PT79988A - Process for preparing prodrugs of anti-inflammatory oxicams - Google Patents

Process for preparing prodrugs of anti-inflammatory oxicams

Info

Publication number
PT79988A
PT79988A PT79988A PT7998885A PT79988A PT 79988 A PT79988 A PT 79988A PT 79988 A PT79988 A PT 79988A PT 7998885 A PT7998885 A PT 7998885A PT 79988 A PT79988 A PT 79988A
Authority
PT
Portugal
Prior art keywords
oxicams
inflammatory
preparing prodrugs
prodrugs
preparing
Prior art date
Application number
PT79988A
Other languages
Portuguese (pt)
Other versions
PT79988B (en
Inventor
Joseph George Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of PT79988A publication Critical patent/PT79988A/en
Publication of PT79988B publication Critical patent/PT79988B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
PT79988A 1984-02-23 1985-02-20 Process for preparing prodrugs of anti-inflammatory oxicams PT79988B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23

Publications (2)

Publication Number Publication Date
PT79988A true PT79988A (en) 1985-03-01
PT79988B PT79988B (en) 1987-02-02

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
PT79988A PT79988B (en) 1984-02-23 1985-02-20 Process for preparing prodrugs of anti-inflammatory oxicams

Country Status (22)

Country Link
JP (1) JPS60184077A (en)
KR (1) KR850006198A (en)
AU (1) AU552478B2 (en)
BE (1) BE901783A (en)
DD (1) DD232045A5 (en)
DE (1) DE3505576A1 (en)
DK (1) DK81185A (en)
ES (1) ES8606312A1 (en)
FI (1) FI850742L (en)
FR (1) FR2565980A1 (en)
GB (1) GB2154585A (en)
GR (1) GR850442B (en)
HU (1) HUT37616A (en)
IL (1) IL74407A0 (en)
IT (1) IT1185514B (en)
LU (1) LU85780A1 (en)
NL (1) NL8500485A (en)
NO (1) NO850725L (en)
PL (1) PL252023A1 (en)
PT (1) PT79988B (en)
SE (1) SE8500889L (en)
ZA (1) ZA851317B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
JP5378221B2 (en) * 2006-10-11 2013-12-25 テックフィールズ バイオケム カンパニー リミテッド Positively charged water-soluble prodrugs of oxicam and related compounds with very high skin permeability
CN101687792B (en) 2007-06-04 2016-03-02 于崇曦 There is prodrug and the medicinal use thereof of the NSAID (non-steroidal anti-inflammatory drug) of fast skin and membranes penetration speed
KR101946297B1 (en) 2008-12-04 2019-02-11 충시 위 High Penetration Compositions and Their Applications

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (en) * 1982-02-05 1982-02-05 Chiesi Farma Spa NEW COMPOUNDS WITH ANTI-INFLAMMATORY ACTIVITY, PROCEDURE FOR THEIR PREPARATION AND RELATED PHARMACEUTICAL COMPOSITIONS.
IT1206525B (en) * 1982-12-10 1989-04-27 Zionale S R L A Roma NONSTEROID ANTI-INFLAMMATORY PREPARATION, FOR THE TREATMENT OF ARTHOREUMATIC AFFECTIONS AND METHOD FOR ITS PREPARATION

Also Published As

Publication number Publication date
SE8500889L (en) 1985-08-24
LU85780A1 (en) 1985-12-11
FI850742A0 (en) 1985-02-22
BE901783A (en) 1985-08-21
PT79988B (en) 1987-02-02
GB2154585A (en) 1985-09-11
DD232045A5 (en) 1986-01-15
IT8519585A0 (en) 1985-02-21
ES540590A0 (en) 1986-04-16
ES8606312A1 (en) 1986-04-16
DE3505576A1 (en) 1985-09-05
AU552478B2 (en) 1986-06-05
GR850442B (en) 1985-06-19
FI850742L (en) 1985-08-24
KR850006198A (en) 1985-10-02
ZA851317B (en) 1986-10-29
NO850725L (en) 1985-08-26
PL252023A1 (en) 1985-11-05
IT1185514B (en) 1987-11-12
AU3906685A (en) 1985-09-05
NL8500485A (en) 1985-09-16
SE8500889D0 (en) 1985-02-22
IL74407A0 (en) 1985-05-31
HUT37616A (en) 1986-01-23
GB8504355D0 (en) 1985-03-20
DK81185D0 (en) 1985-02-22
JPS60184077A (en) 1985-09-19
FR2565980A1 (en) 1985-12-20
DK81185A (en) 1985-09-10

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