UA103746C2 - 2-aminopyridine analogs as glucokinase activators - Google Patents

2-aminopyridine analogs as glucokinase activators

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Publication number
UA103746C2
UA103746C2 UAA200812528A UAA200812528A UA103746C2 UA 103746 C2 UA103746 C2 UA 103746C2 UA A200812528 A UAA200812528 A UA A200812528A UA A200812528 A UAA200812528 A UA A200812528A UA 103746 C2 UA103746 C2 UA 103746C2
Authority
UA
Ukraine
Prior art keywords
glucokinase
glucokinase activators
aminopyridine
analogs
aminopyridine analogs
Prior art date
Application number
UAA200812528A
Other languages
English (en)
Ukrainian (uk)
Inventor
Томас Дениэл Эйчер
Стивен Армен Бойд
Марк Джозеф Чикарелли
Кевин Рональд Кондроски
Рональд Джей Гинклин
Аджей Сингх
Original Assignee
Эррей Биофарма Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эррей Биофарма Инк. filed Critical Эррей Биофарма Инк.
Publication of UA103746C2 publication Critical patent/UA103746C2/ru

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Abstract

Предложены соединения, эффективные при лечении и/или профилактики заболеваний, опосредствованных недостаточными уровнями глюкокиназной активности, таких как сахарный диабет. Также предложены способы лечения или профилактики заболеваний и расстройств, которые характеризуются недостаточной глюкокиназной активностью или которые можно лечить путем активации глюкокиназы.
UAA200812528A 2006-03-24 2007-03-23 2-aminopyridine analogs as glucokinase activators UA103746C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78546006P 2006-03-24 2006-03-24
PCT/US2007/007444 WO2007117381A2 (en) 2006-03-24 2007-03-23 2 -aminopyridine analogs as glucokinase activators

Publications (1)

Publication Number Publication Date
UA103746C2 true UA103746C2 (en) 2013-11-25

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US (3) US8022223B2 (ru)
EP (2) EP2013204B1 (ru)
JP (2) JP5377284B2 (ru)
KR (1) KR101440634B1 (ru)
CN (1) CN101437816B (ru)
AU (1) AU2007235558B2 (ru)
BR (1) BRPI0709171A2 (ru)
CA (1) CA2647208C (ru)
DK (1) DK2013204T3 (ru)
ES (1) ES2536547T3 (ru)
HK (1) HK1128130A1 (ru)
HR (1) HRP20150347T1 (ru)
IL (1) IL194160A (ru)
MX (1) MX2008012168A (ru)
MY (1) MY148985A (ru)
NZ (1) NZ571997A (ru)
PL (1) PL2013204T3 (ru)
PT (1) PT2013204E (ru)
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RU (1) RU2457207C2 (ru)
SG (1) SG170775A1 (ru)
SI (1) SI2013204T1 (ru)
TW (1) TWI393718B (ru)
UA (1) UA103746C2 (ru)
WO (1) WO2007117381A2 (ru)
ZA (1) ZA200809017B (ru)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
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JP5377284B2 (ja) 2006-03-24 2013-12-25 アレイ バイオファーマ、インコーポレイテッド グルコキナーゼアクチベーターとしての２−アミノピリジンアナログ
WO2008091770A1 (en) * 2007-01-24 2008-07-31 Array Biopharma Inc. 2-aminopyridine derivatives as glucokinase activators
EP2173745A2 (en) * 2007-03-23 2010-04-14 Array Biopharma, Inc. 2-aminopyridine analogs as glucokinase activators
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
SI2209778T1 (sl) * 2007-09-21 2012-12-31 Array Biopharma, Inc. Piridin-2-il-amino-I, 2,4-tiadiazol derivati kot aktivatorji glukokinaze za zdravljenje sladkorne bolezni
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