MY7300310A - Process for preparing benzothiazone dioxides - Google Patents

Process for preparing benzothiazone dioxides

Info

Publication number
MY7300310A
MY7300310A MY310/73A MY7300310A MY7300310A MY 7300310 A MY7300310 A MY 7300310A MY 310/73 A MY310/73 A MY 310/73A MY 7300310 A MY7300310 A MY 7300310A MY 7300310 A MY7300310 A MY 7300310A
Authority
MY
Malaysia
Prior art keywords
benzothiazone
dioxides
preparing
preparing benzothiazone
benzothiazone dioxides
Prior art date
Application number
MY310/73A
Other languages
English (en)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MY7300310A publication Critical patent/MY7300310A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
MY310/73A 1968-08-27 1973-12-30 Process for preparing benzothiazone dioxides MY7300310A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76759468A 1968-08-27 1968-08-27

Publications (1)

Publication Number Publication Date
MY7300310A true MY7300310A (en) 1973-12-31

Family

ID=25079964

Family Applications (1)

Application Number Title Priority Date Filing Date
MY310/73A MY7300310A (en) 1968-08-27 1973-12-30 Process for preparing benzothiazone dioxides

Country Status (18)

Country Link
US (1) US3591584A (fr)
JP (2) JPS50677B1 (fr)
AT (2) AT298503B (fr)
BE (1) BE737962A (fr)
BR (1) BR6911817D0 (fr)
CH (1) CH520705A (fr)
DE (2) DE1943265C3 (fr)
DK (1) DK145297C (fr)
ES (1) ES370861A1 (fr)
FI (1) FI51189C (fr)
FR (1) FR2016455B1 (fr)
GB (1) GB1257180A (fr)
IL (1) IL32836A (fr)
MY (1) MY7300310A (fr)
NL (1) NL157013B (fr)
NO (1) NO129746B (fr)
PH (1) PH10029A (fr)
SE (2) SE373854B (fr)

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US3769292A (en) * 1972-04-28 1973-10-30 Warner Lambert Co N-(pyridyl)2h 1-benzothiopyran-3-carboxamide-4-hydroxy 1,1-dioxides
US3927002A (en) * 1973-04-23 1975-12-16 Pfizer N-(pyridyl)-N{40 -alkyl-N{40 -(2-alkoxycarbonylbenzenesulfonyl)-glycineamides and derivatives
US3853862A (en) * 1973-04-23 1974-12-10 Pfizer Production of 4-hydroxy-1,2-benzothiazine-3-carboxamides
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US3891637A (en) * 1974-10-01 1975-06-24 Pfizer Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides
DE2539112C2 (de) * 1975-09-03 1983-12-15 Dr. Karl Thomae Gmbh, 7950 Biberach 4-Hydroxy-2H-naphtho[2,1-e]-1,2-thiazin-3-carboxamid-1,1-dioxide, Verfahren zu ihrer Herstellung und diese enthaltende Arzneimittel
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US4474955A (en) * 1981-06-17 1984-10-02 Vincenzo Iannella Process for preparing 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-[N-(2-pyridinyl)carboxamide]-1,1-dioxide, and its phosphoric ester
GT198276334A (es) * 1981-08-03 1984-01-10 Procedimiento e inter-medios para la produccion de carboxamidas de benzotiazina.
IN159273B (fr) * 1981-10-05 1987-04-25 Pfizer
CA1197244A (fr) * 1982-04-16 1985-11-26 Medichem, S.A. Methode de preparation de 4-hydroxy-2-methyl- 2h-1,2-benzothiazine-3-carboxamide-1,1-dioxydes
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JPS59179683U (ja) * 1983-05-19 1984-11-30 寺田毛織株式会社 貼り合わせふとん
GR80576B (en) * 1983-10-17 1984-11-29 Fujisawa Pharmaceutical Co Thiazine derivatives, process for preparation thereof and pharmaceutical composition comprising the same
US4551452A (en) * 1983-12-21 1985-11-05 Pfizer Inc. Anti-inflammatory 2-methyl-2H-1,2-benzo-(or -thieno-)thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US4656265A (en) * 1984-06-21 1987-04-07 Pfizer Inc. Cyclic prodrugs of antiinflammatory oxicams
DE3437232A1 (de) * 1984-10-10 1986-04-17 Mack Chem Pharm Stabilisierte injektionsloesungen von piroxicam
US4582831A (en) * 1984-11-16 1986-04-15 Pfizer Inc. Anti-inflammatory polymorphic monoethanolamine salt of N-(2-pyridyl)-2-methyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide compound, composition, and method of use therefor
CH663899A5 (fr) * 1985-03-20 1988-01-29 Nestle Sa Procede pour la preparation d'une composition a base d'un principe actif de faible hydrosolubilite finement divise.
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US4610982A (en) * 1985-06-03 1986-09-09 Pfizer Inc. Anti-inflammatory benzo- and thieno-1,2-thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US4761424A (en) * 1985-10-01 1988-08-02 Warner-Lambert Company Enolamides, pharmaceutical compositions and methods for treating inflammation
US4829062A (en) * 1986-05-16 1989-05-09 Pfizer Inc. Benzothiazine dioxide derivatives
EP0259085B1 (fr) * 1986-08-29 1991-08-21 Pfizer Inc. Guanidino-2 aryl-4 thiazole pour le traitement de l'ulcère peptique
US5196410A (en) * 1986-10-31 1993-03-23 Pfizer Inc. Transdermal flux enhancing compositions
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US5081118A (en) * 1987-10-26 1992-01-14 Pfizer Inc. Benzothiazine dioxide derivatives
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HU200926B (en) * 1988-10-28 1990-09-28 Egyt Gyogyszervegyeszeti Gyar Pharmaceutical composition comprising piroxicam and lactose for use in making tablets or capsules
JPH0717589B2 (ja) * 1990-01-22 1995-03-01 ファイザー製薬株式会社 新規１，３―ジカルボニル化合物およびその組成物
JP2988739B2 (ja) * 1990-04-16 1999-12-13 協和醗酵工業株式会社 １，８−ナフチリジン−２−オン誘導体
DE4141218A1 (de) * 1991-12-13 1993-06-17 Luitpold Werk Chem Pharm Thiadiazincarbonsaeureamidderivate, verfahren zu ihrer herstellung und arzneimittel
JP2964195B2 (ja) * 1992-04-28 1999-10-18 エスエス製薬株式会社 ピロキシカム錠及びその製造法
US5362758A (en) * 1992-09-18 1994-11-08 Pfizer Inc. Ophthalmic piroxicam solution
US5420124A (en) * 1994-01-12 1995-05-30 Kim; Young S. Stable, painless piroxicam potassium injectable composition
US5436241A (en) * 1994-01-14 1995-07-25 Bristol-Myers Squibb Company Topical anti-inflammatory compositions containing piroxicam
WO1997046532A1 (fr) * 1996-06-03 1997-12-11 Boehringer Ingelheim Pharmaceuticals, Inc. 2-benzyl-4-sulfonyl-4h-isoquinoline-1,3-diones et leur utilisation comme agents anti-inflammatoires
US5952328A (en) * 1997-11-12 1999-09-14 Cephalon, Inc. Benzothiazo and related heterocyclic group-containing cysteine and serine protease inhibitors
EP1126838A4 (fr) 1998-10-30 2005-02-16 Nitromed Inc Composes anti-inflammatoires non steroidiens nitroses et nitrosyles, compositions et procedes d'utilisation
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IT1318674B1 (it) * 2000-08-08 2003-08-27 Nicox Sa Faramaci per l'incontinenza.
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US20060047171A1 (en) * 2003-12-22 2006-03-02 Harold Meckler Catalytic hydrogenation of nitriles to produce capsaicinoid derivatives and amine compounds, and methods for purifying and obtaining the polymorphs thereof
US20050222227A1 (en) * 2004-04-01 2005-10-06 Pfizer Inc Oxazole-amine compounds for the treatment of neurodegenerative disorders
JP2009529057A (ja) 2006-03-08 2009-08-13 コートリア・コーポレーシヨン Ｃｏｘ−関連胃損傷を予防するための非−選択的ｃｏｘ阻害剤との組み合わせ療法
FR2942797B1 (fr) * 2009-03-03 2011-04-29 Pf Medicament Derives de benzothiazines, leur preparation et leur application a titre de medicaments
CN101665472B (zh) * 2009-06-15 2011-08-24 威海迪素制药有限公司 2-甲基-3，4-二氢-4-氧代-2h-1，2-苯并噻嗪-3-羧酸乙酯-1,1-二氧化物的制备方法
ITUB20152229A1 (it) * 2015-07-16 2017-01-16 Edmond Pharma Srl Processo per la preparazione di farmaci antiinfiammatori non steroidei della classe oxicam

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1302858B (fr) * 1962-09-21 1972-05-04

Also Published As

Publication number Publication date
BE737962A (fr) 1970-02-26
SE402459B (sv) 1978-07-03
PH10029A (en) 1976-07-13
FR2016455A1 (fr) 1970-05-08
DE1943265B2 (de) 1981-05-14
NO129746B (fr) 1974-05-20
DE1943265A1 (de) 1970-08-13
AT298503B (de) 1972-05-10
IL32836A0 (en) 1969-11-12
US3591584A (en) 1971-07-06
ES370861A1 (es) 1971-07-01
NL6912981A (fr) 1970-03-03
DE1967325B2 (de) 1981-08-13
JPS5142114B1 (fr) 1976-11-13
DK145297B (da) 1982-10-25
AT294113B (de) 1971-11-10
FI51189C (fi) 1976-11-10
DK145297C (da) 1983-03-14
FI51189B (fr) 1976-08-02
DE1943265C3 (de) 1982-02-04
NL157013B (nl) 1978-06-15
BR6911817D0 (pt) 1973-02-13
FR2016455B1 (fr) 1974-02-01
SE373854B (fr) 1975-02-17
GB1257180A (fr) 1971-12-15
IL32836A (en) 1972-08-30
DE1967325C2 (de) 1982-03-18
CH520705A (fr) 1972-03-31
JPS50677B1 (fr) 1975-01-10

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