MX2008012168A - Analogos de 2-aminopiridina como activadores de glucocinasa. - Google Patents

Analogos de 2-aminopiridina como activadores de glucocinasa.

Info

Publication number
MX2008012168A
MX2008012168A MX2008012168A MX2008012168A MX2008012168A MX 2008012168 A MX2008012168 A MX 2008012168A MX 2008012168 A MX2008012168 A MX 2008012168A MX 2008012168 A MX2008012168 A MX 2008012168A MX 2008012168 A MX2008012168 A MX 2008012168A
Authority
MX
Mexico
Prior art keywords
alkyl
heteroaryl
saturated
aryl
optionally substituted
Prior art date
Application number
MX2008012168A
Other languages
English (en)
Spanish (es)
Inventor
Kevin Ronald Condroski
Thomas Daniel Aicher
Ronald Jay Hinklin
Mark Joseph Chicarelli
Steven Armen Boyd
Ajay Singh
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of MX2008012168A publication Critical patent/MX2008012168A/es

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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Reproductive Health (AREA)
  • Communicable Diseases (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
MX2008012168A 2006-03-24 2007-03-23 Analogos de 2-aminopiridina como activadores de glucocinasa. MX2008012168A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78546006P 2006-03-24 2006-03-24
PCT/US2007/007444 WO2007117381A2 (en) 2006-03-24 2007-03-23 2 -aminopyridine analogs as glucokinase activators

Publications (1)

Publication Number Publication Date
MX2008012168A true MX2008012168A (es) 2008-10-03

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Application Number Title Priority Date Filing Date
MX2008012168A MX2008012168A (es) 2006-03-24 2007-03-23 Analogos de 2-aminopiridina como activadores de glucocinasa.

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US (3) US8022223B2 (enExample)
EP (2) EP2543667B1 (enExample)
JP (2) JP5377284B2 (enExample)
KR (1) KR101440634B1 (enExample)
CN (1) CN101437816B (enExample)
AU (1) AU2007235558B2 (enExample)
BR (1) BRPI0709171A2 (enExample)
CA (1) CA2647208C (enExample)
DK (1) DK2013204T3 (enExample)
ES (1) ES2536547T3 (enExample)
HR (1) HRP20150347T1 (enExample)
IL (1) IL194160A (enExample)
MX (1) MX2008012168A (enExample)
MY (1) MY148985A (enExample)
NZ (1) NZ571997A (enExample)
PL (1) PL2013204T3 (enExample)
PT (1) PT2013204E (enExample)
RS (1) RS53981B1 (enExample)
RU (1) RU2457207C2 (enExample)
SG (1) SG170775A1 (enExample)
SI (1) SI2013204T1 (enExample)
TW (1) TWI393718B (enExample)
UA (1) UA103746C2 (enExample)
WO (1) WO2007117381A2 (enExample)
ZA (1) ZA200809017B (enExample)

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NZ571997A (en) 2006-03-24 2011-08-26 Array Biopharma Inc 2 -aminopyridine analogs as glucokinase activators
WO2008091770A1 (en) * 2007-01-24 2008-07-31 Array Biopharma Inc. 2-aminopyridine derivatives as glucokinase activators
EP2173745A2 (en) * 2007-03-23 2010-04-14 Array Biopharma, Inc. 2-aminopyridine analogs as glucokinase activators
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
CN101868459B (zh) * 2007-09-21 2013-12-18 阿雷生物药品公司 用于治疗糖尿病的、作为葡糖激酶激活剂的吡啶-2-基-氨基-1,2,4-噻二唑衍生物
JP5567481B2 (ja) * 2007-10-09 2014-08-06 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング グルコキナーゼアクチベーターとして有用なピリジン誘導体
AU2009211718B2 (en) 2008-02-06 2011-08-11 Daiichi Sankyo Company, Limited Novel phenylpyrrole derivative
US7741327B2 (en) 2008-04-16 2010-06-22 Hoffmann-La Roche Inc. Pyrrolidinone glucokinase activators
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
ES2624780T3 (es) 2010-03-31 2017-07-17 The Scripps Research Institute Reprogramación de células
US8178689B2 (en) 2010-06-17 2012-05-15 Hoffman-La Roche Inc. Tricyclic compounds
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