NL8500485A - Voorlopers van antiinflammatoire oxicamen. - Google Patents

Voorlopers van antiinflammatoire oxicamen. Download PDF

Info

Publication number
NL8500485A
NL8500485A NL8500485A NL8500485A NL8500485A NL 8500485 A NL8500485 A NL 8500485A NL 8500485 A NL8500485 A NL 8500485A NL 8500485 A NL8500485 A NL 8500485A NL 8500485 A NL8500485 A NL 8500485A
Authority
NL
Netherlands
Prior art keywords
dioxide
methyl
benzothiazine
compound according
carboxamide
Prior art date
Application number
NL8500485A
Other languages
English (en)
Dutch (nl)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NL8500485A publication Critical patent/NL8500485A/nl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NL8500485A 1984-02-23 1985-02-21 Voorlopers van antiinflammatoire oxicamen. NL8500485A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23
US58268484 1984-02-23

Publications (1)

Publication Number Publication Date
NL8500485A true NL8500485A (nl) 1985-09-16

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8500485A NL8500485A (nl) 1984-02-23 1985-02-21 Voorlopers van antiinflammatoire oxicamen.

Country Status (22)

Country Link
JP (1) JPS60184077A (el)
KR (1) KR850006198A (el)
AU (1) AU552478B2 (el)
BE (1) BE901783A (el)
DD (1) DD232045A5 (el)
DE (1) DE3505576A1 (el)
DK (1) DK81185A (el)
ES (1) ES8606312A1 (el)
FI (1) FI850742L (el)
FR (1) FR2565980A1 (el)
GB (1) GB2154585A (el)
GR (1) GR850442B (el)
HU (1) HUT37616A (el)
IL (1) IL74407A0 (el)
IT (1) IT1185514B (el)
LU (1) LU85780A1 (el)
NL (1) NL8500485A (el)
NO (1) NO850725L (el)
PL (1) PL252023A1 (el)
PT (1) PT79988B (el)
SE (1) SE8500889L (el)
ZA (1) ZA851317B (el)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
JP5378221B2 (ja) * 2006-10-11 2013-12-25 テックフィールズ バイオケム カンパニー リミテッド 非常に高い皮膚浸透率を有するオキシカム及び関連化合物の正荷電水溶性プロドラッグ
KR101853971B1 (ko) 2007-06-04 2018-05-02 테크필즈 인크 매우 높은 피부 및 막 침투율을 가지는 비스테로이드성 소염제(nsaia) 약물전구체 및 이들의 새로운 의약적 용도
RU2765463C2 (ru) 2008-12-04 2022-01-31 Чунси ЮЙ Композиции интенсивного проникновения и их применение

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (it) * 1982-02-05 1982-02-05 Chiesi Farma Spa Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche.
IT1206525B (it) * 1982-12-10 1989-04-27 Zionale S R L A Roma Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione

Also Published As

Publication number Publication date
GR850442B (el) 1985-06-19
PT79988A (en) 1985-03-01
FI850742A0 (fi) 1985-02-22
AU3906685A (en) 1985-09-05
DD232045A5 (de) 1986-01-15
GB2154585A (en) 1985-09-11
DK81185D0 (da) 1985-02-22
JPS60184077A (ja) 1985-09-19
IL74407A0 (en) 1985-05-31
HUT37616A (en) 1986-01-23
KR850006198A (ko) 1985-10-02
BE901783A (fr) 1985-08-21
PL252023A1 (en) 1985-11-05
PT79988B (en) 1987-02-02
GB8504355D0 (en) 1985-03-20
NO850725L (no) 1985-08-26
DK81185A (da) 1985-09-10
SE8500889L (sv) 1985-08-24
FI850742L (fi) 1985-08-24
LU85780A1 (fr) 1985-12-11
IT8519585A0 (it) 1985-02-21
AU552478B2 (en) 1986-06-05
IT1185514B (it) 1987-11-12
ES8606312A1 (es) 1986-04-16
ES540590A0 (es) 1986-04-16
FR2565980A1 (fr) 1985-12-20
ZA851317B (en) 1986-10-29
DE3505576A1 (de) 1985-09-05
SE8500889D0 (sv) 1985-02-22

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