MX354423B - Formulaciones de rasagilina de liberación prolongada y usos de las mismas. - Google Patents

Formulaciones de rasagilina de liberación prolongada y usos de las mismas.

Info

Publication number
MX354423B
MX354423B MX2012009079A MX2012009079A MX354423B MX 354423 B MX354423 B MX 354423B MX 2012009079 A MX2012009079 A MX 2012009079A MX 2012009079 A MX2012009079 A MX 2012009079A MX 354423 B MX354423 B MX 354423B
Authority
MX
Mexico
Prior art keywords
rasagiline
extended release
release formulations
pharmaceutically acceptable
acceptable salt
Prior art date
Application number
MX2012009079A
Other languages
English (en)
Spanish (es)
Other versions
MX2012009079A (es
Inventor
Yoram Sela
Itschak Lamensdorf
Nurit Livnah
Tomer Madmon
Original Assignee
Pharma Two B Ltd Star
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43896855&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX354423(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharma Two B Ltd Star filed Critical Pharma Two B Ltd Star
Publication of MX2012009079A publication Critical patent/MX2012009079A/es
Publication of MX354423B publication Critical patent/MX354423B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
MX2012009079A 2010-02-03 2011-02-03 Formulaciones de rasagilina de liberación prolongada y usos de las mismas. MX354423B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30101910P 2010-02-03 2010-02-03
PCT/IL2011/000126 WO2011095973A1 (en) 2010-02-03 2011-02-03 Extended release formulations of rasagiline and uses thereof

Publications (2)

Publication Number Publication Date
MX2012009079A MX2012009079A (es) 2012-12-17
MX354423B true MX354423B (es) 2018-03-02

Family

ID=43896855

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012009079A MX354423B (es) 2010-02-03 2011-02-03 Formulaciones de rasagilina de liberación prolongada y usos de las mismas.

Country Status (25)

Country Link
US (1) US9943489B2 (https=)
EP (2) EP2531181B1 (https=)
JP (3) JP6045347B2 (https=)
KR (1) KR101791715B1 (https=)
CN (1) CN102791258B (https=)
AU (1) AU2011212068B2 (https=)
BR (1) BR112012019374B1 (https=)
CA (1) CA2789006C (https=)
CL (1) CL2012002175A1 (https=)
CY (1) CY1121781T1 (https=)
DK (1) DK2531181T3 (https=)
ES (1) ES2733133T3 (https=)
HU (1) HUE044221T2 (https=)
IL (1) IL221274A (https=)
LT (1) LT2531181T (https=)
MX (1) MX354423B (https=)
NZ (1) NZ602111A (https=)
PL (1) PL2531181T3 (https=)
PT (1) PT2531181T (https=)
RS (1) RS58988B1 (https=)
RU (2) RU2734632C2 (https=)
SG (1) SG183150A1 (https=)
TR (1) TR201909277T4 (https=)
WO (1) WO2011095973A1 (https=)
ZA (1) ZA201206462B (https=)

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JP6045347B2 (ja) * 2010-02-03 2016-12-14 ファーマ ツー ビー リミテッド ラサギリンの持続放出性製剤およびその使用
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LT2802319T (lt) * 2012-01-12 2018-04-10 Pharma Two B Ltd. Fiksuotos dozės derinio terapija, skirta parkinsono ligai gydyti
US9504657B2 (en) * 2012-01-12 2016-11-29 Pharmatwob Ltd. Fixed dose combination therapy of Parkinson's disease
CN103316026B (zh) 2012-03-23 2016-05-11 中国人民解放军军事医学科学院毒物药物研究所 含芬特明和托吡酯的联合产品及其制备方法
CN102579367B (zh) * 2012-03-23 2014-03-12 中国人民解放军军事医学科学院毒物药物研究所 托吡酯缓释药物组合物、其制备方法及用途
WO2013139292A1 (zh) 2012-03-23 2013-09-26 中国人民解放军军事医学科学院毒物药物研究所 一种含辛弗林和托吡酯的联合产品
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CN107049985B (zh) * 2017-06-07 2020-06-19 广州帝奇医药技术有限公司 一种抗帕金森病药物的长效缓释制剂及其制备方法
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CA3119361A1 (en) 2018-11-19 2020-05-28 Supernus Pharmaceuticals, Inc. Use of higher doses of modified release huperzine formulations
TWI859242B (zh) * 2019-05-31 2024-10-21 美商戴納立製藥公司 嘧啶基胺基-吡唑化合物之修飾釋放調配物及治療方法
KR20210014289A (ko) 2019-07-30 2021-02-09 (주)비씨월드제약 라사길린을 함유하는 서방출성 미립구의 제조방법
AR121619A1 (es) * 2020-03-25 2022-06-22 Inibsa Ginecologia S A Una forma de dosificación oral de múltiples unidades de liberación modificada de succinato de doxilamina y clorhidrato de piridoxina y un procedimiento para su preparación
CN117355296A (zh) * 2021-05-11 2024-01-05 阿德维斯尼公司 用于口服施用舒噻美的延长释放药物组合物
EP4337176B1 (en) * 2021-05-11 2025-07-16 Advicenne Prolonged-release pharmaceutical composition for oral administration of sultiame
CN118680910B (zh) * 2024-08-26 2024-12-03 山东齐都药业有限公司 用于缓释递送雷沙吉兰甲磺酸盐的药物组合物及其制备方法和应用

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Also Published As

Publication number Publication date
AU2011212068A1 (en) 2012-09-20
CA2789006A1 (en) 2011-08-11
US20120301542A1 (en) 2012-11-29
US9943489B2 (en) 2018-04-17
RU2607595C2 (ru) 2017-01-10
SG183150A1 (en) 2012-09-27
CN102791258A (zh) 2012-11-21
JP6045347B2 (ja) 2016-12-14
IL221274A (en) 2017-05-29
JP2013518870A (ja) 2013-05-23
NZ602111A (en) 2014-10-31
CY1121781T1 (el) 2020-07-31
TR201909277T4 (tr) 2019-07-22
MX2012009079A (es) 2012-12-17
EP2531181A1 (en) 2012-12-12
RU2016141314A3 (https=) 2019-12-20
JP2019048855A (ja) 2019-03-28
PT2531181T (pt) 2019-07-17
WO2011095973A1 (en) 2011-08-11
IL221274A0 (en) 2012-10-31
EP3517103A1 (en) 2019-07-31
LT2531181T (lt) 2019-07-10
HUE044221T2 (hu) 2019-10-28
RU2016141314A (ru) 2018-12-14
PL2531181T3 (pl) 2019-09-30
RU2734632C2 (ru) 2020-10-21
KR20120130292A (ko) 2012-11-30
ES2733133T3 (es) 2019-11-27
RU2012136723A (ru) 2014-03-10
CA2789006C (en) 2018-11-27
AU2011212068B2 (en) 2016-08-18
KR101791715B1 (ko) 2017-10-30
EP2531181B1 (en) 2019-04-10
JP2017031189A (ja) 2017-02-09
JP6440662B2 (ja) 2018-12-19
ZA201206462B (en) 2014-02-26
CL2012002175A1 (es) 2013-01-11
RS58988B1 (sr) 2019-08-30
BR112012019374B1 (pt) 2022-01-11
BR112012019374A2 (pt) 2016-05-03
DK2531181T3 (da) 2019-07-15
JP6770564B2 (ja) 2020-10-14
CN102791258B (zh) 2018-05-08

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