NL194273C - Werkwijze voor de resolutie van glycidinezuurderivaten. - Google Patents

Werkwijze voor de resolutie van glycidinezuurderivaten. Download PDF

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Publication number
NL194273C
NL194273C NL9100853A NL9100853A NL194273C NL 194273 C NL194273 C NL 194273C NL 9100853 A NL9100853 A NL 9100853A NL 9100853 A NL9100853 A NL 9100853A NL 194273 C NL194273 C NL 194273C
Authority
NL
Netherlands
Prior art keywords
mmol
thiophenol
formula
solution
methyl ester
Prior art date
Application number
NL9100853A
Other languages
English (en)
Dutch (nl)
Other versions
NL9100853A (nl
NL194273B (nl
Inventor
Claudio Giordano
Roberto Casagrande
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of NL9100853A publication Critical patent/NL9100853A/nl
Publication of NL194273B publication Critical patent/NL194273B/xx
Application granted granted Critical
Publication of NL194273C publication Critical patent/NL194273C/nl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/26—Separation; Purification; Stabilisation; Use of additives
    • C07C319/28—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Saccharide Compounds (AREA)
NL9100853A 1990-05-17 1991-05-16 Werkwijze voor de resolutie van glycidinezuurderivaten. NL194273C (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2034990 1990-05-17
IT20349A IT1240651B (it) 1990-05-17 1990-05-17 Processo per la risoluzione di derivati glicidici

Publications (3)

Publication Number Publication Date
NL9100853A NL9100853A (nl) 1991-12-16
NL194273B NL194273B (nl) 2001-07-02
NL194273C true NL194273C (nl) 2001-11-05

Family

ID=11165943

Family Applications (1)

Application Number Title Priority Date Filing Date
NL9100853A NL194273C (nl) 1990-05-17 1991-05-16 Werkwijze voor de resolutie van glycidinezuurderivaten.

Country Status (13)

Country Link
US (1) US5198557A (it)
JP (1) JP3122953B2 (it)
AT (1) AT401055B (it)
BE (1) BE1004850A3 (it)
CA (1) CA2041305C (it)
CH (1) CH682075A5 (it)
DE (1) DE4115698C2 (it)
ES (1) ES2033575B1 (it)
FR (1) FR2662161B1 (it)
GB (1) GB2244055B (it)
IT (1) IT1240651B (it)
NL (1) NL194273C (it)
SE (1) SE509298C2 (it)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2658513B1 (fr) * 1990-02-21 1994-02-04 Rhone Poulenc Sante Procede de preparation de l'acide cis-beta-phenylglycidique-(2r,3r).
IT1249777B (it) * 1990-05-17 1995-03-18 Zambon Spa Processo per la preparazione di intermedi per la sintesi del diltiazem
DE4209497A1 (de) * 1992-03-24 1993-09-30 Basf Ag Verfahren zur Herstellung von chlorsubstituierten olefinischen Verbindungen
US6262278B1 (en) 1995-03-14 2001-07-17 President And Fellows Of Harvard College Stereoselective ring opening reactions
SG72731A1 (en) * 1996-03-15 2000-05-23 Nabe Seiyaku Co Ltd Process for preparing optically active trans-3-phenylglycidamide compounds
DE60102825T2 (de) 2000-07-31 2005-03-31 Brandeis University, Waltham Kinetische racematspaltung chiraler 2- und 3- substituierter carbonsäuren
US6562967B2 (en) * 2000-07-31 2003-05-13 Brandeis University Kinetic resolutions of chiral 2-and-3-substituted carboxylic acids
US7531662B2 (en) * 2003-06-11 2009-05-12 Brandeis University Cinchona-alkaloid-based catalysts, and asymmetric alcoholysis of cyclic anhydrides using them

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1236467A (en) * 1967-10-28 1971-06-23 Tanabe Seiyaku Co Benzothiazepine derivatives
EP0059335B1 (en) * 1981-02-27 1985-05-15 Tanabe Seiyaku Co., Ltd. Novel process for preparing threo-2-hydroxy-3-(4-methoxyphenyl)-3-(2-nitrophenylthio)-propionic ester
SE449611B (sv) * 1982-07-09 1987-05-11 Tanabe Seiyaku Co Sett att framstella 1,5-bensotiazepinderivat
IT1152721B (it) * 1982-10-15 1987-01-07 Luso Farmaco Inst Risoluzione ottica dell'acido dl-alfa-2-idrossi-3-(4-metossifenil)-3-(2-amminofeniltio)propionico
US4567175A (en) * 1983-06-03 1986-01-28 Tanabe Seiyaku Co., Ltd. 8-Chloro-1,5-benzothiazepine derivatives
JPS6013776A (ja) * 1983-07-05 1985-01-24 Sawai Seiyaku Kk 光学活性３−（ｐ−アルコキシフエニル）グリシツド酸誘導体の製造法
JPS6013775A (ja) * 1983-07-05 1985-01-24 Sawai Seiyaku Kk 光学活性３−（ｐ−アルコキシフエニル）グリシツド酸アルカリ金属塩の製造法
US4594342A (en) * 1984-04-10 1986-06-10 Tanabe Seiyaku Co., Ltd. 1,5-benzothiazepine derivative
GB2167063A (en) * 1984-11-17 1986-05-21 Tanabe Seiyaku Co 6 or 9-chloro-1, 5-benzothiazepine derivatives
EP0320532A1 (en) * 1986-07-15 1989-06-21 Nihon Iyakuhin Kogyo Co., Ltd. Novel optically active carboxylic acid derivative l-lysine salt and process for production thereof
IT1217988B (it) * 1988-01-28 1990-03-30 Ind Chimica Profarmaco Spa Procedimento per la risoluzione ottica di un pacemo
US4864058A (en) * 1988-05-10 1989-09-05 Hoffmann-La Roche Inc. Process for making optically active naphtho[1,2-b][1,4]thiazepin-4(5H)-ones
US4996352A (en) * 1988-05-10 1991-02-26 Hoffmann-La Roche Inc. Enantiomers of β-[(2-amino-1-naphthalenyl) thiol]-α-hydroxy-4-methoxybenzene propanoic acid
US4885375A (en) * 1988-05-18 1989-12-05 Marion Laboratories, Inc. Resolution of 3-(4-methoxyphenyl)glycidic acid with in situ conversion to alkyl esters
NL8801311A (nl) * 1988-05-20 1989-12-18 Stamicarbon Fenylglycidaatstereoisomeren, omzettingsprodukten daarvan met 2-nitrothiofenol en de bereiding van diltiazem.
FR2637285B1 (fr) * 1988-10-03 1991-04-12 Synthelabo Procede de preparation de derives de l'acide propionique et produits obtenus
ATE93516T1 (de) * 1989-06-30 1993-09-15 Richter Gedeon Vegyeszet Verfahren zur resolution von threo-3-((2aminophenyl)-thio>-2-hydroxy-3-(4-methoxyphenyl)propions|ure.

Also Published As

Publication number Publication date
NL9100853A (nl) 1991-12-16
BE1004850A3 (fr) 1993-02-09
CA2041305C (en) 2000-12-12
AT401055B (de) 1996-06-25
SE9101483L (sv) 1991-11-18
SE509298C2 (sv) 1999-01-11
GB9108741D0 (en) 1991-06-12
IT1240651B (it) 1993-12-17
ATA99691A (de) 1995-10-15
DE4115698A1 (de) 1991-11-21
IT9020349A0 (it) 1990-05-17
FR2662161A1 (fr) 1991-11-22
SE9101483D0 (sv) 1991-05-16
GB2244055A (en) 1991-11-20
IT9020349A1 (it) 1991-11-17
ES2033575B1 (es) 1994-02-01
JPH0616652A (ja) 1994-01-25
NL194273B (nl) 2001-07-02
CA2041305A1 (en) 1991-11-18
US5198557A (en) 1993-03-30
ES2033575A1 (es) 1993-03-16
GB2244055B (en) 1993-09-22
FR2662161B1 (fr) 1993-08-06
DE4115698C2 (de) 2001-08-23
JP3122953B2 (ja) 2001-01-09
CH682075A5 (it) 1993-07-15

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BB A search report has been drawn up
BC A request for examination has been filed
V1 Lapsed because of non-payment of the annual fee

Effective date: 20051201