MX2009013833A - Compuestos de piridazina cristalina. - Google Patents

Compuestos de piridazina cristalina.

Info

Publication number
MX2009013833A
MX2009013833A MX2009013833A MX2009013833A MX2009013833A MX 2009013833 A MX2009013833 A MX 2009013833A MX 2009013833 A MX2009013833 A MX 2009013833A MX 2009013833 A MX2009013833 A MX 2009013833A MX 2009013833 A MX2009013833 A MX 2009013833A
Authority
MX
Mexico
Prior art keywords
crystalline
pyridazine compound
crystalline compound
compound
pyridazine
Prior art date
Application number
MX2009013833A
Other languages
English (en)
Inventor
Eric D Dowdy
Vahid Zia
Kenneth M Kent
Norma J Tom
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39790369&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2009013833(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of MX2009013833A publication Critical patent/MX2009013833A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se proporciona un compuesto de la fórmula (1) cristalina y sus sales y solvatos para el tratamiento o profilaxis de las infecciones del virus de hepatitis C (1). Se proporcionan métodos de elaboración y compuestos de formulación cristalina (1).
MX2009013833A 2007-07-06 2008-07-03 Compuestos de piridazina cristalina. MX2009013833A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US95859507P 2007-07-06 2007-07-06
PCT/US2008/008259 WO2009009001A1 (en) 2007-07-06 2008-07-03 Crystalline pyridazine compound

Publications (1)

Publication Number Publication Date
MX2009013833A true MX2009013833A (es) 2010-03-10

Family

ID=39790369

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009013833A MX2009013833A (es) 2007-07-06 2008-07-03 Compuestos de piridazina cristalina.

Country Status (19)

Country Link
US (2) US8106054B2 (es)
EP (1) EP2170881A1 (es)
JP (2) JP5366944B2 (es)
KR (1) KR101229528B1 (es)
CN (1) CN101778847B (es)
AP (1) AP2593A (es)
AR (1) AR066158A1 (es)
AU (1) AU2008275756B2 (es)
BR (1) BRPI0814801A2 (es)
CA (1) CA2691917C (es)
CO (1) CO6251293A2 (es)
EA (2) EA018173B1 (es)
EC (1) ECSP109919A (es)
IL (1) IL202694A0 (es)
MX (1) MX2009013833A (es)
TW (1) TWI447116B (es)
UA (1) UA99466C2 (es)
WO (1) WO2009009001A1 (es)
ZA (1) ZA201000826B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0215293D0 (en) 2002-07-03 2002-08-14 Rega Foundation Viral inhibitors
EP2161273B1 (en) * 2003-12-22 2015-04-15 K.U.Leuven Research & Development Imidazo[4,5-c]pyridine compounds and methods of antiviral treatment
DK1841765T5 (da) * 2004-12-21 2009-12-21 Gilead Sciences Inc Imidazo[4,5-C]pyridinforbindelse og fremgangsmåde til antiviral behandling
JP4958974B2 (ja) * 2006-07-07 2012-06-20 ギリアード サイエンシーズ, インコーポレイテッド 新規ピリダジン化合物およびそれらの使用
EP2094702B1 (en) 2006-12-14 2015-09-02 Gilead Sciences, Inc. Viral inhibitors
UA99466C2 (en) 2007-07-06 2012-08-27 Гилиад Сайенсиз, Инк. Crystalline pyridazine compound
US20130029904A1 (en) 2009-12-18 2013-01-31 Boehringer Ingelheim International Gmbh Hcv combination therapy
WO2011146817A1 (en) 2010-05-21 2011-11-24 Gilead Sciences, Inc. Heterocyclic flaviviridae virus inhibitors
CA2822037A1 (en) 2010-12-20 2012-06-28 Gilead Sciences, Inc. Methods for treating hcv
US20120204871A1 (en) * 2011-02-10 2012-08-16 Julio Cesar Vega Stable, non-corrosive formulations for pressurized metered dose inhalers
DE202012013074U1 (de) 2011-09-16 2014-10-29 Gilead Pharmasset Lcc Zusammensetzungen zur Behandlung von HCV
CN104144682A (zh) 2013-01-31 2014-11-12 吉利德法莫赛特有限责任公司 两个抗病毒化合物的联用制剂
BR112017013858A2 (pt) 2014-12-26 2018-02-27 Univ Emory n4-hidroxicitidina e derivados e usos antivirais relacionados aos mesmos
MX2020005392A (es) 2017-12-07 2020-12-07 Univ Emory N4-hidroxicitidina y derivados y usos antivirales relacionados con los mismos.
CN114195812A (zh) * 2021-12-30 2022-03-18 大连联化化学有限公司 一种合成2,4-二三氟甲基苯硼酸的方法

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Also Published As

Publication number Publication date
CA2691917A1 (en) 2009-01-15
EA018173B1 (ru) 2013-06-28
AR066158A1 (es) 2009-07-29
US20120108601A1 (en) 2012-05-03
ECSP109919A (es) 2010-04-30
UA99466C2 (en) 2012-08-27
JP2013216695A (ja) 2013-10-24
US8569488B2 (en) 2013-10-29
KR101229528B1 (ko) 2013-02-04
IL202694A0 (en) 2010-06-30
JP5366944B2 (ja) 2013-12-11
ZA201000826B (en) 2010-11-24
EA200971080A1 (ru) 2010-08-30
AU2008275756B2 (en) 2012-01-19
TW200918531A (en) 2009-05-01
CN101778847B (zh) 2013-07-24
EA201270275A1 (ru) 2012-09-28
BRPI0814801A2 (pt) 2017-03-28
US8106054B2 (en) 2012-01-31
JP2010532757A (ja) 2010-10-14
TWI447116B (zh) 2014-08-01
CA2691917C (en) 2013-12-03
EP2170881A1 (en) 2010-04-07
WO2009009001A9 (en) 2010-11-11
AP2009005078A0 (en) 2009-12-31
CN101778847A (zh) 2010-07-14
US20090036460A1 (en) 2009-02-05
AU2008275756A1 (en) 2009-01-15
CO6251293A2 (es) 2011-02-21
WO2009009001A1 (en) 2009-01-15
AP2593A (en) 2013-02-07
KR20100044201A (ko) 2010-04-29

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