MY128971A - Solid-state form of celecoxib having enhanced bioavailability - Google Patents

Solid-state form of celecoxib having enhanced bioavailability

Info

Publication number
MY128971A
MY128971A MYPI20005730A MYPI20005730A MY128971A MY 128971 A MY128971 A MY 128971A MY PI20005730 A MYPI20005730 A MY PI20005730A MY PI20005730 A MYPI20005730 A MY PI20005730A MY 128971 A MY128971 A MY 128971A
Authority
MY
Malaysia
Prior art keywords
celecoxib
amorphous
drug substance
composition
solid
Prior art date
Application number
MYPI20005730A
Other languages
English (en)
Inventor
Michael J Hageman
Xiaorong He
Tugrul T Kararli
Lesley A Mackin
Patricia J Miyake
Brian R Rohrs
Kevin J Stefanski
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of MY128971A publication Critical patent/MY128971A/en

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    • C07—ORGANIC CHEMISTRY
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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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MYPI20005730A 1999-12-08 2000-12-06 Solid-state form of celecoxib having enhanced bioavailability MY128971A (en)

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JP4906233B2 (ja) 2002-03-01 2012-03-28 ユニバーシティー オブ サウス フロリダ 少なくとも１種の有効薬剤成分を含有する多構成要素固相
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CN103524416B (zh) * 2013-10-29 2016-08-17 湖北华世通生物医药科技有限公司 一种塞来昔布新晶型a及其制备方法
CN103539739B (zh) * 2013-10-30 2016-02-10 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型b及其制备方法
CN103508958A (zh) * 2013-10-30 2014-01-15 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型c及其制备方法
KR101476096B1 (ko) * 2014-03-28 2014-12-24 대원제약주식회사 용해도가 향상된 쎄레콕시브의 약제학적 조성물

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EA200401397A1 (ru) 2005-08-25
TWI276435B (en) 2007-03-21
NZ529933A (en) 2005-06-24
OA11831A (en) 2005-08-23
ZA200107149B (en) 2003-02-28
CO5251445A1 (es) 2003-02-28
KR20020002386A (ko) 2002-01-09
ES2236011T3 (es) 2005-07-16
HUP0200580A2 (hu) 2002-11-28
MY128366A (en) 2007-01-31
PE20010911A1 (es) 2001-09-10
KR100717570B1 (ko) 2007-05-15
SV2002000235A (es) 2002-06-13
BG105808A (bg) 2002-09-30
CN1411447A (zh) 2003-04-16
BG65239B1 (bg) 2007-09-28
PT1150959E (pt) 2008-04-21
AU2041201A (en) 2001-06-18
WO2001041536A2 (en) 2001-06-14
ECSP003807A (es) 2005-07-06
AR030039A1 (es) 2003-08-13
PT1150960E (pt) 2005-06-30
ZA200107146B (en) 2002-08-29
CZ20012875A3 (cs) 2002-02-13
YU57801A (sh) 2005-07-19
CN1216869C (zh) 2005-08-31
HUP0200580A3 (en) 2002-12-28
AR027897A1 (es) 2003-04-16

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