MX369358B - Nuevos agonistas del receptor de somatostatina subtipo 4 (sstr4). - Google Patents

Nuevos agonistas del receptor de somatostatina subtipo 4 (sstr4).

Info

Publication number
MX369358B
MX369358B MX2015015620A MX2015015620A MX369358B MX 369358 B MX369358 B MX 369358B MX 2015015620 A MX2015015620 A MX 2015015620A MX 2015015620 A MX2015015620 A MX 2015015620A MX 369358 B MX369358 B MX 369358B
Authority
MX
Mexico
Prior art keywords
sstr4
agonists
receptor subtype
somatostatin receptor
processes
Prior art date
Application number
MX2015015620A
Other languages
English (en)
Spanish (es)
Other versions
MX2015015620A (es
Inventor
Rudolf Klaus
Doods Henri
Kuelzer Raimund
Giovannini Riccardo
Mazzaferro Rocco
Ferrara Marco
Lingard Iain
Cui Yunhai
Just Stefan
Original Assignee
Centrexion Therapeutics Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centrexion Therapeutics Corp filed Critical Centrexion Therapeutics Corp
Publication of MX2015015620A publication Critical patent/MX2015015620A/es
Publication of MX369358B publication Critical patent/MX369358B/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
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MX2015015620A 2013-05-17 2014-05-15 Nuevos agonistas del receptor de somatostatina subtipo 4 (sstr4). MX369358B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP13168224 2013-05-17
PCT/EP2014/059905 WO2014184275A1 (en) 2013-05-17 2014-05-15 New somatostatin receptor subtype 4 (sstr4) agonists

Publications (2)

Publication Number Publication Date
MX2015015620A MX2015015620A (es) 2016-03-07
MX369358B true MX369358B (es) 2019-11-06

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MX2015015620A MX369358B (es) 2013-05-17 2014-05-15 Nuevos agonistas del receptor de somatostatina subtipo 4 (sstr4).

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