MX2007004936A - Compuestos y composiciones como inhibidores de la actividad del receptor canabinoide 1. - Google Patents
Compuestos y composiciones como inhibidores de la actividad del receptor canabinoide 1.Info
- Publication number
- MX2007004936A MX2007004936A MX2007004936A MX2007004936A MX2007004936A MX 2007004936 A MX2007004936 A MX 2007004936A MX 2007004936 A MX2007004936 A MX 2007004936A MX 2007004936 A MX2007004936 A MX 2007004936A MX 2007004936 A MX2007004936 A MX 2007004936A
- Authority
- MX
- Mexico
- Prior art keywords
- compounds
- activity
- cannabinoid receptor
- compositions
- inhibitors
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 102100033868 Cannabinoid receptor 1 Human genes 0.000 title abstract 3
- 101710187010 Cannabinoid receptor 1 Proteins 0.000 title abstract 3
- 239000003112 inhibitor Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
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- General Health & Medical Sciences (AREA)
- Public Health (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Neurology (AREA)
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- Diabetes (AREA)
- Immunology (AREA)
- Cardiology (AREA)
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- Pulmonology (AREA)
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- Endocrinology (AREA)
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- Obesity (AREA)
- Pain & Pain Management (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US62250804P | 2004-10-26 | 2004-10-26 | |
| US67267005P | 2005-04-18 | 2005-04-18 | |
| PCT/US2005/038361 WO2006047516A2 (en) | 2004-10-26 | 2005-10-26 | Compounds and compositions as inhibitors of cannabinoid receptor 1 activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007004936A true MX2007004936A (es) | 2007-06-25 |
Family
ID=36228382
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007004936A MX2007004936A (es) | 2004-10-26 | 2005-10-26 | Compuestos y composiciones como inhibidores de la actividad del receptor canabinoide 1. |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US8158634B2 (enExample) |
| EP (1) | EP1807429A4 (enExample) |
| JP (2) | JP2008518016A (enExample) |
| KR (1) | KR100919524B1 (enExample) |
| CN (2) | CN102241680A (enExample) |
| AR (1) | AR051596A1 (enExample) |
| AU (2) | AU2005299421B2 (enExample) |
| BR (1) | BRPI0517015A (enExample) |
| CA (2) | CA2581225C (enExample) |
| EC (1) | ECSP077421A (enExample) |
| IL (1) | IL182527A0 (enExample) |
| IN (1) | IN2007DN02514A (enExample) |
| MA (1) | MA28937B1 (enExample) |
| MX (1) | MX2007004936A (enExample) |
| NO (1) | NO20072352L (enExample) |
| PE (1) | PE20060599A1 (enExample) |
| RU (1) | RU2431635C2 (enExample) |
| TN (1) | TNSN07161A1 (enExample) |
| TW (1) | TW200630096A (enExample) |
| WO (1) | WO2006047516A2 (enExample) |
Families Citing this family (76)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT1599468E (pt) | 2003-01-14 | 2008-01-14 | Arena Pharm Inc | Derivados de arilo e heteroarilo 1,2,3.-trissubstituídos comomoduladores do metabolismo, e profilaxia e tratamento dedesordens relacionadas tais como diabetes e hiperglicemia |
| EP2287165A3 (en) | 2003-07-14 | 2011-06-22 | Arena Pharmaceuticals, Inc. | Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto |
| JP2007519754A (ja) * | 2004-01-30 | 2007-07-19 | スミスクライン ビーチャム コーポレーション | 化合物 |
| AR051596A1 (es) * | 2004-10-26 | 2007-01-24 | Irm Llc | Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios |
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- 2005-10-25 PE PE2005001251A patent/PE20060599A1/es not_active Application Discontinuation
- 2005-10-25 TW TW094137369A patent/TW200630096A/zh unknown
- 2005-10-26 JP JP2007539039A patent/JP2008518016A/ja not_active Withdrawn
- 2005-10-26 CN CN2011101210450A patent/CN102241680A/zh active Pending
- 2005-10-26 BR BRPI0517015-0A patent/BRPI0517015A/pt not_active IP Right Cessation
- 2005-10-26 RU RU2007119449/04A patent/RU2431635C2/ru not_active IP Right Cessation
- 2005-10-26 EP EP05813001A patent/EP1807429A4/en not_active Withdrawn
- 2005-10-26 US US11/718,016 patent/US8158634B2/en not_active Expired - Fee Related
- 2005-10-26 AU AU2005299421A patent/AU2005299421B2/en not_active Ceased
- 2005-10-26 CA CA2581225A patent/CA2581225C/en not_active Expired - Fee Related
- 2005-10-26 WO PCT/US2005/038361 patent/WO2006047516A2/en not_active Ceased
- 2005-10-26 MX MX2007004936A patent/MX2007004936A/es not_active Application Discontinuation
- 2005-10-26 CN CN2005800368900A patent/CN101048408B/zh not_active Expired - Fee Related
- 2005-10-26 IN IN2514DEN2007 patent/IN2007DN02514A/en unknown
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- 2007-04-25 TN TNP2007000161A patent/TNSN07161A1/fr unknown
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- 2007-05-07 NO NO20072352A patent/NO20072352L/no not_active Application Discontinuation
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2009
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2011
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| NO20072352L (no) | 2007-05-31 |
| AR051596A1 (es) | 2007-01-24 |
| KR20070057980A (ko) | 2007-06-07 |
| WO2006047516A3 (en) | 2006-10-12 |
| AU2009251216A1 (en) | 2010-01-28 |
| KR100919524B1 (ko) | 2009-10-01 |
| ECSP077421A (es) | 2007-05-30 |
| RU2431635C2 (ru) | 2011-10-20 |
| BRPI0517015A (pt) | 2008-09-30 |
| CA2730374A1 (en) | 2006-05-04 |
| WO2006047516A2 (en) | 2006-05-04 |
| JP2011190281A (ja) | 2011-09-29 |
| IN2007DN02514A (enExample) | 2007-08-03 |
| JP2008518016A (ja) | 2008-05-29 |
| EP1807429A4 (en) | 2010-03-24 |
| TNSN07161A1 (en) | 2008-11-21 |
| AU2005299421A1 (en) | 2006-05-04 |
| CN102241680A (zh) | 2011-11-16 |
| TW200630096A (en) | 2006-09-01 |
| CN101048408B (zh) | 2011-07-06 |
| CA2581225C (en) | 2011-10-25 |
| IL182527A0 (en) | 2007-09-20 |
| AU2005299421B2 (en) | 2010-01-28 |
| US8158634B2 (en) | 2012-04-17 |
| PE20060599A1 (es) | 2006-08-22 |
| CA2581225A1 (en) | 2006-05-04 |
| MA28937B1 (fr) | 2007-10-01 |
| CN101048408A (zh) | 2007-10-03 |
| US20120225869A1 (en) | 2012-09-06 |
| EP1807429A2 (en) | 2007-07-18 |
| US20090247517A1 (en) | 2009-10-01 |
| RU2007119449A (ru) | 2008-12-10 |
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