NO171501C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive 2-metoksymetylpenem-derivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive 2-metoksymetylpenem-derivater

Info

Publication number
NO171501C
NO171501C NO882528A NO882528A NO171501C NO 171501 C NO171501 C NO 171501C NO 882528 A NO882528 A NO 882528A NO 882528 A NO882528 A NO 882528A NO 171501 C NO171501 C NO 171501C
Authority
NO
Norway
Prior art keywords
methoxymethylpenem
derivatives
preparation
therapeutic active
analogy procedure
Prior art date
Application number
NO882528A
Other languages
English (en)
Norwegian (no)
Other versions
NO882528L (no
NO882528D0 (no
NO171501B (no
Inventor
Marco Alpegiani
Giovanni Franceschi
Ettore Perrone
Franco Zarini
Constantino Della Bruna
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of NO882528D0 publication Critical patent/NO882528D0/no
Publication of NO882528L publication Critical patent/NO882528L/no
Publication of NO171501B publication Critical patent/NO171501B/no
Publication of NO171501C publication Critical patent/NO171501C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
NO882528A 1987-06-10 1988-06-08 Analogifremgangsmaate ved fremstilling av terapeutisk aktive 2-metoksymetylpenem-derivater NO171501C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB878713515A GB8713515D0 (en) 1987-06-10 1987-06-10 Methoxymethyl compounds

Publications (4)

Publication Number Publication Date
NO882528D0 NO882528D0 (no) 1988-06-08
NO882528L NO882528L (no) 1988-12-12
NO171501B NO171501B (no) 1992-12-14
NO171501C true NO171501C (no) 1993-03-24

Family

ID=10618657

Family Applications (1)

Application Number Title Priority Date Filing Date
NO882528A NO171501C (no) 1987-06-10 1988-06-08 Analogifremgangsmaate ved fremstilling av terapeutisk aktive 2-metoksymetylpenem-derivater

Country Status (30)

Country Link
US (1) US4952577A (it)
EP (1) EP0295100B1 (it)
JP (1) JP2547341B2 (it)
KR (1) KR890000495A (it)
CN (2) CN1056420A (it)
AT (1) AT395590B (it)
AU (2) AU609488B2 (it)
CA (1) CA1300604C (it)
CH (2) CH682324A5 (it)
CS (2) CS268197B2 (it)
DE (1) DE3851470T2 (it)
DK (1) DK313788A (it)
ES (1) ES2009935A6 (it)
FI (1) FI89490C (it)
FR (1) FR2616434B1 (it)
GB (2) GB8713515D0 (it)
HK (1) HK65291A (it)
HU (1) HU198943B (it)
IE (1) IE61905B1 (it)
IL (1) IL86640A (it)
IT (1) IT1221792B (it)
MY (1) MY103733A (it)
NO (1) NO171501C (it)
NZ (1) NZ224923A (it)
PH (1) PH26311A (it)
PT (1) PT87679B (it)
SG (1) SG60791G (it)
SU (1) SU1586517A3 (it)
YU (1) YU46914B (it)
ZA (1) ZA884081B (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8915392D0 (en) * 1989-07-05 1989-08-23 Erba Carlo Spa Process for penems
US5416208A (en) * 1989-07-05 1995-05-16 Farmitalia Carlo Erba S R L Process for penems
DE69133273T2 (de) * 1990-08-20 2004-05-13 Daiichi Suntory Pharma Co., Ltd. Antibakterielle Penem-Ester-Derivate
US5506225A (en) * 1990-08-20 1996-04-09 Suntory Limited Antibacterial penem compounds
US5703068A (en) * 1990-08-20 1997-12-30 Suntory Limited Penem compounds
GB9210371D0 (en) * 1992-05-14 1992-07-01 Erba Carlo Spa Hydroxy protecting group removal in penems
US5399679A (en) * 1992-06-16 1995-03-21 Farmitalia Carlo Erba S.R.L. (1'R,3S,4R)4-acylthio azetidinones
GB9216102D0 (en) * 1992-07-29 1992-09-09 Smithkline Beecham Plc Pharmaceutical substances
PE20080940A1 (es) * 2006-06-28 2008-07-09 Pfizer Prod Inc Profarmacos de penem

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
EP0042026B1 (de) * 1978-02-02 1986-01-08 Ciba-Geigy Ag 3,4-Disubstituierte Azetidin-2-onverbindungen und Verfahren zu ihrer Herstellung
JPS5625110A (en) * 1978-12-18 1981-03-10 Bristol Myers Co Antibacterial
US4272437A (en) * 1978-12-18 1981-06-09 Bristol-Myers Company Antibacterial agents, and 4-thio azetidinone intermediates
US4482565A (en) * 1980-02-22 1984-11-13 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
US4558042A (en) * 1981-05-06 1985-12-10 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
AT379399B (de) * 1981-12-11 1985-12-27 Erba Farmitalia Verfahren zur herstellung von optisch aktiven penemen
GB8321677D0 (en) * 1983-08-11 1983-09-14 Erba Farmitalia Preparation of penems
JPH075463B2 (ja) * 1985-03-09 1995-01-25 サントリー株式会社 抗菌剤
EP0201459A1 (de) * 1985-05-06 1986-11-12 Ciba-Geigy Ag Acylaminomethylpenemverbindungen, ihre Herstellung und sie enthaltende pharmazeutische Präparate
GB2166435B (en) * 1985-05-09 1988-08-24 Erba Carlo Spa Penams, their preparation and their use
EP0233155A1 (de) * 1986-02-14 1987-08-19 Ciba-Geigy Ag Aminoacyloxymethyl-Verbindungen
GB8624686D0 (en) * 1986-10-15 1986-11-19 Erba Farmitalia Preparing penems
JPH01207387A (ja) * 1988-02-15 1989-08-21 Res Assoc Util Of Light Oil 炭化水素の製造方法

Also Published As

Publication number Publication date
CN1030079A (zh) 1989-01-04
CS268197B2 (en) 1990-03-14
IT8820868A0 (it) 1988-06-06
CA1300604C (en) 1992-05-12
IE881687L (en) 1988-12-10
PT87679B (pt) 1992-10-30
CS414991A3 (en) 1992-06-17
NO882528L (no) 1988-12-12
JPS63316784A (ja) 1988-12-26
SG60791G (en) 1991-08-23
PH26311A (en) 1992-04-29
CN1025032C (zh) 1994-06-15
GB2205831B (en) 1991-03-27
HK65291A (en) 1991-08-23
ZA884081B (en) 1989-02-22
DE3851470T2 (de) 1995-02-09
DK313788D0 (da) 1988-06-09
GB8813622D0 (en) 1988-07-13
AU8146191A (en) 1991-10-24
GB2205831A (en) 1988-12-21
ATA146488A (de) 1992-06-15
FI89490C (fi) 1993-10-11
IE61905B1 (en) 1994-11-30
FR2616434A1 (fr) 1988-12-16
NO882528D0 (no) 1988-06-08
ES2009935A6 (es) 1989-10-16
SU1586517A3 (ru) 1990-08-15
IT1221792B (it) 1990-07-12
CS397588A2 (en) 1989-04-14
GB8713515D0 (en) 1987-07-15
FR2616434B1 (fr) 1994-04-08
FI882696A0 (fi) 1988-06-08
KR890000495A (ko) 1989-03-15
US4952577A (en) 1990-08-28
MY103733A (en) 1993-09-30
AU1746188A (en) 1988-12-15
EP0295100A1 (en) 1988-12-14
AU609488B2 (en) 1991-05-02
AT395590B (de) 1993-01-25
YU112188A (en) 1989-06-30
CH682324A5 (it) 1993-08-31
IL86640A0 (en) 1988-11-30
NZ224923A (en) 1989-08-29
CH678058A5 (it) 1991-07-31
IL86640A (en) 1993-01-31
EP0295100B1 (en) 1994-09-14
CN1056420A (zh) 1991-11-27
DK313788A (da) 1988-12-11
JP2547341B2 (ja) 1996-10-23
DE3851470D1 (de) 1994-10-20
PT87679A (pt) 1988-07-01
FI89490B (fi) 1993-06-30
HUT47295A (en) 1989-02-28
YU46914B (sh) 1994-06-24
NO171501B (no) 1992-12-14
HU198943B (en) 1989-12-28
FI882696A (fi) 1988-12-11

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