MX2007004482A - Derivados de piridina y la preparacion y el uso terapeutico de los mismos. - Google Patents

Derivados de piridina y la preparacion y el uso terapeutico de los mismos.

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Publication number
MX2007004482A
MX2007004482A MX2007004482A MX2007004482A MX2007004482A MX 2007004482 A MX2007004482 A MX 2007004482A MX 2007004482 A MX2007004482 A MX 2007004482A MX 2007004482 A MX2007004482 A MX 2007004482A MX 2007004482 A MX2007004482 A MX 2007004482A
Authority
MX
Mexico
Prior art keywords
preparation
therapeutic use
pyridine derivatives
group
substituted
Prior art date
Application number
MX2007004482A
Other languages
English (en)
Inventor
Murielle Rinaldi-Carmona
Christian Congy
Lionel Barre
Francisd Barth
Philippe Pointeau
Original Assignee
Sanofi Aventis
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Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MX2007004482A publication Critical patent/MX2007004482A/es

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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Abstract

La invencion se refiere a compuestos de la formula (I), en donde Z es un grupo N(R1)XR2, N(R1)COOR'2 o OCON(R1)R'2; X es un -CO-, -SO2-, -CON(R10)- o -CSN(R10)-; R1 es un atomo de hidrogeno o un grupo alquilo (C1-C4); R2 es un grupo alquilo (C3-C10) no sustituido o sustituido con un grupo CF3; un radical carbociclico no aromatico de (C3-C12), un radical heterociclico, un fenilo sustituido o no sustituido y un alquileno (C1-C2) sustituido por uno o dos sustituyentes diferentes o iguales; R3 es un atomo de hidrogeno, o un grupo alquilo (C1-C4), ciano, alcoximetilo (C1-C4) o hidroximetilo. El metodo inventivo puede utilizarse para preparar y utilizar terapeuticamente dichos compuestos.
MX2007004482A 2004-10-18 2005-10-17 Derivados de piridina y la preparacion y el uso terapeutico de los mismos. MX2007004482A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0411030A FR2876691B1 (fr) 2004-10-18 2004-10-18 Derives de pyridine, leur preparation, leur application en therapeutique
PCT/FR2005/002566 WO2006042955A1 (fr) 2004-10-18 2005-10-17 Derives de pyridine, leur preparation, leur application en therapeutique

Publications (1)

Publication Number Publication Date
MX2007004482A true MX2007004482A (es) 2007-06-13

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FR2899899A1 (fr) * 2006-04-14 2007-10-19 Sanofi Aventis Sa Derives d'aminomethyl pyridine, leur preparation et leur application en therapeutique
TW200815438A (en) * 2006-06-13 2008-04-01 Bayer Schering Pharma Ag Substituted pyrazolopyridines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same
US7781593B2 (en) 2006-09-14 2010-08-24 Hoffmann-La Roche Inc. 5-phenyl-nicotinamide derivatives
FR2922209B1 (fr) * 2007-10-12 2010-06-11 Sanofi Aventis 5,6-DIARYLES PYRIDINES SUBSTITUES EN POSITION 2 et 3, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE.
JP5659224B2 (ja) 2009-05-15 2015-01-28 ノバルティス アーゲー アルドステロンシンターゼ阻害剤としてのアリールピリジン
CN109476599A (zh) * 2016-07-29 2019-03-15 东丽株式会社 胍衍生物和其医药用途
WO2018159650A1 (ja) * 2017-02-28 2018-09-07 東レ株式会社 グアニジン誘導体及びその医薬用途

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FR2198737B1 (es) * 1972-09-13 1975-11-28 Serdex
US5686470A (en) * 1995-02-10 1997-11-11 Weier; Richard M. 2, 3-substituted pyridines for the treatment of inflammation
WO2002055502A1 (en) * 2001-01-02 2002-07-18 Fujisawa Pharmaceutical Co., Ltd. Pyridine derivatives useful as cyclooxygenase inhibitor
US7271266B2 (en) * 2002-03-28 2007-09-18 Merck & Co., Inc. Substituted 2,3-diphenyl pyridines
FR2838439B1 (fr) * 2002-04-11 2005-05-20 Sanofi Synthelabo Derives de terphenyle, leur preparation, les compositions pharmaceutqiues en contenant
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FR2876691A1 (fr) 2006-04-21
AR051221A1 (es) 2006-12-27
EP1805143A1 (fr) 2007-07-11
FR2876691B1 (fr) 2006-12-29
CA2582778A1 (fr) 2006-04-27
US20080021070A1 (en) 2008-01-24
AU2005296959A1 (en) 2006-04-27
NO20072454L (no) 2007-05-14
TW200628450A (en) 2006-08-16
NZ554952A (en) 2009-08-28
JP2008516934A (ja) 2008-05-22
TNSN07114A1 (fr) 2008-06-02
CN101039912A (zh) 2007-09-19
EA200700891A1 (ru) 2007-08-31
ECSP077400A (es) 2007-05-30
IL182385A0 (en) 2007-07-24
UY29163A1 (es) 2006-04-28
BRPI0516926A (pt) 2008-09-23
MA29016B1 (fr) 2007-11-01
WO2006042955A1 (fr) 2006-04-27
KR20070063008A (ko) 2007-06-18
PE20060584A1 (es) 2006-08-18

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