MX2012004074A - Pirimidonas fusionadas de tiazolo y oxazolo. - Google Patents
Pirimidonas fusionadas de tiazolo y oxazolo.Info
- Publication number
- MX2012004074A MX2012004074A MX2012004074A MX2012004074A MX2012004074A MX 2012004074 A MX2012004074 A MX 2012004074A MX 2012004074 A MX2012004074 A MX 2012004074A MX 2012004074 A MX2012004074 A MX 2012004074A MX 2012004074 A MX2012004074 A MX 2012004074A
- Authority
- MX
- Mexico
- Prior art keywords
- pyrimidinones
- oxazolo
- compounds
- pharmaceutically acceptable
- present
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/16—Peri-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Epidemiology (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se relaciona con compuestos novedosos, sus sales farmacéuticamente aceptables, y sus isómeros, esteroisómeros, conformadores, tautómeros, polimorfos, hidratos y solvatos. La presente invención también abarca composiciones farmacéuticamente aceptables de dichos compuestos y procesos para la preparación de compuestos novedosos. La invención, además, se relaciona con el uso de los compuestos antes mencionados para la preparación de medicamentos para su uso como farmacéuticos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN1249KO2009 | 2009-10-13 | ||
PCT/IN2010/000579 WO2011045811A1 (en) | 2009-10-13 | 2010-08-31 | Fused thiazolo and oxazolo pyrimidinones |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2012004074A true MX2012004074A (es) | 2012-05-22 |
Family
ID=43034589
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2012004074A MX2012004074A (es) | 2009-10-13 | 2010-08-31 | Pirimidonas fusionadas de tiazolo y oxazolo. |
Country Status (27)
Country | Link |
---|---|
EP (1) | EP2385948B1 (es) |
JP (1) | JP5681195B2 (es) |
KR (1) | KR101710430B1 (es) |
CN (1) | CN102549000B (es) |
AR (1) | AR080616A1 (es) |
AU (1) | AU2010307984B2 (es) |
BR (1) | BR112012006233B8 (es) |
CA (1) | CA2772995C (es) |
CY (1) | CY1119710T1 (es) |
DK (1) | DK2385948T3 (es) |
EA (1) | EA020228B1 (es) |
ES (1) | ES2653931T3 (es) |
HR (1) | HRP20171976T1 (es) |
HU (1) | HUE038051T2 (es) |
IL (1) | IL219116A (es) |
LT (1) | LT2385948T (es) |
MX (1) | MX2012004074A (es) |
MY (1) | MY157629A (es) |
NO (1) | NO2385948T3 (es) |
NZ (1) | NZ598020A (es) |
PL (1) | PL2385948T3 (es) |
RS (1) | RS56630B1 (es) |
SI (1) | SI2385948T1 (es) |
TW (1) | TWI500623B (es) |
UA (1) | UA107473C2 (es) |
WO (1) | WO2011045811A1 (es) |
ZA (1) | ZA201203262B (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI661828B (zh) | 2013-05-14 | 2019-06-11 | 印度商托仁特生技有限公司 | 低劑量藥物組合物及其用途 |
AU2015311333B2 (en) | 2014-09-02 | 2017-11-16 | Sunshine Lake Pharma Co., Ltd. | Quinolinone compound and use thereof |
CN106905348B (zh) * | 2017-02-13 | 2018-12-04 | 牡丹江医学院 | 一种预防和治疗急性肾损伤的药物及其制备方法和用途 |
CN110511233B (zh) * | 2019-08-08 | 2022-01-25 | 成都大学 | 一种噻唑并[2,3-b]噁唑酮类化合物及其制备方法和用途 |
CN112778333B (zh) * | 2021-01-23 | 2022-07-05 | 中国科学院新疆理化技术研究所 | 一种四氢噁唑并吡啶并氮氧杂酮类衍生物及其用途 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4072679A (en) * | 1976-06-15 | 1978-02-07 | E. R. Squibb & Sons, Inc. | 1,4- AND 4,10-DIHYDRO-4-OXO-PYRIMIDO (1,2-A)-benzimidazole-3-carboxylic acids, esters and amides |
DK151811C (da) * | 1979-11-23 | 1988-06-06 | Pfizer | Analogifremgangsmaade til fremstilling af n-(5-tetrazolyl)-1-oxo-1h-thiazolooe3,2-aaa-pyrimidin-2-carboxamider eller farmaceutisk acceptable kationsalte deraf samt 1-oxo-1h-thiazolooe3,2-aaapyrimidin-2-carboxylsyrer til anvendelse som udgangsmaterialer ved fremgangsmaaden |
US4423048A (en) | 1979-11-23 | 1983-12-27 | Pfizer Inc. | Antiallergic and antiulcer 1-oxo-1H-thiazolo[3,2-a]pyrimidine-2-carboxamides and intermediates therefor |
JPH0539293A (ja) | 1991-01-23 | 1993-02-19 | Kyowa Hakko Kogyo Co Ltd | 免疫調節剤及びチアゾロピリミジン誘導体 |
TW406076B (en) | 1993-12-30 | 2000-09-21 | Hoechst Ag | Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals |
CN100522946C (zh) | 2001-12-06 | 2009-08-05 | 法布罗根股份有限公司 | 低氧诱导因子(HIF)α的稳定化 |
KR20050110612A (ko) | 2002-12-25 | 2005-11-23 | 다이이찌 세이야꾸 가부시기가이샤 | 디아민 유도체 |
US8614204B2 (en) | 2003-06-06 | 2013-12-24 | Fibrogen, Inc. | Enhanced erythropoiesis and iron metabolism |
WO2007115315A2 (en) * | 2006-04-04 | 2007-10-11 | Fibrogen, Inc. | Pyrrolo- and thiazolo-pyridine compounds as hif modulators |
US7713986B2 (en) | 2006-06-15 | 2010-05-11 | Fibrogen, Inc. | Compounds and methods for treatment of chemotherapy-induced anemia |
US20070293575A1 (en) | 2006-06-15 | 2007-12-20 | Fibrogen, Inc. | Compounds and methods for treatment of cancer-related anemia |
TWI394747B (zh) * | 2006-06-23 | 2013-05-01 | Smithkline Beecham Corp | 脯胺醯基羥化酶抑制劑 |
WO2009039321A1 (en) * | 2007-09-19 | 2009-03-26 | Smithkline Beecham Corporation | Prolyl hydroxylase inhibitors |
WO2009039322A1 (en) * | 2007-09-19 | 2009-03-26 | Smithkline Beecham Corporation | Prolyl hydroxylase inhibitors |
-
2010
- 2010-08-30 TW TW099129121A patent/TWI500623B/zh active
- 2010-08-31 JP JP2012533740A patent/JP5681195B2/ja active Active
- 2010-08-31 WO PCT/IN2010/000579 patent/WO2011045811A1/en active Application Filing
- 2010-08-31 DK DK10760108.0T patent/DK2385948T3/en active
- 2010-08-31 MX MX2012004074A patent/MX2012004074A/es active IP Right Grant
- 2010-08-31 EA EA201270556A patent/EA020228B1/ru not_active IP Right Cessation
- 2010-08-31 UA UAA201205825A patent/UA107473C2/uk unknown
- 2010-08-31 AU AU2010307984A patent/AU2010307984B2/en not_active Ceased
- 2010-08-31 BR BR112012006233A patent/BR112012006233B8/pt active IP Right Grant
- 2010-08-31 PL PL10760108T patent/PL2385948T3/pl unknown
- 2010-08-31 ES ES10760108.0T patent/ES2653931T3/es active Active
- 2010-08-31 EP EP10760108.0A patent/EP2385948B1/en active Active
- 2010-08-31 CN CN201080038159.2A patent/CN102549000B/zh active Active
- 2010-08-31 HU HUE10760108A patent/HUE038051T2/hu unknown
- 2010-08-31 MY MYPI2012001679A patent/MY157629A/en unknown
- 2010-08-31 NZ NZ598020A patent/NZ598020A/xx not_active IP Right Cessation
- 2010-08-31 LT LTEP10760108.0T patent/LT2385948T/lt unknown
- 2010-08-31 NO NO10760108A patent/NO2385948T3/no unknown
- 2010-08-31 RS RS20171226A patent/RS56630B1/sr unknown
- 2010-08-31 CA CA2772995A patent/CA2772995C/en active Active
- 2010-08-31 KR KR1020127011052A patent/KR101710430B1/ko active IP Right Grant
- 2010-08-31 SI SI201031610T patent/SI2385948T1/en unknown
- 2010-10-12 AR ARP100103718A patent/AR080616A1/es active IP Right Grant
-
2012
- 2012-04-05 IL IL219116A patent/IL219116A/en active IP Right Grant
- 2012-05-04 ZA ZA2012/03262A patent/ZA201203262B/en unknown
-
2017
- 2017-12-20 HR HRP20171976TT patent/HRP20171976T1/hr unknown
- 2017-12-28 CY CY20171101352T patent/CY1119710T1/el unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant or registration |