ZA851317B - Ester prodrugs of oxicams - Google Patents
Ester prodrugs of oxicamsInfo
- Publication number
- ZA851317B ZA851317B ZA851317A ZA851317A ZA851317B ZA 851317 B ZA851317 B ZA 851317B ZA 851317 A ZA851317 A ZA 851317A ZA 851317 A ZA851317 A ZA 851317A ZA 851317 B ZA851317 B ZA 851317B
- Authority
- ZA
- South Africa
- Prior art keywords
- oxicams
- ester prodrugs
- prodrugs
- ester
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US58268484A | 1984-02-23 | 1984-02-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA851317B true ZA851317B (en) | 1986-10-29 |
Family
ID=24330094
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA851317A ZA851317B (en) | 1984-02-23 | 1985-02-21 | Ester prodrugs of oxicams |
Country Status (22)
| Country | Link |
|---|---|
| JP (1) | JPS60184077A (el) |
| KR (1) | KR850006198A (el) |
| AU (1) | AU552478B2 (el) |
| BE (1) | BE901783A (el) |
| DD (1) | DD232045A5 (el) |
| DE (1) | DE3505576A1 (el) |
| DK (1) | DK81185A (el) |
| ES (1) | ES8606312A1 (el) |
| FI (1) | FI850742L (el) |
| FR (1) | FR2565980A1 (el) |
| GB (1) | GB2154585A (el) |
| GR (1) | GR850442B (el) |
| HU (1) | HUT37616A (el) |
| IL (1) | IL74407A0 (el) |
| IT (1) | IT1185514B (el) |
| LU (1) | LU85780A1 (el) |
| NL (1) | NL8500485A (el) |
| NO (1) | NO850725L (el) |
| PL (1) | PL252023A1 (el) |
| PT (1) | PT79988B (el) |
| SE (1) | SE8500889L (el) |
| ZA (1) | ZA851317B (el) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4623486A (en) * | 1985-05-29 | 1986-11-18 | Pfizer Inc. | [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity |
| US4610982A (en) * | 1985-06-03 | 1986-09-09 | Pfizer Inc. | Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor |
| US20090221703A1 (en) | 2006-07-09 | 2009-09-03 | Chongxi Yu | High penetration composition and uses thereof |
| US20090238763A1 (en) | 2006-07-09 | 2009-09-24 | Chongxi Yu | High penetration compositions and uses thereof |
| CN101522692A (zh) * | 2006-10-11 | 2009-09-02 | 于崇曦 | 具有快速皮肤穿透速度的带正电荷的水溶性的昔康及其相关化合物的前药 |
| JP2010529101A (ja) | 2007-06-04 | 2010-08-26 | テックフィールズ インコーポレイテッド | 非常に速い皮膚及び膜浸透速度を有するｎｓａｉａプロドラッグ及びその新規医薬使用 |
| MX362949B (es) | 2008-12-04 | 2019-02-27 | Yu Chongxi | Composiciones de alta penetracion y sus aplicaciones. |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3591574A (en) * | 1968-05-29 | 1971-07-06 | American Home Prod | Tri-n-phenylglycyl derivatives of insulin |
| US3787324A (en) * | 1971-03-01 | 1974-01-22 | Warner Lambert Co | 4-hydroxy-3-(3-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,dioxides and process for their production |
| US3704298A (en) * | 1971-06-22 | 1972-11-28 | Warner Lambert Co | 4-acyloxy-3-(2-isoxazolocarbamyl)-2h-1,2-benzothiazine 1,1-dioxides |
| AU518216B2 (en) * | 1977-09-06 | 1981-09-17 | Hafslund Nycomed Pharma Aktiengesellschaft | Thienothiazine derivatives |
| JPS5714589A (en) * | 1980-06-27 | 1982-01-25 | Mitsui Toatsu Chem Inc | Benzothiazine derivative, its preparation and drug composition |
| US4309427A (en) * | 1981-01-15 | 1982-01-05 | Pfizer Inc. | Benzothiazine dioxide derivatives |
| IT8219486A0 (it) * | 1982-02-05 | 1982-02-05 | Chiesi Farma Spa | Nuovi composti ad attivita'antiinfiammatoria, procedimento per la loro preparazione e relative composizioni farmaceutiche. |
| IT1206525B (it) * | 1982-12-10 | 1989-04-27 | Zionale S R L A Roma | Preparato anti-infiammatorio nonsteroideo, per il trattamento delle affezioni artroreumatiche e metodo per la sua preparazione |
-
1985
- 1985-01-23 JP JP60010722A patent/JPS60184077A/ja active Pending
- 1985-02-18 DE DE19853505576 patent/DE3505576A1/de not_active Ceased
- 1985-02-19 PL PL25202385A patent/PL252023A1/xx unknown
- 1985-02-20 GR GR850442A patent/GR850442B/el unknown
- 1985-02-20 LU LU85780A patent/LU85780A1/fr unknown
- 1985-02-20 PT PT79988A patent/PT79988B/pt unknown
- 1985-02-20 GB GB08504355A patent/GB2154585A/en not_active Withdrawn
- 1985-02-21 ZA ZA851317A patent/ZA851317B/xx unknown
- 1985-02-21 NL NL8500485A patent/NL8500485A/nl not_active Application Discontinuation
- 1985-02-21 ES ES540590A patent/ES8606312A1/es not_active Expired
- 1985-02-21 BE BE0/214544A patent/BE901783A/fr not_active IP Right Cessation
- 1985-02-21 DD DD85273451A patent/DD232045A5/de unknown
- 1985-02-21 IL IL74407A patent/IL74407A0/xx unknown
- 1985-02-21 IT IT8519585A patent/IT1185514B/it active
- 1985-02-22 AU AU39066/85A patent/AU552478B2/en not_active Ceased
- 1985-02-22 HU HU85678A patent/HUT37616A/hu unknown
- 1985-02-22 FI FI850742A patent/FI850742L/fi not_active Application Discontinuation
- 1985-02-22 DK DK81185A patent/DK81185A/da not_active Application Discontinuation
- 1985-02-22 KR KR1019850001106A patent/KR850006198A/ko not_active Application Discontinuation
- 1985-02-22 FR FR8502586A patent/FR2565980A1/fr active Pending
- 1985-02-22 SE SE8500889A patent/SE8500889L/xx not_active Application Discontinuation
- 1985-02-22 NO NO850725A patent/NO850725L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BE901783A (fr) | 1985-08-21 |
| GB8504355D0 (en) | 1985-03-20 |
| FR2565980A1 (fr) | 1985-12-20 |
| GR850442B (el) | 1985-06-19 |
| HUT37616A (en) | 1986-01-23 |
| NL8500485A (nl) | 1985-09-16 |
| DK81185D0 (da) | 1985-02-22 |
| FI850742A0 (fi) | 1985-02-22 |
| NO850725L (no) | 1985-08-26 |
| FI850742L (fi) | 1985-08-24 |
| DE3505576A1 (de) | 1985-09-05 |
| PT79988B (en) | 1987-02-02 |
| KR850006198A (ko) | 1985-10-02 |
| ES8606312A1 (es) | 1986-04-16 |
| AU3906685A (en) | 1985-09-05 |
| ES540590A0 (es) | 1986-04-16 |
| JPS60184077A (ja) | 1985-09-19 |
| DD232045A5 (de) | 1986-01-15 |
| SE8500889L (sv) | 1985-08-24 |
| LU85780A1 (fr) | 1985-12-11 |
| IT8519585A0 (it) | 1985-02-21 |
| GB2154585A (en) | 1985-09-11 |
| IT1185514B (it) | 1987-11-12 |
| SE8500889D0 (sv) | 1985-02-22 |
| PT79988A (en) | 1985-03-01 |
| AU552478B2 (en) | 1986-06-05 |
| PL252023A1 (en) | 1985-11-05 |
| DK81185A (da) | 1985-09-10 |
| IL74407A0 (en) | 1985-05-31 |
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