MX375960B - Proceso para la preparacion de pirazoles. - Google Patents

Proceso para la preparacion de pirazoles.

Info

Publication number
MX375960B
MX375960B MX2017001462A MX2017001462A MX375960B MX 375960 B MX375960 B MX 375960B MX 2017001462 A MX2017001462 A MX 2017001462A MX 2017001462 A MX2017001462 A MX 2017001462A MX 375960 B MX375960 B MX 375960B
Authority
MX
Mexico
Prior art keywords
formula
pyrazole
preparation
reagent
compounds
Prior art date
Application number
MX2017001462A
Other languages
English (en)
Other versions
MX2017001462A (es
Inventor
Birgit Gockel
Daniel Sälinger
Michael Rack
Sebastian Sörgel
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of MX2017001462A publication Critical patent/MX2017001462A/es
Publication of MX375960B publication Critical patent/MX375960B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Plant Pathology (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención se refiere a un proceso para la preparación de un compuesto de pirazol de la fórmula V, que comprende la ciclación de un compuesto de carbonilo a,ß-insaturado sustituido por hidrazona de la fórmula IV por medio de la reacción con un reactivo adecuado, por ej., un agente reductor, un reactivo organometálico o un reactivo nucleófilo. Los compuestos de la fórmula y son herramientas versátiles de reacción para la preparación de productos químicos finos derivados de pirazol. La presente invención también se refiere a compuestos de pirazol de las fórmulas Va, Vb, Vc, y VI.
MX2017001462A 2014-07-31 2015-07-30 Proceso para la preparacion de pirazoles. MX375960B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14179249 2014-07-31
PCT/EP2015/067507 WO2016016369A1 (en) 2014-07-31 2015-07-30 Process for preparing pyrazoles

Publications (2)

Publication Number Publication Date
MX2017001462A MX2017001462A (es) 2017-05-23
MX375960B true MX375960B (es) 2025-03-06

Family

ID=51257363

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2017001462A MX375960B (es) 2014-07-31 2015-07-30 Proceso para la preparacion de pirazoles.

Country Status (19)

Country Link
US (2) US10414733B2 (es)
EP (1) EP3174858B1 (es)
JP (1) JP6625610B2 (es)
KR (1) KR102531217B1 (es)
CN (1) CN106573893B (es)
AU (1) AU2015295287B2 (es)
BR (1) BR112016030863B1 (es)
CA (1) CA2954212C (es)
DK (1) DK3174858T3 (es)
ES (1) ES2741831T3 (es)
IL (1) IL249730B (es)
MX (1) MX375960B (es)
PL (1) PL3174858T3 (es)
PT (1) PT3174858T (es)
RU (1) RU2712192C2 (es)
TR (1) TR201909606T4 (es)
UA (1) UA121395C2 (es)
WO (1) WO2016016369A1 (es)
ZA (1) ZA201701415B (es)

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Also Published As

Publication number Publication date
AU2015295287B2 (en) 2019-07-04
ES2741831T3 (es) 2020-02-12
US20180086715A9 (en) 2018-03-29
CN106573893B (zh) 2020-06-09
JP2017522342A (ja) 2017-08-10
CN106573893A (zh) 2017-04-19
EP3174858B1 (en) 2019-04-17
US10414733B2 (en) 2019-09-17
KR102531217B1 (ko) 2023-05-10
JP6625610B2 (ja) 2019-12-25
TR201909606T4 (tr) 2019-07-22
RU2017106265A (ru) 2018-08-30
PT3174858T (pt) 2019-07-23
CA2954212A1 (en) 2016-02-04
MX2017001462A (es) 2017-05-23
US10513498B2 (en) 2019-12-24
ZA201701415B (en) 2019-06-26
RU2712192C2 (ru) 2020-01-24
US20170210712A1 (en) 2017-07-27
CA2954212C (en) 2023-09-19
BR112016030863B1 (pt) 2021-05-04
PL3174858T3 (pl) 2019-10-31
RU2017106265A3 (es) 2019-02-25
DK3174858T3 (da) 2019-07-15
UA121395C2 (uk) 2020-05-25
IL249730B (en) 2019-12-31
WO2016016369A1 (en) 2016-02-04
EP3174858A1 (en) 2017-06-07
IL249730A0 (en) 2017-02-28
AU2015295287A1 (en) 2017-02-16
US20190194141A1 (en) 2019-06-27
KR20170036094A (ko) 2017-03-31

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