MX2014009033A - Metodo para la sintesis estereoselectiva de 9-hidroxi-5-oxo-1,4-di aza-espiro[5,5]undecanos 1,4-protegidos. - Google Patents
Metodo para la sintesis estereoselectiva de 9-hidroxi-5-oxo-1,4-di aza-espiro[5,5]undecanos 1,4-protegidos.Info
- Publication number
- MX2014009033A MX2014009033A MX2014009033A MX2014009033A MX2014009033A MX 2014009033 A MX2014009033 A MX 2014009033A MX 2014009033 A MX2014009033 A MX 2014009033A MX 2014009033 A MX2014009033 A MX 2014009033A MX 2014009033 A MX2014009033 A MX 2014009033A
- Authority
- MX
- Mexico
- Prior art keywords
- formula
- compound
- tautomers
- salts
- give
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
- C07D491/113—Spiro-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12154688 | 2012-02-09 | ||
| PCT/EP2013/052287 WO2013117568A1 (de) | 2012-02-09 | 2013-02-06 | Verfahren zur stereoselektiven synthese von 1,4-geschützten 9-hydroxy-5-oxo-1,4-diaza-spiro [5.5] undecane |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2014009033A true MX2014009033A (es) | 2014-10-17 |
Family
ID=47678813
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2014009033A MX2014009033A (es) | 2012-02-09 | 2013-02-06 | Metodo para la sintesis estereoselectiva de 9-hidroxi-5-oxo-1,4-di aza-espiro[5,5]undecanos 1,4-protegidos. |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US8629146B2 (https=) |
| EP (1) | EP2812317B1 (https=) |
| JP (1) | JP6105631B2 (https=) |
| KR (1) | KR20140128318A (https=) |
| CN (1) | CN104080775A (https=) |
| AU (1) | AU2013218119A1 (https=) |
| BR (1) | BR112014019196A8 (https=) |
| CA (1) | CA2862520A1 (https=) |
| CL (1) | CL2014001823A1 (https=) |
| EA (1) | EA201400882A1 (https=) |
| IL (1) | IL233370A (https=) |
| MX (1) | MX2014009033A (https=) |
| PH (1) | PH12014501760B1 (https=) |
| WO (1) | WO2013117568A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2289881A1 (de) * | 2009-08-06 | 2011-03-02 | Boehringer Ingelheim International GmbH | Verfahren zur stereoselektiven Synthese bicyclischer Heterocyclen |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4575507A (en) * | 1985-05-29 | 1986-03-11 | Pfizer Inc. | Spiro-imidazolidines as aldose reductase inhibitors and their pharmaceutical use |
| JP4776882B2 (ja) | 2002-03-30 | 2011-09-21 | ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | 二環式複素環化合物、これらの化合物を含む医薬組成物、それらの使用及びそれらの調製方法 |
| US6924285B2 (en) | 2002-03-30 | 2005-08-02 | Boehringer Ingelheim Pharma Gmbh & Co. | Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them |
| JP2009518450A (ja) | 2005-12-12 | 2009-05-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 二環式複素環化合物、その化合物を含む薬剤、その使用及び製造方法 |
| US8497369B2 (en) * | 2008-02-07 | 2013-07-30 | Boehringer Ingelheim International Gmbh | Spirocyclic heterocycles medicaments containing said compounds, use thereof and method for their production |
| EP2289881A1 (de) * | 2009-08-06 | 2011-03-02 | Boehringer Ingelheim International GmbH | Verfahren zur stereoselektiven Synthese bicyclischer Heterocyclen |
| AP3531A (en) | 2011-02-01 | 2016-01-13 | Boehringer Ingelheim Int | 9-[4-(3-chlor-2-fluor-phenylamino)-7-methoxy-quinazolin-6-yloxy]-1,4-diaza-spiro[5.5]undecan-5-one dimaleate, use thereof as a drug, and production thereof |
-
2013
- 2013-02-06 KR KR1020147021922A patent/KR20140128318A/ko not_active Withdrawn
- 2013-02-06 MX MX2014009033A patent/MX2014009033A/es not_active Application Discontinuation
- 2013-02-06 BR BR112014019196A patent/BR112014019196A8/pt not_active IP Right Cessation
- 2013-02-06 AU AU2013218119A patent/AU2013218119A1/en not_active Abandoned
- 2013-02-06 JP JP2014556029A patent/JP6105631B2/ja active Active
- 2013-02-06 EA EA201400882A patent/EA201400882A1/ru unknown
- 2013-02-06 WO PCT/EP2013/052287 patent/WO2013117568A1/de not_active Ceased
- 2013-02-06 CA CA2862520A patent/CA2862520A1/en not_active Abandoned
- 2013-02-06 EP EP13703045.8A patent/EP2812317B1/de active Active
- 2013-02-06 CN CN201380006918.0A patent/CN104080775A/zh active Pending
- 2013-02-07 US US13/761,211 patent/US8629146B2/en active Active
-
2014
- 2014-06-25 IL IL233370A patent/IL233370A/en not_active IP Right Cessation
- 2014-07-09 CL CL2014001823A patent/CL2014001823A1/es unknown
- 2014-08-05 PH PH12014501760A patent/PH12014501760B1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2015506966A (ja) | 2015-03-05 |
| KR20140128318A (ko) | 2014-11-05 |
| IL233370A0 (en) | 2014-08-31 |
| US20130211081A1 (en) | 2013-08-15 |
| PH12014501760A1 (en) | 2014-11-10 |
| PH12014501760B1 (en) | 2014-11-10 |
| US8629146B2 (en) | 2014-01-14 |
| WO2013117568A1 (de) | 2013-08-15 |
| AU2013218119A1 (en) | 2014-07-17 |
| CA2862520A1 (en) | 2013-08-15 |
| EA201400882A1 (ru) | 2015-01-30 |
| EP2812317A1 (de) | 2014-12-17 |
| BR112014019196A8 (pt) | 2017-07-11 |
| BR112014019196A2 (https=) | 2017-06-20 |
| IL233370A (en) | 2015-04-30 |
| EP2812317B1 (de) | 2016-02-03 |
| JP6105631B2 (ja) | 2017-03-29 |
| CL2014001823A1 (es) | 2015-03-06 |
| CN104080775A (zh) | 2014-10-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |