MX337364B - Formulaciones farmaceuticas de azol para la administracion parenteral y metodos para preparar y usar las mismas como tratamiento de las enfermedades sensibles a los compuestos de azol. - Google Patents

Formulaciones farmaceuticas de azol para la administracion parenteral y metodos para preparar y usar las mismas como tratamiento de las enfermedades sensibles a los compuestos de azol.

Info

Publication number
MX337364B
MX337364B MX2013006816A MX2013006816A MX337364B MX 337364 B MX337364 B MX 337364B MX 2013006816 A MX2013006816 A MX 2013006816A MX 2013006816 A MX2013006816 A MX 2013006816A MX 337364 B MX337364 B MX 337364B
Authority
MX
Mexico
Prior art keywords
azole
treatment
water
preparing
methods
Prior art date
Application number
MX2013006816A
Other languages
English (en)
Spanish (es)
Other versions
MX2013006816A (es
Inventor
Borje S Andersson
Jeffery Tarrand
Benigno C Valdez
Original Assignee
Borje S Andersson
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Borje S Andersson filed Critical Borje S Andersson
Publication of MX2013006816A publication Critical patent/MX2013006816A/es
Publication of MX337364B publication Critical patent/MX337364B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/417Imidazole-alkylamines, e.g. histamine, phentolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41961,2,4-Triazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Oncology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
MX2013006816A 2010-12-16 2011-12-16 Formulaciones farmaceuticas de azol para la administracion parenteral y metodos para preparar y usar las mismas como tratamiento de las enfermedades sensibles a los compuestos de azol. MX337364B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US42393710P 2010-12-16 2010-12-16
US201161509154P 2011-07-19 2011-07-19
PCT/US2011/065422 WO2012083138A2 (en) 2010-12-16 2011-12-16 Azole pharmaceutical formulations for parenteral administration and methods for preparing and using the same as treatment of diseases sensitive to azole compounds

Publications (2)

Publication Number Publication Date
MX2013006816A MX2013006816A (es) 2013-11-01
MX337364B true MX337364B (es) 2016-02-29

Family

ID=46245384

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013006816A MX337364B (es) 2010-12-16 2011-12-16 Formulaciones farmaceuticas de azol para la administracion parenteral y metodos para preparar y usar las mismas como tratamiento de las enfermedades sensibles a los compuestos de azol.

Country Status (15)

Country Link
US (2) US10307418B2 (enExample)
EP (1) EP2651450B1 (enExample)
JP (2) JP6086539B2 (enExample)
CN (1) CN103402543B (enExample)
AU (1) AU2011343576B2 (enExample)
BR (1) BR112013015085A8 (enExample)
CA (1) CA2821823C (enExample)
DK (1) DK2651450T3 (enExample)
ES (1) ES2565353T3 (enExample)
HU (1) HUE028667T2 (enExample)
IL (1) IL226977A (enExample)
MX (1) MX337364B (enExample)
NZ (1) NZ613167A (enExample)
RU (2) RU2618456C2 (enExample)
WO (1) WO2012083138A2 (enExample)

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RU2618456C2 (ru) * 2010-12-16 2017-05-03 Плэтформ Брайтворкс Ту, Лтд Фармацевтические препараты азолов для парентерального введения и способы их получения и применения для лечения заболеваний, чувствительных к азольным соединениям
CN103635179B (zh) * 2011-04-28 2017-12-29 普拉福姆五金器具第二有限公司 亲脂性药剂的改进的胃肠外制剂以及制备和使用其的方法
SG11201504976UA (en) * 2012-12-28 2015-07-30 Suntory Holdings Ltd Non-alcohol, beer-taste beverage having shimari in taste
CN105394045B (zh) * 2014-09-04 2020-02-14 中国科学院上海巴斯德研究所 一种肠道病毒的小分子化合物抑制剂及其应用
CN105943500B (zh) * 2016-07-08 2019-01-04 河南省立眼科医院 一种含有艾沙康唑的眼用纳米胶束抗真菌溶液
TWI834808B (zh) * 2019-02-19 2024-03-11 西班牙商薩爾瓦特實驗室有限公司 以單劑包裝的克氯黴唑液體組成物
CN111665301A (zh) * 2020-05-29 2020-09-15 南京品生医疗科技有限公司 超高效液相色谱串联质谱技术检测血清中抗真菌药物的试剂盒
AU2021379990A1 (en) * 2020-11-16 2023-06-29 W. L. Gore & Associates, Inc. Formulations, methods, and pre-filled multi-dose injection devices without cloud point
CN113671086B (zh) * 2021-08-31 2023-06-16 重庆华邦制药有限公司 分离、测定泊沙康唑z2及其杂质的方法
CN114660200A (zh) * 2022-03-29 2022-06-24 中国人民解放军总医院 一种高效液相色谱串联质谱技术同时测定血浆中4种三唑类抗真菌药物的方法

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DE3702105A1 (de) 1987-01-24 1988-08-04 Bayer Ag Parenterale loesung
JPH01242525A (ja) 1988-03-25 1989-09-27 Nippon Nohyaku Co Ltd 抗真菌外用剤
PH30929A (en) * 1992-09-03 1997-12-23 Janssen Pharmaceutica Nv Beads having a core coated with an antifungal and a polymer.
TW349870B (en) * 1993-09-30 1999-01-11 Janssen Pharmaceutica Nv An antifungal pharmaceutical composition for oral administration and a process for the preparation thereof
KR0159730B1 (ko) * 1996-01-15 1998-12-01 손경식 케토코나졸 수성 제제
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US6362172B2 (en) * 2000-01-20 2002-03-26 Bristol-Myers Squibb Company Water soluble prodrugs of azole compounds
GB2365770B (en) * 2000-08-18 2002-07-31 Diomed Dev Ltd Antifungal ketoconazole composition for topical use
US20050048126A1 (en) * 2000-12-22 2005-03-03 Barrett Rabinow Formulation to render an antimicrobial drug potent against organisms normally considered to be resistant to the drug
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JP2002322056A (ja) * 2001-04-27 2002-11-08 Nippon Kayaku Co Ltd トリアゾール誘導体の溶液製剤
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WO2004014431A1 (en) * 2002-08-12 2004-02-19 Ranbaxy Laboratories Limited A parenteral dosage form of selective cox-2 inhibitors
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CN103635179B (zh) * 2011-04-28 2017-12-29 普拉福姆五金器具第二有限公司 亲脂性药剂的改进的胃肠外制剂以及制备和使用其的方法

Also Published As

Publication number Publication date
EP2651450B1 (en) 2015-12-16
ES2565353T3 (es) 2016-04-04
CA2821823C (en) 2019-05-07
US20140031366A1 (en) 2014-01-30
CN103402543A (zh) 2013-11-20
HK1190643A1 (zh) 2014-07-11
WO2012083138A3 (en) 2012-11-01
NZ613167A (en) 2015-09-25
CN103402543B (zh) 2015-09-16
RU2734128C2 (ru) 2020-10-13
RU2013132703A (ru) 2015-01-27
JP6086539B2 (ja) 2017-03-01
AU2011343576B2 (en) 2016-09-08
AU2011343576A1 (en) 2013-07-11
WO2012083138A2 (en) 2012-06-21
BR112013015085A8 (pt) 2018-04-03
EP2651450A2 (en) 2013-10-23
RU2016149770A (ru) 2018-11-05
US20190240216A1 (en) 2019-08-08
CA2821823A1 (en) 2012-06-21
JP2013545819A (ja) 2013-12-26
DK2651450T3 (en) 2016-03-14
IL226977A (en) 2017-01-31
BR112013015085A2 (pt) 2016-08-09
JP6529527B2 (ja) 2019-06-12
RU2016149770A3 (enExample) 2020-02-04
US10307418B2 (en) 2019-06-04
HUE028667T2 (en) 2016-12-28
RU2618456C2 (ru) 2017-05-03
EP2651450A4 (en) 2014-07-09
JP2017114869A (ja) 2017-06-29
MX2013006816A (es) 2013-11-01

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