155573A0/xx
Priority to PL01366704A priority patent/PL366704A1/xx
Priority to JP2002544412A priority patent/JP2004520283A/ja
Priority to AU2002229546A priority patent/AU2002229546B2/en
Priority to NZ525550A priority patent/NZ525550A/en
Priority to CNA018192890A priority patent/CN1476436A/zh
Priority to MXPA03004534A priority patent/MXPA03004534A/es
Priority to PCT/EP2001/013068 priority patent/WO2002042277A1/en
Priority to BR0115566-0A priority patent/BR0115566A/pt
Priority to RU2003117468/04A priority patent/RU2265016C2/ru
Priority to SK760-2003A priority patent/SK7602003A3/sk
Priority to US09/999,082 priority patent/US6472404B1/en
Priority to PA20018533401A priority patent/PA8533401A1/es
Priority to GT200100233A priority patent/GT200100233A/es
Priority to ARP010105431A priority patent/AR031763A1/es
Priority to UY27033A priority patent/UY27033A1/es
Priority to PE2001001170A priority patent/PE20020610A1/es
Priority to NO20032290A priority patent/NO20032290D0/no
Priority to EC2003004618A priority patent/ECSP034618A/es
Priority to BG107839A priority patent/BG107839A/bg
Priority to MA27172A priority patent/MA26966A1/fr
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
GBGB0028483.6A 2000-11-22 2000-11-22 Hydroxyethylamine HIV protease inhibitors Ceased GB0028483D0 (en)

Priority Applications (28)

Application Number Priority Date Filing Date Title
GBGB0028483.6A GB0028483D0 (en) 2000-11-22 2000-11-22 Hydroxyethylamine HIV protease inhibitors
SK760-2003A SK7602003A3 (en) 2000-11-22 2001-11-12 Novel compounds for use as HIV protease inhibitors
CNA018192890A CN1476436A (zh) 2000-11-22 2001-11-12 用作hiv蛋白酶抑制剂的新化合物
PCT/EP2001/013068 WO2002042277A1 (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors
KR10-2003-7006907A KR20030060953A (ko) 2000-11-22 2001-11-12 Hiv 프로테아제 억제제로서 사용하기 위한 신규한 화합물
HU0303007A HUP0303007A2 (hu) 2000-11-22 2001-11-12 Új vegyületek HIV proteáz inhibitorként történő felhasználásra és a vegyületeket tartalmazó gyógyszerkészítmények
CA002428459A CA2428459A1 (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors
EP01990405A EP1339692A1 (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors
IL15557301A IL155573A0 (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors
PL01366704A PL366704A1 (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors
JP2002544412A JP2004520283A (ja) 2000-11-22 2001-11-12 Hivプロテアーゼインヒビターとして使用するための新規な化合物
AU2002229546A AU2002229546B2 (en) 2000-11-22 2001-11-12 Novel compounds for use as HIV protease inhibitors
NZ525550A NZ525550A (en) 2000-11-22 2001-11-12 Novel compounds for use as HIV protease inhibitors
CZ20031667A CZ20031667A3 (cs) 2000-11-22 2001-11-12 Nové sloučeniny použitelné jako inhibitory HIV proteázy
MXPA03004534A MXPA03004534A (es) 2000-11-22 2001-11-12 Compuestos novedosos para su uso como inhibidores de la proteasa del virus de inmunodeficiencia humana (vih).
AU2954602A AU2954602A (en) 2000-11-22 2001-11-12 Novel compounds for use as hiv protease inhibitors
BR0115566-0A BR0115566A (pt) 2000-11-22 2001-11-12 Compostos para emprego como inibidores de protease de hiv
RU2003117468/04A RU2265016C2 (ru) 2000-11-22 2001-11-12 Изохинолинкарбоксамиды и лекарственное средство на их основе для применения в качестве ингибиторов протеазы вич
US09/999,082 US6472404B1 (en) 2000-11-22 2001-11-20 HIV protease inhibitors
PA20018533401A PA8533401A1 (es) 2000-11-22 2001-11-21 Inhibidores de la proteasa hidroxietilamina del vih
GT200100233A GT200100233A (es) 2000-11-22 2001-11-21 Nuevos inhibidores de la proteasa de vih.
ARP010105431A AR031763A1 (es) 2000-11-22 2001-11-21 Nuevos compuestos para el uso como inhibidores de proteasas hiv
UY27033A UY27033A1 (es) 2000-11-22 2001-11-21 Nuevos compuestos para su uso como inhibidores de la proteasa de vih
PE2001001170A PE20020610A1 (es) 2000-11-22 2001-11-22 Compuestos hidroxietilamina tripeptidos mimeticos como inhibidores de la aspartil proteasa de vih
NO20032290A NO20032290D0 (no) 2000-11-22 2003-05-21 Nye forbindelser for anvendelse som HIV-protease-inhibitorer
EC2003004618A ECSP034618A (es) 2000-11-22 2003-05-21 Nuevos compuestos para usarse como inhibidores de proteasa vih
BG107839A BG107839A (bg) 2000-11-22 2003-05-22 Нови съединения за използване като hiv протеазни инхибитори
MA27172A MA26966A1 (fr) 2000-11-22 2003-05-22 Nouveaux composes utilisables en tant qu'inhibiteurs de protease hiv

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0028483.6A GB0028483D0 (en) 2000-11-22 2000-11-22 Hydroxyethylamine HIV protease inhibitors

Publications (1)

Publication Number Publication Date
GB0028483D0 true GB0028483D0 (en) 2001-01-10

Family

ID=9903670

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB0028483.6A Ceased GB0028483D0 (en) 2000-11-22 2000-11-22 Hydroxyethylamine HIV protease inhibitors

Country Status (27)

Country Link
US (1) US6472404B1 (es)
EP (1) EP1339692A1 (es)
JP (1) JP2004520283A (es)
KR (1) KR20030060953A (es)
CN (1) CN1476436A (es)
AR (1) AR031763A1 (es)
AU (2) AU2954602A (es)
BG (1) BG107839A (es)
BR (1) BR0115566A (es)
CA (1) CA2428459A1 (es)
CZ (1) CZ20031667A3 (es)
EC (1) ECSP034618A (es)
GB (1) GB0028483D0 (es)
GT (1) GT200100233A (es)
HU (1) HUP0303007A2 (es)
IL (1) IL155573A0 (es)
MA (1) MA26966A1 (es)
MX (1) MXPA03004534A (es)
NO (1) NO20032290D0 (es)
NZ (1) NZ525550A (es)
PA (1) PA8533401A1 (es)
PE (1) PE20020610A1 (es)
PL (1) PL366704A1 (es)
RU (1) RU2265016C2 (es)
SK (1) SK7602003A3 (es)
UY (1) UY27033A1 (es)
WO (1) WO2002042277A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101014572B (zh) * 2004-09-15 2011-07-06 盐野义制药株式会社 具有hiv整合酶抑制活性的氨基甲酰基吡啶酮衍生物
UA87884C2 (uk) * 2004-12-03 2009-08-25 Мерк Энд Ко., Инк. Безводна кристалічна калієва сіль інгібітора віл-інтегрази
MY161992A (en) * 2008-03-26 2017-05-31 Daiichi Sankyo Co Ltd Novel tetrahydroisoquinoline derivative

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8927913D0 (en) 1989-12-11 1990-02-14 Hoffmann La Roche Amino acid derivatives
MX9308016A (es) * 1992-12-22 1994-08-31 Lilly Co Eli Compuestos inhibidores de la proteasa del virus de la inmunodeficiencia humana, procedimiento para su preparacion y formulacion farmaceutica que los contiene.

Also Published As

Publication number Publication date
NO20032290L (no) 2003-05-21
BG107839A (bg) 2004-06-30
NO20032290D0 (no) 2003-05-21
RU2003117468A (ru) 2005-01-27
BR0115566A (pt) 2003-09-30
MXPA03004534A (es) 2003-09-10
RU2265016C2 (ru) 2005-11-27
GT200100233A (es) 2002-07-04
EP1339692A1 (en) 2003-09-03
AR031763A1 (es) 2003-10-01
CZ20031667A3 (cs) 2004-01-14
PA8533401A1 (es) 2002-10-31
WO2002042277A1 (en) 2002-05-30
CA2428459A1 (en) 2002-05-30
SK7602003A3 (en) 2004-01-08
HUP0303007A2 (hu) 2003-12-29
MA26966A1 (fr) 2004-12-20
KR20030060953A (ko) 2003-07-16
AU2954602A (en) 2002-06-03
PE20020610A1 (es) 2002-07-13
ECSP034618A (es) 2003-06-25
JP2004520283A (ja) 2004-07-08
CN1476436A (zh) 2004-02-18
PL366704A1 (en) 2005-02-07
US6472404B1 (en) 2002-10-29
NZ525550A (en) 2004-11-26
IL155573A0 (en) 2003-11-23
AU2002229546B2 (en) 2006-05-04
UY27033A1 (es) 2002-06-20

Similar Documents

Publication Publication Date Title
AU4344101A (en) Protease inhibitors
GB0125445D0 (en) Protease Inhibitors
AU2001247589A1 (en) Non-amidine containing protease inhibitors
IL153421A0 (en) Protease inhibitors
IL151087A0 (en) Protease inhibitors
AU2002360673A8 (en) Gp41 inhibitor
EP1229912A4 (en) PROTEASE INHIBITORS
EP1229914A4 (en) PROTEASE INHIBITORS
EP1173429A4 (en) PROTEASE INHIBITORS
EP1229911A4 (en) PROTEASE INHIBITORS
EP1161237A4 (en) PROTEASE INHIBITORS
EP1401453A4 (en) PROTEASE INHIBITORS
IL155961A0 (en) Cysteine protease inhibitors
GB0028483D0 (en) Hydroxyethylamine HIV protease inhibitors
IL155997A0 (en) Protease inhibitors
GB0123467D0 (en) Carbocyclic HIV Protease inhibitors
AU6407701A (en) Serine protease inhibitors
AU2003287325A8 (en) N-cycloalkylglycines as hiv protease inhibitors
GB0009123D0 (en) Protease inhibitor
AU2002255485A8 (en) Hiv/fiv protease inhibitors
ZA200207478B (en) Protease inhibitors.
AU2001296247A1 (en) Cysteine protease inhibitors
IL160626A0 (en) Antiviral protease inhibitors
AU2001244658A1 (en) Gamma-secretase-like protease inhibitors
GB0028863D0 (en) Protease

Legal Events

Date Code Title Description
AT Applications terminated before publication under section 16(1)