MX351368B - Compuestos heteroarilo y metodos para utilizarlos. - Google Patents
Compuestos heteroarilo y metodos para utilizarlos.Info
- Publication number
- MX351368B MX351368B MX2012013624A MX2012013624A MX351368B MX 351368 B MX351368 B MX 351368B MX 2012013624 A MX2012013624 A MX 2012013624A MX 2012013624 A MX2012013624 A MX 2012013624A MX 351368 B MX351368 B MX 351368B
- Authority
- MX
- Mexico
- Prior art keywords
- methods
- compounds
- disorders
- heteroaryl compounds
- heteroaryl
- Prior art date
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/06—Peri-condensed systems
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- Otolaryngology (AREA)
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- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34868310P | 2010-05-26 | 2010-05-26 | |
| US41141010P | 2010-11-08 | 2010-11-08 | |
| PCT/US2011/038057 WO2011150156A2 (en) | 2010-05-26 | 2011-05-26 | Heteroaryl compounds and methods of use thereof |
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| WO2011053559A1 (en) * | 2009-10-30 | 2011-05-05 | Merck Sharp & Dohme Corp. | Aryl aminopyridine pde10 inhibitors |
| TWI485151B (zh) | 2009-12-17 | 2015-05-21 | Lundbeck & Co As H | 作為pde10a酵素抑制劑之雜芳香族苯基咪唑衍生物 |
| WO2011122815A2 (en) * | 2010-03-29 | 2011-10-06 | Dong-A Pharm.Co.,Ltd. | Novel quinoxaline derivatives |
| NZ603789A (en) | 2010-05-26 | 2015-03-27 | Sunovion Pharmaceuticals Inc | Heteroaryl compounds and methods of use thereof |
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2011
- 2011-05-26 NZ NZ60378911A patent/NZ603789A/en not_active IP Right Cessation
- 2011-05-26 EP EP17205058.5A patent/EP3318561B1/en not_active Not-in-force
- 2011-05-26 US US13/700,051 patent/US8969349B2/en active Active
- 2011-05-26 MX MX2012013624A patent/MX351368B/es active IP Right Grant
- 2011-05-26 AU AU2011258217A patent/AU2011258217B2/en not_active Ceased
- 2011-05-26 WO PCT/US2011/038057 patent/WO2011150156A2/en not_active Ceased
- 2011-05-26 CA CA2800618A patent/CA2800618C/en active Active
- 2011-05-26 JP JP2013512231A patent/JP5911476B2/ja not_active Expired - Fee Related
- 2011-05-26 CN CN201180036842.7A patent/CN103038229B/zh not_active Expired - Fee Related
- 2011-05-26 NZ NZ705135A patent/NZ705135A/en not_active IP Right Cessation
- 2011-05-26 EP EP11787386.9A patent/EP2576540B1/en active Active
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2012
- 2012-11-25 IL IL223240A patent/IL223240B/en active IP Right Grant
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2015
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- 2015-09-29 JP JP2015191866A patent/JP2016028092A/ja active Pending
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2017
- 2017-10-19 US US15/787,880 patent/US10562916B2/en active Active
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| Publication number | Publication date |
|---|---|
| US10562916B2 (en) | 2020-02-18 |
| US20180037590A1 (en) | 2018-02-08 |
| EP2576540B1 (en) | 2019-09-04 |
| MX2012013624A (es) | 2013-02-11 |
| NZ705135A (en) | 2017-10-27 |
| US9834564B2 (en) | 2017-12-05 |
| EP2576540A2 (en) | 2013-04-10 |
| JP5911476B2 (ja) | 2016-04-27 |
| WO2011150156A3 (en) | 2012-04-19 |
| IL223240B (en) | 2019-05-30 |
| EP2576540A4 (en) | 2013-12-04 |
| NZ603789A (en) | 2015-03-27 |
| AU2011258217A1 (en) | 2012-12-20 |
| CN103038229B (zh) | 2016-05-11 |
| US20130158003A1 (en) | 2013-06-20 |
| JP2016028092A (ja) | 2016-02-25 |
| WO2011150156A2 (en) | 2011-12-01 |
| EP3318561A1 (en) | 2018-05-09 |
| IL266168A (en) | 2019-06-30 |
| IL223240A0 (en) | 2013-02-03 |
| CA2800618C (en) | 2018-08-28 |
| CN103038229A (zh) | 2013-04-10 |
| CA2800618A1 (en) | 2011-12-01 |
| JP2013526615A (ja) | 2013-06-24 |
| US8969349B2 (en) | 2015-03-03 |
| AU2011258217B2 (en) | 2016-12-15 |
| US20150166571A1 (en) | 2015-06-18 |
| EP3318561B1 (en) | 2021-12-22 |
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