MX373658B - Derivado de acido 4-(4-(4-fenilureido-naftalen-1-il)oxi-piridin-2-il)amino-benzoico como inhibidor de quinasa p38. - Google Patents

Derivado de acido 4-(4-(4-fenilureido-naftalen-1-il)oxi-piridin-2-il)amino-benzoico como inhibidor de quinasa p38.

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Publication number
MX373658B
MX373658B MX2017004129A MX2017004129A MX373658B MX 373658 B MX373658 B MX 373658B MX 2017004129 A MX2017004129 A MX 2017004129A MX 2017004129 A MX2017004129 A MX 2017004129A MX 373658 B MX373658 B MX 373658B
Authority
MX
Mexico
Prior art keywords
phenylureido
naphthalen
pyridin
oxy
amino
Prior art date
Application number
MX2017004129A
Other languages
English (en)
Spanish (es)
Other versions
MX2017004129A (es
Inventor
Matthew Colin Thor Fyfe
Original Assignee
Topivert Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1417344.7A external-priority patent/GB201417344D0/en
Priority claimed from GBGB1510694.1A external-priority patent/GB201510694D0/en
Application filed by Topivert Pharma Ltd filed Critical Topivert Pharma Ltd
Publication of MX2017004129A publication Critical patent/MX2017004129A/es
Publication of MX373658B publication Critical patent/MX373658B/es

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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MX2017004129A 2014-10-01 2015-10-01 Derivado de acido 4-(4-(4-fenilureido-naftalen-1-il)oxi-piridin-2-il)amino-benzoico como inhibidor de quinasa p38. MX373658B (es)

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PCT/GB2015/052877 WO2016051188A1 (en) 2014-10-01 2015-10-01 4-(4-(4-phenylureido-naphthalen-1-yl)oxy-pyridin-2-yl)amino-benzoic acid derivative as p38 kinase inhibitor

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US20190330155A1 (en) 2019-10-31
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US20180319748A1 (en) 2018-11-08
CN106999478A (zh) 2017-08-01
AU2015326614A1 (en) 2017-05-04
US20160096805A1 (en) 2016-04-07
EA035478B1 (ru) 2020-06-23
MA40775A (fr) 2017-08-08
MX2017004129A (es) 2017-07-07
CN107001274A (zh) 2017-08-01
US9751837B2 (en) 2017-09-05
US20170253563A1 (en) 2017-09-07
KR20170057445A (ko) 2017-05-24
US20160102059A1 (en) 2016-04-14
US10941115B2 (en) 2021-03-09
JP2017533895A (ja) 2017-11-16
WO2016051187A1 (en) 2016-04-07
CA2961870A1 (en) 2016-04-07
US10392346B2 (en) 2019-08-27
BR112017005531A2 (pt) 2017-12-05
EA201790660A1 (ru) 2017-07-31
EA032694B1 (ru) 2019-07-31
MX2017004128A (es) 2017-07-07
MA40774A (fr) 2017-08-08
JP2017535525A (ja) 2017-11-30

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