MX336789B - Farmacos resistentes al abuso, metodo de uso y metodo de fabricacion. - Google Patents
Farmacos resistentes al abuso, metodo de uso y metodo de fabricacion.Info
- Publication number
- MX336789B MX336789B MX2010001812A MX2010001812A MX336789B MX 336789 B MX336789 B MX 336789B MX 2010001812 A MX2010001812 A MX 2010001812A MX 2010001812 A MX2010001812 A MX 2010001812A MX 336789 B MX336789 B MX 336789B
- Authority
- MX
- Mexico
- Prior art keywords
- layer
- polymer
- making
- barrier layer
- abuse resistant
- Prior art date
Links
Classifications
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- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Abstract
Una composición farmacéutica oral resistente al abuso, la cual comprende: una capa de barrera que comprende un primer polímero; una capa de difusión que comprende un segundo polímero, la cual cubre sustancialmente a la capa de barrera, en donde la capa de difusión se enlaza a la capa de barrera y comprende un fármaco que se distribuye de una manera sustancialmente homogénea dentro del segundo polímero y se difunde desde la capa de difusión dentro del tracto gastrointestinal (GI); y opcionalmente una capa de expansión que comprende un polímero expandible, en donde la capa de expansión es sustancialmente cubierta por la capa de barrera. Los métodos de fabricación de la misma y los métodos de uso de la misma también se proporcionan.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US95558407P | 2007-08-13 | 2007-08-13 | |
PCT/US2008/072914 WO2009023672A2 (en) | 2007-08-13 | 2008-08-12 | Abuse resistant drugs, method of use and method of making |
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MX2010001812A MX2010001812A (es) | 2010-08-04 |
MX336789B true MX336789B (es) | 2016-02-02 |
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Application Number | Title | Priority Date | Filing Date |
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MX2010001812A MX336789B (es) | 2007-08-13 | 2008-08-12 | Farmacos resistentes al abuso, metodo de uso y metodo de fabricacion. |
Country Status (11)
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US (23) | US10736850B2 (es) |
EP (1) | EP2187873B1 (es) |
JP (2) | JP5965583B2 (es) |
CN (2) | CN105534936B (es) |
AU (4) | AU2008286914B2 (es) |
BR (1) | BRPI0815387B8 (es) |
CA (2) | CA2923102C (es) |
ES (1) | ES2692437T3 (es) |
MX (1) | MX336789B (es) |
PL (1) | PL2187873T3 (es) |
WO (1) | WO2009023672A2 (es) |
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