DK81185A - CARBOXICAM ENOLESTER COMPOUNDS AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE - Google Patents

CARBOXICAM ENOLESTER COMPOUNDS AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE Download PDF

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Publication number
DK81185A
DK81185A DK81185A DK81185A DK81185A DK 81185 A DK81185 A DK 81185A DK 81185 A DK81185 A DK 81185A DK 81185 A DK81185 A DK 81185A DK 81185 A DK81185 A DK 81185A
Authority
DK
Denmark
Prior art keywords
carboxicam
enolester
compounds
pharmaceutical preparations
preparations containing
Prior art date
Application number
DK81185A
Other languages
Danish (da)
Other versions
DK81185D0 (en
Inventor
Joseph George Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK81185D0 publication Critical patent/DK81185D0/en
Publication of DK81185A publication Critical patent/DK81185A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
DK81185A 1984-02-23 1985-02-22 CARBOXICAM ENOLESTER COMPOUNDS AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE DK81185A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23

Publications (2)

Publication Number Publication Date
DK81185D0 DK81185D0 (en) 1985-02-22
DK81185A true DK81185A (en) 1985-09-10

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
DK81185A DK81185A (en) 1984-02-23 1985-02-22 CARBOXICAM ENOLESTER COMPOUNDS AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE

Country Status (22)

Country Link
JP (1) JPS60184077A (en)
KR (1) KR850006198A (en)
AU (1) AU552478B2 (en)
BE (1) BE901783A (en)
DD (1) DD232045A5 (en)
DE (1) DE3505576A1 (en)
DK (1) DK81185A (en)
ES (1) ES8606312A1 (en)
FI (1) FI850742L (en)
FR (1) FR2565980A1 (en)
GB (1) GB2154585A (en)
GR (1) GR850442B (en)
HU (1) HUT37616A (en)
IL (1) IL74407A0 (en)
IT (1) IT1185514B (en)
LU (1) LU85780A1 (en)
NL (1) NL8500485A (en)
NO (1) NO850725L (en)
PL (1) PL252023A1 (en)
PT (1) PT79988B (en)
SE (1) SE8500889L (en)
ZA (1) ZA851317B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
EP2084165B1 (en) * 2006-10-11 2013-06-12 Techfields Biochem Co. Ltd Positively charged water-soluble prodrugs of oxicams and related compounds with very high skin penetration rate
WO2008149181A1 (en) 2007-06-04 2008-12-11 Techfields Inc Pro-drugs of nsaias with very high skin and membranes penetration rates and their new medicinal uses
CN108191846B (en) 2008-12-04 2021-08-20 于崇曦 High penetration composition and application thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (en) * 1982-02-05 1982-02-05 Chiesi Farma Spa NEW COMPOUNDS WITH ANTI-INFLAMMATORY ACTIVITY, PROCEDURE FOR THEIR PREPARATION AND RELATED PHARMACEUTICAL COMPOSITIONS.
IT1206525B (en) * 1982-12-10 1989-04-27 Zionale S R L A Roma NONSTEROID ANTI-INFLAMMATORY PREPARATION, FOR THE TREATMENT OF ARTHOREUMATIC AFFECTIONS AND METHOD FOR ITS PREPARATION

Also Published As

Publication number Publication date
HUT37616A (en) 1986-01-23
FR2565980A1 (en) 1985-12-20
PT79988B (en) 1987-02-02
PT79988A (en) 1985-03-01
LU85780A1 (en) 1985-12-11
AU3906685A (en) 1985-09-05
NL8500485A (en) 1985-09-16
JPS60184077A (en) 1985-09-19
GR850442B (en) 1985-06-19
ES540590A0 (en) 1986-04-16
SE8500889D0 (en) 1985-02-22
FI850742L (en) 1985-08-24
IT1185514B (en) 1987-11-12
KR850006198A (en) 1985-10-02
GB8504355D0 (en) 1985-03-20
PL252023A1 (en) 1985-11-05
GB2154585A (en) 1985-09-11
IL74407A0 (en) 1985-05-31
FI850742A0 (en) 1985-02-22
NO850725L (en) 1985-08-26
IT8519585A0 (en) 1985-02-21
ZA851317B (en) 1986-10-29
DE3505576A1 (en) 1985-09-05
SE8500889L (en) 1985-08-24
DK81185D0 (en) 1985-02-22
AU552478B2 (en) 1986-06-05
ES8606312A1 (en) 1986-04-16
BE901783A (en) 1985-08-21
DD232045A5 (en) 1986-01-15

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Legal Events

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AHB Application shelved due to non-payment