BRPI0517015A - compostos e composições como inibidores de atividade de receptor 1 de canabinóide - Google Patents

compostos e composições como inibidores de atividade de receptor 1 de canabinóide

Info

Publication number
BRPI0517015A
BRPI0517015A BRPI0517015-0A BRPI0517015A BRPI0517015A BR PI0517015 A BRPI0517015 A BR PI0517015A BR PI0517015 A BRPI0517015 A BR PI0517015A BR PI0517015 A BRPI0517015 A BR PI0517015A
Authority
BR
Brazil
Prior art keywords
compounds
activity
compositions
inhibitors
cannabinoid receptor
Prior art date
Application number
BRPI0517015-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Hong Liu
Xiaohui He
Ha-Soon Choi
Kunyong Yang
David H Woodmansee
Zhichneg Wang
David Archer Ellis
Baogen Wu
Yun He
Truc Ngoc Nguyen
Original Assignee
Irm Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Irm Llc filed Critical Irm Llc
Publication of BRPI0517015A publication Critical patent/BRPI0517015A/pt

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/18—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 one oxygen and one nitrogen atom, e.g. guanine
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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  • Health & Medical Sciences (AREA)
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  • Pulmonology (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
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  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
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BRPI0517015-0A 2004-10-26 2005-10-26 compostos e composições como inibidores de atividade de receptor 1 de canabinóide BRPI0517015A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US62250804P 2004-10-26 2004-10-26
US67267005P 2005-04-18 2005-04-18
PCT/US2005/038361 WO2006047516A2 (en) 2004-10-26 2005-10-26 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity

Publications (1)

Publication Number Publication Date
BRPI0517015A true BRPI0517015A (pt) 2008-09-30

Family

ID=36228382

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0517015-0A BRPI0517015A (pt) 2004-10-26 2005-10-26 compostos e composições como inibidores de atividade de receptor 1 de canabinóide

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Country Link
US (2) US8158634B2 (enExample)
EP (1) EP1807429A4 (enExample)
JP (2) JP2008518016A (enExample)
KR (1) KR100919524B1 (enExample)
CN (2) CN102241680A (enExample)
AR (1) AR051596A1 (enExample)
AU (2) AU2005299421B2 (enExample)
BR (1) BRPI0517015A (enExample)
CA (2) CA2581225C (enExample)
EC (1) ECSP077421A (enExample)
IL (1) IL182527A0 (enExample)
IN (1) IN2007DN02514A (enExample)
MA (1) MA28937B1 (enExample)
MX (1) MX2007004936A (enExample)
NO (1) NO20072352L (enExample)
PE (1) PE20060599A1 (enExample)
RU (1) RU2431635C2 (enExample)
TN (1) TNSN07161A1 (enExample)
TW (1) TW200630096A (enExample)
WO (1) WO2006047516A2 (enExample)

Families Citing this family (76)

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Publication number Priority date Publication date Assignee Title
CN102558155A (zh) 2003-01-14 2012-07-11 阿伦纳药品公司 作为代谢调节剂的芳基和杂芳基衍生物及其所涉及的疾病如糖尿病和高血糖症的预防和治疗
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