MX2007013766A - Combinacion de inhibidor pde4 de roflumilast y un derivado de tetrahidrobiopterina. - Google Patents
Combinacion de inhibidor pde4 de roflumilast y un derivado de tetrahidrobiopterina.Info
- Publication number
- MX2007013766A MX2007013766A MX2007013766A MX2007013766A MX2007013766A MX 2007013766 A MX2007013766 A MX 2007013766A MX 2007013766 A MX2007013766 A MX 2007013766A MX 2007013766 A MX2007013766 A MX 2007013766A MX 2007013766 A MX2007013766 A MX 2007013766A
- Authority
- MX
- Mexico
- Prior art keywords
- pharmaceutically acceptable
- roflumilast
- acceptable salt
- combination product
- treatment
- Prior art date
Links
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP05103938 | 2005-05-11 | ||
| PCT/EP2006/062117 WO2006120176A2 (en) | 2005-05-11 | 2006-05-08 | Combination of the pde4 inhibitor roflumilast and a tetrahydrobiopterin derivative |
Publications (1)
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| MX2007013766A true MX2007013766A (es) | 2008-01-28 |
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| MX2007013766A MX2007013766A (es) | 2005-05-11 | 2006-05-08 | Combinacion de inhibidor pde4 de roflumilast y un derivado de tetrahidrobiopterina. |
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| MX (1) | MX2007013766A (enExample) |
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| AU2006321942A1 (en) * | 2005-12-05 | 2007-06-14 | Biomarin Pharmaceutical Inc. | Methods and compositions for the treatment of disease |
| WO2008089148A1 (en) * | 2007-01-12 | 2008-07-24 | Biomarin Pharmaceutical Inc. | Method of treating a metabolic or neuropsychiatry disorder with a bh4 derivative prodrug |
| MY153979A (en) | 2007-10-19 | 2015-04-30 | Boehringer Ingelheim Int | Substituted piperidino-dihydrothienopyrimidine |
| JP2011530540A (ja) * | 2008-08-12 | 2011-12-22 | オルファ スイス ゲーエムベーハー | テトラヒドロビオプテリンを含有する医薬剤形 |
| CN102256963B (zh) | 2008-12-19 | 2014-06-11 | 贝林格尔.英格海姆国际有限公司 | 作为ccr2受体拮抗剂用于治疗炎症、哮喘和copd的环状嘧啶-4-甲酰胺 |
| WO2010097374A1 (de) | 2009-02-26 | 2010-09-02 | Boehringer Ingelheim International Gmbh | Verbindungen als bradykinin-b1-antagonisten |
| WO2010097373A1 (de) | 2009-02-26 | 2010-09-02 | Boehringer Ingelheim International Gmbh | Verbindungen als bradykinin b1 antagonisten |
| CA2759126C (en) | 2009-02-26 | 2017-08-22 | Boehringer Ingelheim International Gmbh | Compounds as bradykinin b1 antagonists |
| CA2790952C (en) | 2010-02-23 | 2017-07-04 | Boehringer Ingelheim International Gmbh | Compounds as bradykinin b1 antagonists |
| WO2011132435A1 (ja) | 2010-04-22 | 2011-10-27 | 学校法人日本大学 | 脳機能障害予防・改善用の薬剤及び飲食物 |
| CN102274222B (zh) * | 2011-08-18 | 2013-04-10 | 天津市汉康医药生物技术有限公司 | 高生物利用度的罗氟司特药物组合物及其制备方法 |
| US20130059866A1 (en) | 2011-08-24 | 2013-03-07 | Boehringer Ingelheim International Gmbh | Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma |
| WO2014037832A2 (en) | 2012-09-06 | 2014-03-13 | Mahesh Kandula | Compositions and methods for the treatment of epilepsy and neurological diseases |
| EP2847158A4 (en) | 2012-05-07 | 2015-12-30 | Cellix Bio Private Ltd | COMPOSITIONS AND METHODS FOR THE TREATMENT OF NEUROMUSCULAR DISORDERS AND NEURODEGENERATIVE DISORDERS |
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| US9309233B2 (en) | 2012-05-08 | 2016-04-12 | Cellix Bio Private Limited | Compositions and methods for the treatment of blood clotting disorders |
| US9522884B2 (en) | 2012-05-08 | 2016-12-20 | Cellix Bio Private Limited | Compositions and methods for the treatment of metabolic disorders |
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| US9315461B2 (en) | 2012-05-10 | 2016-04-19 | Cellix Bio Private Limited | Compositions and methods for the treatment of neurologic diseases |
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| US9242939B2 (en) | 2012-05-10 | 2016-01-26 | Cellix Bio Private Limited | Compositions and methods for the treatment of respiratory disorders |
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| SG11201407319YA (en) | 2012-05-23 | 2014-12-30 | Cellix Bio Private Ltd | Compositions and methods for treatment of inflammatory bowel disease |
| CA2873098A1 (en) | 2012-05-23 | 2013-11-28 | Cellixbio Private Limited | Compositions and methods for the treatment of multiple sclerosis |
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| CN106139161A (zh) * | 2016-08-12 | 2016-11-23 | 合肥久诺医药科技有限公司 | 一种罗氟司特包合物及其固体制剂 |
| WO2019147824A1 (en) | 2018-01-26 | 2019-08-01 | Progenity, Inc. | Treatment of a disease of the gastrointestinal tract with a pde4 inhibitor |
| CN116726361A (zh) | 2018-11-19 | 2023-09-12 | 比奥拉治疗股份有限公司 | 用生物治疗剂治疗疾病的方法和装置 |
| US11707610B2 (en) | 2019-12-13 | 2023-07-25 | Biora Therapeutics, Inc. | Ingestible device for delivery of therapeutic agent to the gastrointestinal tract |
| WO2021213455A1 (zh) * | 2020-04-23 | 2021-10-28 | 浙江养生堂天然药物研究所有限公司 | 药物组合及其用途 |
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| US5877176A (en) * | 1991-12-26 | 1999-03-02 | Cornell Research Foundation, Inc. | Blocking induction of tetrahydrobiopterin to block induction of nitric oxide synthesis |
| US5830461A (en) * | 1992-11-25 | 1998-11-03 | University Of Pittsburgh Of The Commonwealth System Of Higher Education | Methods for promoting wound healing and treating transplant-associated vasculopathy |
| SI0706513T1 (en) * | 1993-07-02 | 2002-10-31 | Altana Pharma Ag | Fluoroalkoxy-substituted benzamides and their use as cyclic nucleotide phosphodiesterase inhibitors |
| DE4418097A1 (de) * | 1994-05-24 | 1995-11-30 | Cassella Ag | Verwendung von Tetrahydropteridin-Derivaten als Hemmstoffe der NO-Synthase |
| ATE252385T1 (de) * | 1996-08-30 | 2003-11-15 | Daiichi Suntory Pharma Co Ltd | Vorbeugende oder heilende mittel für krankheiten, die durch mangel an stickoxid-synthase (nos) ausgelöst sind |
| SE0000307D0 (sv) * | 2000-01-31 | 2000-01-31 | Univ Zuerich | Method and formulation för treatment of vasoconstriction |
| US6544994B2 (en) * | 2000-06-07 | 2003-04-08 | Eprov Ag | Pharmaceutical preparation for treating or preventing cardiovascular or neurological disorders by modulating of the activity of nitric oxide synthase |
| MXPA06004687A (es) * | 2003-10-31 | 2006-06-27 | Altana Pharma Ag | Uso de bh4 para el tratamiento de enfermedades respiratorias. |
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- 2006-05-08 KR KR1020077028279A patent/KR20080005601A/ko not_active Withdrawn
- 2006-05-08 CA CA002607331A patent/CA2607331A1/en not_active Abandoned
- 2006-05-08 CN CNA2006800148286A patent/CN101171005A/zh active Pending
- 2006-05-08 AU AU2006245770A patent/AU2006245770A1/en not_active Abandoned
- 2006-05-08 JP JP2008510556A patent/JP2008540486A/ja not_active Withdrawn
- 2006-05-08 US US11/919,742 patent/US20080221111A1/en not_active Abandoned
- 2006-05-08 EA EA200702358A patent/EA200702358A1/ru unknown
- 2006-05-08 MX MX2007013766A patent/MX2007013766A/es not_active Application Discontinuation
- 2006-05-08 BR BRPI0612796-7A patent/BRPI0612796A2/pt not_active IP Right Cessation
- 2006-05-08 EP EP06755065A patent/EP1940392A2/en not_active Withdrawn
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| WO2006120176A2 (en) | 2006-11-16 |
| CN101171005A (zh) | 2008-04-30 |
| US20080221111A1 (en) | 2008-09-11 |
| NO20076206L (no) | 2007-12-11 |
| CA2607331A1 (en) | 2006-11-16 |
| WO2006120176A3 (en) | 2007-04-19 |
| JP2008540486A (ja) | 2008-11-20 |
| EP1940392A2 (en) | 2008-07-09 |
| ZA200708776B (en) | 2008-10-29 |
| BRPI0612796A2 (pt) | 2010-11-30 |
| IL186804A0 (en) | 2008-06-05 |
| KR20080005601A (ko) | 2008-01-14 |
| AU2006245770A1 (en) | 2006-11-16 |
| EA200702358A1 (ru) | 2008-04-28 |
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