NO150158C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive 6,7-dimetoksyquinazolinderivater - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive 6,7-dimetoksyquinazolinderivater

Info

Publication number
NO150158C
NO150158C NO783705A NO783705A NO150158C NO 150158 C NO150158 C NO 150158C NO 783705 A NO783705 A NO 783705A NO 783705 A NO783705 A NO 783705A NO 150158 C NO150158 C NO 150158C
Authority
NO
Norway
Prior art keywords
dimetoxyquinazoline
derivatives
preparation
therapeutic active
analogy procedure
Prior art date
Application number
NO783705A
Other languages
English (en)
Norwegian (no)
Other versions
NO150158B (no
NO783705L (no
Inventor
Simon Fraser Campbell
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO783705L publication Critical patent/NO783705L/no
Publication of NO150158B publication Critical patent/NO150158B/no
Publication of NO150158C publication Critical patent/NO150158C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D319/00Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/101,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/141,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/161,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/201,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring with substituents attached to the hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NO783705A 1977-11-05 1978-11-03 Analogifremgangsmaate ved fremstilling av terapeutisk aktive 6,7-dimetoksyquinazolinderivater NO150158C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4612877 1977-11-05

Publications (3)

Publication Number Publication Date
NO783705L NO783705L (no) 1979-05-08
NO150158B NO150158B (no) 1984-05-21
NO150158C true NO150158C (no) 1984-08-29

Family

ID=10439957

Family Applications (1)

Application Number Title Priority Date Filing Date
NO783705A NO150158C (no) 1977-11-05 1978-11-03 Analogifremgangsmaate ved fremstilling av terapeutisk aktive 6,7-dimetoksyquinazolinderivater

Country Status (36)

Country Link
JP (1) JPS5498792A (fi)
AR (2) AR219562A1 (fi)
AT (1) AT365186B (fi)
AU (1) AU509329B2 (fi)
BE (1) BE871771A (fi)
CA (1) CA1088059A (fi)
CH (1) CH643255A5 (fi)
CS (2) CS207671B2 (fi)
DD (1) DD139850A5 (fi)
DE (1) DE2847623C2 (fi)
DK (1) DK154082C (fi)
EG (1) EG13594A (fi)
ES (2) ES474805A1 (fi)
FI (1) FI64366C (fi)
FR (1) FR2407929A1 (fi)
GR (1) GR81514B (fi)
HK (1) HK94284A (fi)
HU (1) HU176306B (fi)
IE (1) IE47888B1 (fi)
IL (1) IL55857A (fi)
IN (1) IN148828B (fi)
IT (1) IT1100919B (fi)
KE (1) KE3350A (fi)
LU (2) LU80470A1 (fi)
MY (1) MY8500286A (fi)
NL (2) NL174549C (fi)
NO (1) NO150158C (fi)
NZ (1) NZ188813A (fi)
PH (1) PH13966A (fi)
PL (2) PL119419B1 (fi)
PT (1) PT68735A (fi)
SE (1) SE437518B (fi)
SU (1) SU816403A3 (fi)
UA (1) UA8324A1 (fi)
YU (2) YU40204B (fi)
ZA (1) ZA786184B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1986002644A1 (en) * 1984-11-01 1986-05-09 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1985002617A1 (en) * 1983-12-14 1985-06-20 Takeda Chemical Industries. Ltd. 1,5-benzoxathiepin derivatives and process for their preparation
WO1985004658A1 (en) * 1984-04-04 1985-10-24 Takeda Chemical Industries, Ltd. 1,5-benzoxathiepine derivatives and their preparation
EP0849264A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von doxazosinmesylat (Form I)
EP0849265A1 (de) * 1996-12-20 1998-06-24 HEUMANN PHARMA GmbH Neue polymorphe Form von Doxazosin-Mesylat (Form II)
ES2282997T3 (es) * 1996-12-20 2007-10-16 Heumann Pcs Gmbh Nueva forma polimorfa de mesilato e doxazosina (forma iii).
TW448155B (en) * 1999-03-29 2001-08-01 Dev Center Biotechnology Method for producing amide compounds and quinazolin derivatives
EP1403263B1 (en) * 2002-09-27 2005-06-22 Council of Scientific and Industrial Research Process for the preparation of N-(2,3-dihydrobenzo 1,4 dioxin-2-carbonyl) piperazine

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3635979A (en) * 1969-09-29 1972-01-18 Pfizer Certain 6- and/or 7-alkoxy-substituted-2 4-bis(disubstituted amino) quinazolines
US3669968A (en) * 1970-05-21 1972-06-13 Pfizer Trialkoxy quinazolines

Also Published As

Publication number Publication date
CA1088059A (en) 1980-10-21
GR81514B (fi) 1984-12-11
FR2407929A1 (fr) 1979-06-01
NL930062I2 (nl) 1993-11-16
NL7810909A (nl) 1979-05-08
CS354491A3 (en) 1992-06-17
NL174549C (nl) 1984-07-02
ZA786184B (en) 1979-10-31
YU40204B (en) 1985-08-31
DK428678A (da) 1979-05-06
MY8500286A (en) 1985-12-31
HK94284A (en) 1984-12-07
CS207671B2 (en) 1981-08-31
ES474805A1 (es) 1980-01-16
CH643255A5 (en) 1984-05-30
FI783347A (fi) 1979-05-06
PH13966A (en) 1980-11-12
SE437518B (sv) 1985-03-04
EG13594A (en) 1982-03-31
YU38683A (en) 1983-06-30
AR223015A1 (es) 1981-07-15
SU816403A3 (ru) 1981-03-23
IL55857A0 (en) 1979-01-31
DD139850A5 (de) 1980-01-23
NL930062I1 (nl) 1993-09-01
DK154082B (da) 1988-10-10
ATA784378A (de) 1981-05-15
YU255378A (en) 1983-06-30
LU88331I2 (fr) 1994-05-04
KE3350A (en) 1983-12-16
AR219562A1 (es) 1980-08-29
NL174549B (nl) 1984-02-01
NO150158B (no) 1984-05-21
IE782179L (en) 1979-05-05
IT1100919B (it) 1985-09-28
HU176306B (en) 1981-01-28
PL119419B1 (en) 1981-12-31
IN148828B (fi) 1981-06-27
NO783705L (no) 1979-05-08
ES8308559A1 (es) 1980-07-16
UA8324A1 (uk) 1996-03-29
DE2847623C2 (de) 1983-06-01
IT7829434A0 (it) 1978-11-03
AU4132278A (en) 1979-05-17
YU40419B (en) 1985-12-31
AT365186B (de) 1981-12-28
PL119586B1 (en) 1982-01-30
NZ188813A (en) 1980-10-08
ES480121A0 (es) 1980-07-16
FI64366B (fi) 1983-07-29
SE7811382L (sv) 1979-05-06
FI64366C (fi) 1983-11-10
PT68735A (en) 1978-12-01
JPS5625233B2 (fi) 1981-06-11
DK154082C (da) 1989-02-27
IE47888B1 (en) 1984-07-11
DE2847623A1 (de) 1979-05-23
JPS5498792A (en) 1979-08-03
BE871771A (fr) 1979-05-03
PL210681A1 (fi) 1979-11-05
IL55857A (en) 1982-07-30
AU509329B2 (en) 1980-05-08
FR2407929B1 (fi) 1981-02-27
LU80470A1 (fr) 1980-06-05

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