DK2531181T3 - Formuleringer af rasagilin med forlænget afgivelse og anvendelser deraf - Google Patents

Formuleringer af rasagilin med forlænget afgivelse og anvendelser deraf Download PDF

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Publication number
DK2531181T3
DK2531181T3 DK11707489.8T DK11707489T DK2531181T3 DK 2531181 T3 DK2531181 T3 DK 2531181T3 DK 11707489 T DK11707489 T DK 11707489T DK 2531181 T3 DK2531181 T3 DK 2531181T3
Authority
DK
Denmark
Prior art keywords
rasagilin
formulations
extended delivery
delivery
extended
Prior art date
Application number
DK11707489.8T
Other languages
English (en)
Inventor
Yoram Sela
Nurit Livnah
Tomer Madmon
Itschak Lamensdorf
Original Assignee
Pharma Two B Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43896855&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2531181(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharma Two B Ltd filed Critical Pharma Two B Ltd
Application granted granted Critical
Publication of DK2531181T3 publication Critical patent/DK2531181T3/da

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK11707489.8T 2010-02-03 2011-02-03 Formuleringer af rasagilin med forlænget afgivelse og anvendelser deraf DK2531181T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30101910P 2010-02-03 2010-02-03
PCT/IL2011/000126 WO2011095973A1 (en) 2010-02-03 2011-02-03 Extended release formulations of rasagiline and uses thereof

Publications (1)

Publication Number Publication Date
DK2531181T3 true DK2531181T3 (da) 2019-07-15

Family

ID=43896855

Family Applications (1)

Application Number Title Priority Date Filing Date
DK11707489.8T DK2531181T3 (da) 2010-02-03 2011-02-03 Formuleringer af rasagilin med forlænget afgivelse og anvendelser deraf

Country Status (25)

Country Link
US (1) US9943489B2 (da)
EP (2) EP2531181B1 (da)
JP (3) JP6045347B2 (da)
KR (1) KR101791715B1 (da)
CN (1) CN102791258B (da)
AU (1) AU2011212068B2 (da)
BR (1) BR112012019374B1 (da)
CA (1) CA2789006C (da)
CL (1) CL2012002175A1 (da)
CY (1) CY1121781T1 (da)
DK (1) DK2531181T3 (da)
ES (1) ES2733133T3 (da)
HU (1) HUE044221T2 (da)
IL (1) IL221274A (da)
LT (1) LT2531181T (da)
MX (1) MX354423B (da)
NZ (1) NZ602111A (da)
PL (1) PL2531181T3 (da)
PT (1) PT2531181T (da)
RS (1) RS58988B1 (da)
RU (2) RU2734632C2 (da)
SG (1) SG183150A1 (da)
TR (1) TR201909277T4 (da)
WO (1) WO2011095973A1 (da)
ZA (1) ZA201206462B (da)

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US9504657B2 (en) * 2012-01-12 2016-11-29 Pharmatwob Ltd. Fixed dose combination therapy of Parkinson's disease
CN103316026B (zh) 2012-03-23 2016-05-11 中国人民解放军军事医学科学院毒物药物研究所 含芬特明和托吡酯的联合产品及其制备方法
EP2829270B1 (en) 2012-03-23 2020-11-11 Institute of Pharmacology and Toxicology Academy of Military Medical Sciences P.L.A. China Joint product containing synephrine and topiramate
CN102579367B (zh) * 2012-03-23 2014-03-12 中国人民解放军军事医学科学院毒物药物研究所 托吡酯缓释药物组合物、其制备方法及用途
AR092168A1 (es) * 2012-08-17 2015-03-25 Teva Pharma Formulaciones parenterales de rasagilina
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US20180333365A1 (en) * 2017-05-19 2018-11-22 Biscayne Neurotherapeutics, Inc. Modified release pharmaceutical compositions of huperzine and methods of using the same
CN107049985B (zh) * 2017-06-07 2020-06-19 广州帝奇医药技术有限公司 一种抗帕金森病药物的长效缓释制剂及其制备方法
KR20210014289A (ko) 2019-07-30 2021-02-09 (주)비씨월드제약 라사길린을 함유하는 서방출성 미립구의 제조방법
WO2022238401A1 (en) * 2021-05-11 2022-11-17 Advicenne Prolonged-release pharmaceutical composition for oral administration of sultiame

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Also Published As

Publication number Publication date
EP2531181B1 (en) 2019-04-10
PL2531181T3 (pl) 2019-09-30
BR112012019374A2 (pt) 2016-05-03
MX354423B (es) 2018-03-02
KR20120130292A (ko) 2012-11-30
IL221274A (en) 2017-05-29
RU2012136723A (ru) 2014-03-10
JP6045347B2 (ja) 2016-12-14
RS58988B1 (sr) 2019-08-30
US20120301542A1 (en) 2012-11-29
WO2011095973A1 (en) 2011-08-11
ZA201206462B (en) 2014-02-26
CA2789006C (en) 2018-11-27
JP2019048855A (ja) 2019-03-28
NZ602111A (en) 2014-10-31
LT2531181T (lt) 2019-07-10
CN102791258A (zh) 2012-11-21
CY1121781T1 (el) 2020-07-31
TR201909277T4 (tr) 2019-07-22
CL2012002175A1 (es) 2013-01-11
US9943489B2 (en) 2018-04-17
HUE044221T2 (hu) 2019-10-28
SG183150A1 (en) 2012-09-27
IL221274A0 (en) 2012-10-31
CA2789006A1 (en) 2011-08-11
EP2531181A1 (en) 2012-12-12
KR101791715B1 (ko) 2017-10-30
JP2013518870A (ja) 2013-05-23
RU2016141314A (ru) 2018-12-14
JP6440662B2 (ja) 2018-12-19
JP6770564B2 (ja) 2020-10-14
EP3517103A1 (en) 2019-07-31
JP2017031189A (ja) 2017-02-09
PT2531181T (pt) 2019-07-17
MX2012009079A (es) 2012-12-17
ES2733133T3 (es) 2019-11-27
AU2011212068B2 (en) 2016-08-18
RU2016141314A3 (da) 2019-12-20
CN102791258B (zh) 2018-05-08
RU2734632C2 (ru) 2020-10-21
AU2011212068A1 (en) 2012-09-20
RU2607595C2 (ru) 2017-01-10
BR112012019374B1 (pt) 2022-01-11

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