AU2005299421B2 - Compounds and compositions as inhibitors of Cannabinoid Receptor 1 activity - Google Patents

Compounds and compositions as inhibitors of Cannabinoid Receptor 1 activity Download PDF

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Publication number
AU2005299421B2
AU2005299421B2 AU2005299421A AU2005299421A AU2005299421B2 AU 2005299421 B2 AU2005299421 B2 AU 2005299421B2 AU 2005299421 A AU2005299421 A AU 2005299421A AU 2005299421 A AU2005299421 A AU 2005299421A AU 2005299421 B2 AU2005299421 B2 AU 2005299421B2
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Australia
Prior art keywords
phenyl
dihydro
chloro
pyrazolo
pyrimidin
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Ceased
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AU2005299421A
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AU2005299421A1 (en
Inventor
Ha-Soon Choi
David Archer Ellis
Xiaohui He
Yun He
Hong Liu
Truc Ngoc Nguyen
Zhicheng Wang
David Woodmansee
Baogen Wu
Kunyong Yang
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Novartis AG
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Novartis AG
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Publication of AU2005299421A1 publication Critical patent/AU2005299421A1/en
Priority to AU2009251216A priority Critical patent/AU2009251216A1/en
Application granted granted Critical
Publication of AU2005299421B2 publication Critical patent/AU2005299421B2/en
Assigned to NOVARTIS AG reassignment NOVARTIS AG Request for Assignment Assignors: IRM LLC
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • C07D471/04—Ortho-condensed systems
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    • C07D473/28—Oxygen atom
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    • C07D473/32—Nitrogen atom
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AU2005299421A 2004-10-26 2005-10-26 Compounds and compositions as inhibitors of Cannabinoid Receptor 1 activity Ceased AU2005299421B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2009251216A AU2009251216A1 (en) 2004-10-26 2009-12-24 Compounds and compositions as inhibitors of Cannabinoid Receptor 1 activity

Applications Claiming Priority (5)

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US62250804P 2004-10-26 2004-10-26
US60/622,508 2004-10-26
US67267005P 2005-04-18 2005-04-18
US60/672,670 2005-04-18
PCT/US2005/038361 WO2006047516A2 (en) 2004-10-26 2005-10-26 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity

Related Child Applications (2)

Application Number Title Priority Date Filing Date
AU2007239033A Addition AU2007239033B2 (en) 2006-03-30 2007-03-30 Azolopyrimidines as inhibitors of Cannabinoid 1 activity
AU2009251216A Division AU2009251216A1 (en) 2004-10-26 2009-12-24 Compounds and compositions as inhibitors of Cannabinoid Receptor 1 activity

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AU2005299421A1 AU2005299421A1 (en) 2006-05-04
AU2005299421B2 true AU2005299421B2 (en) 2010-01-28

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US20090247517A1 (en) 2009-10-01
TW200630096A (en) 2006-09-01
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IL182527A0 (en) 2007-09-20
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PE20060599A1 (es) 2006-08-22
CN101048408A (zh) 2007-10-03
WO2006047516A2 (en) 2006-05-04
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US8158634B2 (en) 2012-04-17
EP1807429A4 (en) 2010-03-24
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RU2431635C2 (ru) 2011-10-20
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EP1807429A2 (en) 2007-07-18
BRPI0517015A (pt) 2008-09-30
RU2007119449A (ru) 2008-12-10
TNSN07161A1 (en) 2008-11-21
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IN2007DN02514A (enExample) 2007-08-03
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