MX2013006836A - Inhibidores de la replicacion de los virus de la influenza. - Google Patents
Inhibidores de la replicacion de los virus de la influenza.Info
- Publication number
- MX2013006836A MX2013006836A MX2013006836A MX2013006836A MX2013006836A MX 2013006836 A MX2013006836 A MX 2013006836A MX 2013006836 A MX2013006836 A MX 2013006836A MX 2013006836 A MX2013006836 A MX 2013006836A MX 2013006836 A MX2013006836 A MX 2013006836A
- Authority
- MX
- Mexico
- Prior art keywords
- alkyl
- independently
- group
- optionally
- halogen
- Prior art date
Links
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
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- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| US201161527273P | 2011-08-25 | 2011-08-25 | |
| PCT/US2011/065371 WO2012083117A1 (en) | 2010-12-16 | 2011-12-16 | Inhibitors of influenza viruses replication |
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| RU (1) | RU2013132681A (enExample) |
| WO (1) | WO2012083117A1 (enExample) |
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-
2011
- 2011-12-16 RU RU2013132681/04A patent/RU2013132681A/ru not_active Application Discontinuation
- 2011-12-16 MX MX2013006836A patent/MX2013006836A/es not_active Application Discontinuation
- 2011-12-16 EP EP11808474.8A patent/EP2651940A1/en not_active Withdrawn
- 2011-12-16 JP JP2013544808A patent/JP2013545816A/ja active Pending
- 2011-12-16 CA CA2822057A patent/CA2822057A1/en not_active Abandoned
- 2011-12-16 AU AU2011343642A patent/AU2011343642A1/en not_active Abandoned
- 2011-12-16 KR KR1020137018521A patent/KR20140014110A/ko not_active Withdrawn
- 2011-12-16 CN CN201180066550.8A patent/CN103492381A/zh active Pending
- 2011-12-16 WO PCT/US2011/065371 patent/WO2012083117A1/en not_active Ceased
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2013
- 2013-06-14 US US13/918,048 patent/US8871774B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AU2011343642A1 (en) | 2013-05-02 |
| RU2013132681A (ru) | 2015-01-27 |
| CA2822057A1 (en) | 2012-06-21 |
| CN103492381A (zh) | 2014-01-01 |
| KR20140014110A (ko) | 2014-02-05 |
| JP2013545816A (ja) | 2013-12-26 |
| EP2651940A1 (en) | 2013-10-23 |
| WO2012083117A1 (en) | 2012-06-21 |
| US8871774B2 (en) | 2014-10-28 |
| US20140005192A1 (en) | 2014-01-02 |
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