MX2016001464A - Derivados de tieno[3,2-d]pirimidinas para el tratamiento de infecciones virales. - Google Patents

Derivados de tieno[3,2-d]pirimidinas para el tratamiento de infecciones virales.

Info

Publication number
MX2016001464A
MX2016001464A MX2016001464A MX2016001464A MX2016001464A MX 2016001464 A MX2016001464 A MX 2016001464A MX 2016001464 A MX2016001464 A MX 2016001464A MX 2016001464 A MX2016001464 A MX 2016001464A MX 2016001464 A MX2016001464 A MX 2016001464A
Authority
MX
Mexico
Prior art keywords
thieno
viral infections
treatment
pyrimidines derivatives
pyrimidines
Prior art date
Application number
MX2016001464A
Other languages
English (en)
Other versions
MX368625B (es
Inventor
Pierre Jean-Marie Bernard Raboisson
Gowan David Craig Mc
Original Assignee
Janssen Sciences Ireland Uc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of MX2016001464A publication Critical patent/MX2016001464A/es
Publication of MX368625B publication Critical patent/MX368625B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Esta invención se refiere a derivados de tieno[3,2-d]pirimidinas, procesos para su preparación, composiciones farmacéuticas y su uso en el tratamiento de infecciones virales.
MX2016001464A 2013-07-30 2014-07-29 Derivados de tieno[3,2-d]pirimidinas para el tratamiento de infecciones virales. MX368625B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP13178534 2013-07-30
PCT/EP2014/066219 WO2015014815A1 (en) 2013-07-30 2014-07-29 THIENO[3,2-d]PYRIMIDINES DERIVATIVES FOR THE TREATMENT OF VIRAL INFECTIONS

Publications (2)

Publication Number Publication Date
MX2016001464A true MX2016001464A (es) 2016-06-02
MX368625B MX368625B (es) 2019-10-08

Family

ID=48874951

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016001464A MX368625B (es) 2013-07-30 2014-07-29 Derivados de tieno[3,2-d]pirimidinas para el tratamiento de infecciones virales.

Country Status (21)

Country Link
US (3) US9556199B2 (es)
EP (2) EP3027624B1 (es)
JP (1) JP6401788B2 (es)
KR (1) KR102322425B1 (es)
CN (2) CN105492446B (es)
AU (2) AU2014298540B2 (es)
BR (1) BR112016001570B1 (es)
CA (1) CA2913691C (es)
CL (1) CL2015003767A1 (es)
DK (2) DK3027624T3 (es)
EA (1) EA036162B1 (es)
ES (2) ES2836881T3 (es)
HK (1) HK1217707A1 (es)
IL (2) IL242872B (es)
MX (1) MX368625B (es)
MY (1) MY179503A (es)
PH (1) PH12015502797B1 (es)
SG (2) SG11201510736PA (es)
UA (1) UA117253C2 (es)
WO (1) WO2015014815A1 (es)
ZA (1) ZA201600655B (es)

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LT2872515T (lt) 2012-07-13 2016-10-10 Janssen Sciences Ireland Uc Makrocikliniai purinai, skirti virusinių infekcijų gydymui
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AU2014242954B2 (en) 2013-03-29 2018-03-15 Janssen Sciences Ireland Uc Macrocyclic deaza-purinones for the treatment of viral infections
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