NL8104938A - 1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan. - Google Patents

1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan. Download PDF

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Publication number
NL8104938A
NL8104938A NL8104938A NL8104938A NL8104938A NL 8104938 A NL8104938 A NL 8104938A NL 8104938 A NL8104938 A NL 8104938A NL 8104938 A NL8104938 A NL 8104938A NL 8104938 A NL8104938 A NL 8104938A
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NL
Netherlands
Prior art keywords
tosylate
compound
preparation
amino
compound according
Prior art date
Application number
NL8104938A
Other languages
English (en)
Dutch (nl)
Original Assignee
Leo Pharm Prod Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd
Publication of NL8104938A publication Critical patent/NL8104938A/nl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NL8104938A 1980-10-31 1981-10-30 1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan. NL8104938A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8035156 1980-10-31
GB8035156 1980-10-31

Publications (1)

Publication Number Publication Date
NL8104938A true NL8104938A (nl) 1982-05-17

Family

ID=10517019

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8104938A NL8104938A (nl) 1980-10-31 1981-10-30 1.1-dioxopenicillanoyloxymethyl-6-(d-alfa-amino-alfa-fenylaceetamido)penicillanaat, werkwijze voor de bereiding en toepassing daarvan.

Country Status (26)

Country Link
US (1) US4831025A (cs)
JP (1) JPS57126493A (cs)
KR (1) KR870001982B1 (cs)
AT (1) AT373893B (cs)
AU (1) AU543870B2 (cs)
BE (1) BE890938A (cs)
CA (1) CA1180696A (cs)
CH (1) CH647527A5 (cs)
DE (1) DE3143219A1 (cs)
DK (1) DK154219C (cs)
ES (1) ES506751A0 (cs)
FI (1) FI813331L (cs)
FR (1) FR2493322B1 (cs)
GB (1) GB2114969B (cs)
GR (1) GR75369B (cs)
IE (1) IE51640B1 (cs)
IL (1) IL64009A (cs)
IT (1) IT1193735B (cs)
LU (1) LU83727A1 (cs)
NL (1) NL8104938A (cs)
NO (1) NO813683L (cs)
NZ (1) NZ198622A (cs)
PH (1) PH17820A (cs)
PT (1) PT73913B (cs)
SE (1) SE452322B (cs)
ZA (1) ZA817091B (cs)

Families Citing this family (43)

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US4432987A (en) * 1982-04-23 1984-02-21 Pfizer Inc. Crystalline benzenesulfonate salts of sultamicillin
PH20068A (en) * 1982-12-06 1986-09-18 Pfizer Process and intermediates for sultamicillin and analogs
KR910009271B1 (ko) * 1989-06-20 1991-11-08 김영설 1,1-디옥소페닐실라노일 옥시메틸 D-6-[α-(메틸렌아미노)페닐-아세트아미도]-페니실라네이트와 그의 파라-톨루엔술폰산염
ES2161602B1 (es) * 1999-04-08 2003-02-16 Asturpharma S A Sintesis de 6-(d-alfa-(bencilidenaminofenilacetamido))penicilanato de 1,1-dioxopenicilanoiloximetilo y analogos. nuevos intermedios para la sintesis de sultamicilina.
US6663891B2 (en) 2000-02-24 2003-12-16 Advancis Pharmaceutical Corp. Erythromyacin antibiotic product, use and formulation thereof
US6669948B2 (en) 2000-02-24 2003-12-30 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6632453B2 (en) 2000-02-24 2003-10-14 Advancis Pharmaceutical Corp. Ciprofoxacin-metronidazole antibiotic composition
US6991807B2 (en) * 2000-02-24 2006-01-31 Advancis Pharmaceutical, Corp. Antibiotic composition
US6667057B2 (en) 2000-02-24 2003-12-23 Advancis Pharmaceutical Corp. Levofloxacin antibiotic product, use and formulation thereof
US6730320B2 (en) 2000-02-24 2004-05-04 Advancis Pharmaceutical Corp. Tetracycline antibiotic product, use and formulation thereof
JP2003523378A (ja) * 2000-02-24 2003-08-05 アドバンシス ファーマシューティカル コーポレイション 治療剤製品、その使用及び製剤形態
US6663890B2 (en) 2000-02-24 2003-12-16 Advancis Pharmaceutical Corp. Metronidazole antibiotic product, use and formulation thereof
US6610328B2 (en) 2000-02-24 2003-08-26 Advancis Pharmaceutical Corp. Amoxicillin-clarithromycin antibiotic composition
US6627222B2 (en) 2000-02-24 2003-09-30 Advancis Pharmaceutical Corp. Amoxicillin-dicloxacillin antibiotic composition
US7025989B2 (en) * 2000-02-24 2006-04-11 Advancis Pharmaceutical Corp. Multiple-delayed released antibiotic product, use and formulation thereof
WO2001062195A1 (en) * 2000-02-24 2001-08-30 Advancis Pharmaceutical Corporation Antibiotic and antifungal compositions
US6638532B2 (en) 2000-02-24 2003-10-28 Advancis Pharmaceutical Corp. Tetracycline—doxycycline antibiotic composition
US6565882B2 (en) 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6667042B2 (en) 2000-02-24 2003-12-23 Advancis Pharmaceutical Corp. Fluroquinilone antibiotic product, use and formulation thereof
US6623758B2 (en) 2000-02-24 2003-09-23 Advancis Pharmaceutical Corp. Cephalosporin-metronidazole antibiotic composition
US7074417B2 (en) * 2000-10-13 2006-07-11 Advancis Pharmaceutical Corporation Multiple-delayed release anti-viral product, use and formulation thereof
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US7157095B2 (en) * 2000-10-13 2007-01-02 Advancis Pharmaceutical Corporation Multiple-delayed release antifungal product, use and formulation thereof
US7105174B2 (en) * 2000-10-13 2006-09-12 Advancis Pharmaceutical Corporation Multiple-delayed release anti-neoplastic product, use and formulation thereof
US20020197314A1 (en) * 2001-02-23 2002-12-26 Rudnic Edward M. Anti-fungal composition
US20040114368A1 (en) * 2002-12-13 2004-06-17 Shyu Shing Jy Light device having rotatable or movable view
US20040265323A1 (en) * 2003-05-16 2004-12-30 Mccormick Beth A. Compositions comprising pathogen elicited epithelial chemoattractant (eicosanoid hepoxilin A3), inhibitors thereof and methods of use thereof
CA2533358C (en) 2003-07-21 2014-03-11 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
US8313776B2 (en) 2003-07-21 2012-11-20 Shionogi Inc. Antibiotic product, use and formulation thereof
JP2006528190A (ja) 2003-07-21 2006-12-14 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
AU2004264939A1 (en) 2003-08-11 2005-02-24 Middlebrook Pharmaceuticals, Inc. Robust pellet
JP2007502294A (ja) 2003-08-12 2007-02-08 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
WO2005023184A2 (en) 2003-08-29 2005-03-17 Advancis Pharmaceuticals Corporation Antibiotic product, use and formulation thereof
EP1663169A4 (en) 2003-09-15 2010-11-24 Middlebrook Pharmaceuticals In ANTIBIOTICS, ITS USE AND FORMULATION
JP2008505124A (ja) 2004-07-02 2008-02-21 アドバンシス ファーマスーティカル コーポレイション パルス送達用錠剤
WO2007004239A1 (en) * 2005-07-06 2007-01-11 Morepen Laboratories Limited New polymorphic form of sultamicillin tosylate and a process therefor
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8299052B2 (en) * 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication
WO2014014364A1 (en) 2012-07-17 2014-01-23 Bayer New Zealand Limited Injectable antibiotic formulations and their methods of use
ES2752034T3 (es) 2012-07-17 2020-04-02 Bayer New Zealand Ltd Formaciones inyectables de antibiótico y sus procedimientos de uso
US11116737B1 (en) 2020-04-10 2021-09-14 University Of Georgia Research Foundation, Inc. Methods of using probenecid for treatment of coronavirus infections

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1532222A (fr) * 1963-10-28 1968-07-12 Bristol Myers Co Procédé de préparation de dérivés de la pénicilline
IE49880B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd Penicillin derivatives
BE881675A (fr) * 1979-02-13 1980-08-12 Leo Pharm Prod Ltd B-lactames derives de l'acide penicillanique leur preparation et leurs utilisations therapeutiques
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
IE51516B1 (en) * 1980-10-06 1987-01-07 Leo Pharm Prod Ltd 1,1-dioxapenicillanoyloxymethyl 6-(d-alpha-amino-alpha-phenylacetamido)penicillanate napsylate

Also Published As

Publication number Publication date
JPS57126493A (en) 1982-08-06
DE3143219A1 (de) 1982-08-12
IE812361L (en) 1982-04-30
FI813331A7 (fi) 1982-05-01
IL64009A (en) 1984-09-30
IT1193735B (it) 1988-08-24
NO813683L (no) 1982-05-03
PT73913A (en) 1981-11-01
SE8106404L (sv) 1982-05-01
DE3143219C2 (cs) 1990-05-17
NZ198622A (en) 1985-07-12
IE51640B1 (en) 1987-01-21
DK154219B (da) 1988-10-24
DK154219C (da) 1989-03-20
AT373893B (de) 1984-02-27
DK472181A (da) 1982-05-01
GB2114969B (en) 1985-02-20
JPH027957B2 (cs) 1990-02-21
KR870001982B1 (ko) 1987-10-24
CH647527A5 (de) 1985-01-31
FI813331L (fi) 1982-05-01
FR2493322B1 (fr) 1986-06-13
SE452322B (sv) 1987-11-23
PH17820A (en) 1985-01-07
GR75369B (cs) 1984-07-13
KR830007671A (ko) 1983-11-04
ATA447781A (de) 1983-07-15
FR2493322A1 (fr) 1982-05-07
IL64009A0 (en) 1982-01-31
GB2114969A (en) 1983-09-01
ES8206531A1 (es) 1982-08-16
LU83727A1 (fr) 1982-05-07
ZA817091B (en) 1982-10-27
AU543870B2 (en) 1985-05-09
BE890938A (fr) 1982-04-30
US4831025A (en) 1989-05-16
PT73913B (en) 1984-05-29
ES506751A0 (es) 1982-08-16
AU7636581A (en) 1982-05-06
CA1180696A (en) 1985-01-08
IT8168383A0 (it) 1981-10-23

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
BN A decision not to publish the application has become irrevocable