SE8500889L - ANTI-INFLAMMATORY OXICAN ANIMALS - Google Patents

ANTI-INFLAMMATORY OXICAN ANIMALS

Info

Publication number
SE8500889L
SE8500889L SE8500889A SE8500889A SE8500889L SE 8500889 L SE8500889 L SE 8500889L SE 8500889 A SE8500889 A SE 8500889A SE 8500889 A SE8500889 A SE 8500889A SE 8500889 L SE8500889 L SE 8500889L
Authority
SE
Sweden
Prior art keywords
oxican
inflammatory
animals
toluoyl
benzoyl
Prior art date
Application number
SE8500889A
Other languages
Swedish (sv)
Other versions
SE8500889D0 (en
Inventor
J G Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of SE8500889D0 publication Critical patent/SE8500889D0/en
Publication of SE8500889L publication Critical patent/SE8500889L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Novel enol esters of the formula <IMAGE> wherein R1 is an C2-8 alkanoyl, benzoyl, toluoyl, C1-8 alkylsulfonyl or benzene-sulfonyl group; R2 is 5-methylisoxazol-3-yl or 6-chloro-2-pyridyl and R3 is benzoyl, toluoyl, C1-8alkylsulfonyl or benzene sulfonyl; are ### MPW Shell - /s must occur in pairs. useful as prodrug forms of the known unesterified antiinflammatory and analgesic oxicams.
SE8500889A 1984-02-23 1985-02-22 ANTI-INFLAMMATORY OXICAN ANIMALS SE8500889L (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58268484A 1984-02-23 1984-02-23

Publications (2)

Publication Number Publication Date
SE8500889D0 SE8500889D0 (en) 1985-02-22
SE8500889L true SE8500889L (en) 1985-08-24

Family

ID=24330094

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8500889A SE8500889L (en) 1984-02-23 1985-02-22 ANTI-INFLAMMATORY OXICAN ANIMALS

Country Status (22)

Country Link
JP (1) JPS60184077A (en)
KR (1) KR850006198A (en)
AU (1) AU552478B2 (en)
BE (1) BE901783A (en)
DD (1) DD232045A5 (en)
DE (1) DE3505576A1 (en)
DK (1) DK81185A (en)
ES (1) ES8606312A1 (en)
FI (1) FI850742L (en)
FR (1) FR2565980A1 (en)
GB (1) GB2154585A (en)
GR (1) GR850442B (en)
HU (1) HUT37616A (en)
IL (1) IL74407A0 (en)
IT (1) IT1185514B (en)
LU (1) LU85780A1 (en)
NL (1) NL8500485A (en)
NO (1) NO850725L (en)
PL (1) PL252023A1 (en)
PT (1) PT79988B (en)
SE (1) SE8500889L (en)
ZA (1) ZA851317B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US20090238763A1 (en) 2006-07-09 2009-09-24 Chongxi Yu High penetration compositions and uses thereof
US20090221703A1 (en) 2006-07-09 2009-09-03 Chongxi Yu High penetration composition and uses thereof
CN101522692A (en) * 2006-10-11 2009-09-02 于崇曦 Positively charged water-soluble prodrugs of oxicams and related compounds with very high skin penetration rate
US9371284B2 (en) 2007-06-04 2016-06-21 Techfields Pharma Co., Ltd. Pro-drugs of NSAIAS with very high skin and membranes penetration rates and their new medicinal uses
KR20230085223A (en) 2008-12-04 2023-06-13 충시 위 High Penetration Compositions and Their Applications

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591574A (en) * 1968-05-29 1971-07-06 American Home Prod Tri-n-phenylglycyl derivatives of insulin
US3787324A (en) * 1971-03-01 1974-01-22 Warner Lambert Co 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production
US3704298A (en) * 1971-06-22 1972-11-28 Warner Lambert Co 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides
AU518216B2 (en) * 1977-09-06 1981-09-17 Hafslund Nycomed Pharma Aktiengesellschaft Thienothiazine derivatives
JPS5714589A (en) * 1980-06-27 1982-01-25 Mitsui Toatsu Chem Inc Benzothiazine derivative, its preparation and drug composition
US4309427A (en) * 1981-01-15 1982-01-05 Pfizer Inc. Benzothiazine dioxide derivatives
IT8219486A0 (en) * 1982-02-05 1982-02-05 Chiesi Farma Spa NEW COMPOUNDS WITH ANTI-INFLAMMATORY ACTIVITY, PROCEDURE FOR THEIR PREPARATION AND RELATED PHARMACEUTICAL COMPOSITIONS.
IT1206525B (en) * 1982-12-10 1989-04-27 Zionale S R L A Roma NONSTEROID ANTI-INFLAMMATORY PREPARATION, FOR THE TREATMENT OF ARTHOREUMATIC AFFECTIONS AND METHOD FOR ITS PREPARATION

Also Published As

Publication number Publication date
IT1185514B (en) 1987-11-12
JPS60184077A (en) 1985-09-19
AU552478B2 (en) 1986-06-05
GB8504355D0 (en) 1985-03-20
NO850725L (en) 1985-08-26
FI850742L (en) 1985-08-24
IL74407A0 (en) 1985-05-31
ES540590A0 (en) 1986-04-16
KR850006198A (en) 1985-10-02
DE3505576A1 (en) 1985-09-05
PL252023A1 (en) 1985-11-05
AU3906685A (en) 1985-09-05
HUT37616A (en) 1986-01-23
DK81185D0 (en) 1985-02-22
SE8500889D0 (en) 1985-02-22
GB2154585A (en) 1985-09-11
BE901783A (en) 1985-08-21
FI850742A0 (en) 1985-02-22
FR2565980A1 (en) 1985-12-20
DK81185A (en) 1985-09-10
PT79988B (en) 1987-02-02
ES8606312A1 (en) 1986-04-16
ZA851317B (en) 1986-10-29
PT79988A (en) 1985-03-01
GR850442B (en) 1985-06-19
LU85780A1 (en) 1985-12-11
NL8500485A (en) 1985-09-16
DD232045A5 (en) 1986-01-15
IT8519585A0 (en) 1985-02-21

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