KR20170063783A - P38 키나제 저해제로서의 4-(4-(4-페닐우레이도나프탈렌-1-일)옥시피리딘-2-일)아미노벤조산 유도체 - Google Patents

P38 키나제 저해제로서의 4-(4-(4-페닐우레이도나프탈렌-1-일)옥시피리딘-2-일)아미노벤조산 유도체 Download PDF

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KR20170063783A
KR20170063783A KR1020177010961A KR20177010961A KR20170063783A KR 20170063783 A KR20170063783 A KR 20170063783A KR 1020177010961 A KR1020177010961 A KR 1020177010961A KR 20177010961 A KR20177010961 A KR 20177010961A KR 20170063783 A KR20170063783 A KR 20170063783A
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compound
formula
cells
pharmaceutically acceptable
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매튜 콜린 토르 파이프
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레스피버트 리미티드
토피버트 파마 리미티드
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Priority claimed from GBGB1417344.7A external-priority patent/GB201417344D0/en
Priority claimed from GBGB1510694.1A external-priority patent/GB201510694D0/en
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Publication of KR20170063783A publication Critical patent/KR20170063783A/ko
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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KR1020177010961A 2014-10-01 2015-10-01 P38 키나제 저해제로서의 4-(4-(4-페닐우레이도나프탈렌-1-일)옥시피리딘-2-일)아미노벤조산 유도체 Withdrawn KR20170063783A (ko)

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GB1510694.1 2015-06-18
PCT/GB2015/052877 WO2016051188A1 (en) 2014-10-01 2015-10-01 4-(4-(4-phenylureido-naphthalen-1-yl)oxy-pyridin-2-yl)amino-benzoic acid derivative as p38 kinase inhibitor

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EP3201189A1 (en) 2014-10-01 2017-08-09 Respivert Limited N-phenyl-3-quinazolin-6-yl-benzamide derivatives as p38 kinase inhibitors

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