NO173185C - Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxalinforbindelser - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxalinforbindelser

Info

Publication number
NO173185C
NO173185C NO892204A NO892204A NO173185C NO 173185 C NO173185 C NO 173185C NO 892204 A NO892204 A NO 892204A NO 892204 A NO892204 A NO 892204A NO 173185 C NO173185 C NO 173185C
Authority
NO
Norway
Prior art keywords
imidazokinoxal
compounds
preparation
therapeutic active
analogy procedure
Prior art date
Application number
NO892204A
Other languages
English (en)
Other versions
NO892204L (no
NO173185B (no
NO892204D0 (no
Inventor
Holger Claus Hansen
Frank Waetjen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DK297188A external-priority patent/DK297188D0/da
Priority claimed from DK625988A external-priority patent/DK625988D0/da
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of NO892204D0 publication Critical patent/NO892204D0/no
Publication of NO892204L publication Critical patent/NO892204L/no
Publication of NO173185B publication Critical patent/NO173185B/no
Publication of NO173185C publication Critical patent/NO173185C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO892204A 1988-06-01 1989-05-31 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxalinforbindelser NO173185C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DK297188A DK297188D0 (da) 1988-06-01 1988-06-01 Imidazoquinoxalinforbindelser, deres fremstilling og anvendelse
DK625988A DK625988D0 (da) 1988-11-10 1988-11-10 Imidazoquinoxalinforbindelser, deres fremstilling og anvendelse

Publications (4)

Publication Number Publication Date
NO892204D0 NO892204D0 (no) 1989-05-31
NO892204L NO892204L (no) 1989-12-04
NO173185B NO173185B (no) 1993-08-02
NO173185C true NO173185C (no) 1993-11-10

Family

ID=26066829

Family Applications (1)

Application Number Title Priority Date Filing Date
NO892204A NO173185C (no) 1988-06-01 1989-05-31 Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazokinoxalinforbindelser

Country Status (12)

Country Link
US (1) US5075304A (no)
EP (1) EP0344943A1 (no)
JP (1) JPH0225486A (no)
KR (1) KR900018102A (no)
AU (1) AU627181B2 (no)
CA (1) CA1315786C (no)
FI (1) FI92203C (no)
IL (1) IL90315A0 (no)
NO (1) NO173185C (no)
NZ (1) NZ229346A (no)
PH (1) PH26379A (no)
PT (1) PT90721B (no)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
DK626288D0 (da) * 1988-11-10 1988-11-10 Ferrosan As Kemisk proces til fremstilling af imidazoquinoxaliner og mellemprodukter til brug i processen
US5276028A (en) * 1990-06-22 1994-01-04 Nordisk A/S Imidazoquinoxaline compounds
DK151890D0 (da) * 1990-06-22 1990-06-22 Ferrosan As Heterocykliske forbindelser deres fremstilling og brug
US5371080A (en) * 1990-06-22 1994-12-06 Novo Nordisk A/S Imidazoquinazoline compounds and their use
WO1992004350A1 (en) * 1990-09-04 1992-03-19 The Upjohn Company Oxygenated quinoxalines
CA2110942A1 (en) * 1991-06-14 1992-12-23 Pharmacia & Upjohn Company Llc Imidazo¬1,5-a|quinoxalines
US5182386A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands
US5597920A (en) * 1992-04-30 1997-01-28 Neurogen Corporation Gabaa receptor subtypes and methods for screening drug compounds using imidazoquinoxalines and pyrrolopyrimidines to bind to gabaa receptor subtypes
DE4228095A1 (de) * 1992-08-24 1994-03-03 Asta Medica Ag Neue 4,5-Dihydro-4-oxo-pyrrolo[1,2-a]chinoxaline und entsprechende Aza-analoga und Verfahren zu deren Herstellung
IL109397A0 (en) * 1993-04-28 1994-07-31 Schering Ag Quinoxalinedione derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
US5792766A (en) * 1996-03-13 1998-08-11 Neurogen Corporation Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands
RU2750151C2 (ru) 2015-11-20 2021-06-22 Форма Терапьютикс, Инк. Гипоксантины в качестве ингибиторов убиквитин-специфической протеазы 1

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440929A (en) * 1981-07-16 1984-04-03 Usv Pharmaceutical Corporation Imidazoquinoxaline compounds
DK476885D0 (da) * 1985-10-17 1985-10-17 Ferrosan As Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf
DK155524C (da) * 1987-03-18 1989-09-11 Ferrosan As Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse
DK160876C (da) * 1987-12-08 1991-10-14 Novo Nordisk As Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar

Also Published As

Publication number Publication date
PT90721A (pt) 1989-12-29
FI92203C (fi) 1994-10-10
NO892204L (no) 1989-12-04
FI892684L (fi) 1989-12-02
AU3517489A (en) 1989-12-07
AU627181B2 (en) 1992-08-20
KR900018102A (ko) 1990-12-20
FI92203B (fi) 1994-06-30
US5075304A (en) 1991-12-24
JPH0225486A (ja) 1990-01-26
NO173185B (no) 1993-08-02
CA1315786C (en) 1993-04-06
NO892204D0 (no) 1989-05-31
NZ229346A (en) 1991-11-26
EP0344943A1 (en) 1989-12-06
PT90721B (pt) 1994-11-30
IL90315A0 (en) 1989-12-15
PH26379A (en) 1992-06-01
FI892684A0 (fi) 1989-06-01

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