LU85033A1 - Acide azetidinyl-sulfonique et ses analogues - Google Patents

Acide azetidinyl-sulfonique et ses analogues Download PDF

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Publication number
LU85033A1
LU85033A1 LU85033A LU85033A LU85033A1 LU 85033 A1 LU85033 A1 LU 85033A1 LU 85033 A LU85033 A LU 85033A LU 85033 A LU85033 A LU 85033A LU 85033 A1 LU85033 A1 LU 85033A1
Authority
LU
Luxembourg
Prior art keywords
group
amino
hydrogen atom
methyl
substituted
Prior art date
Application number
LU85033A
Other languages
English (en)
French (fr)
Inventor
William A Slusarchyk
David R Kronenthal
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of LU85033A1 publication Critical patent/LU85033A1/fr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
LU85033A 1982-10-06 1983-10-05 Acide azetidinyl-sulfonique et ses analogues LU85033A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43317582A 1982-10-06 1982-10-06
US43317582 1982-10-06

Publications (1)

Publication Number Publication Date
LU85033A1 true LU85033A1 (fr) 1984-05-10

Family

ID=23719123

Family Applications (1)

Application Number Title Priority Date Filing Date
LU85033A LU85033A1 (fr) 1982-10-06 1983-10-05 Acide azetidinyl-sulfonique et ses analogues

Country Status (27)

Country Link
JP (1) JPS5988462A (de)
KR (1) KR900005132B1 (de)
AU (1) AU568312B2 (de)
BE (1) BE897883A (de)
CA (1) CA1253501A (de)
CH (1) CH658858A5 (de)
DD (1) DD222016A5 (de)
DE (1) DE3336262A1 (de)
DK (1) DK457983A (de)
ES (1) ES526282A0 (de)
FI (1) FI833631A (de)
FR (1) FR2534253B1 (de)
GB (1) GB2129428B (de)
GR (1) GR79704B (de)
HU (1) HU190507B (de)
IE (1) IE56600B1 (de)
IL (1) IL69917A (de)
IT (1) IT1171722B (de)
LU (1) LU85033A1 (de)
NL (1) NL8303410A (de)
NO (1) NO833626L (de)
NZ (1) NZ205642A (de)
PH (1) PH24175A (de)
PT (1) PT77458B (de)
SE (1) SE8305509L (de)
SU (1) SU1318146A3 (de)
ZA (1) ZA837491B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0135194A1 (de) * 1983-09-16 1985-03-27 Takeda Chemical Industries, Ltd. Azetidinone und ihre Herstellung
WO1985004876A1 (en) * 1984-04-24 1985-11-07 Takeda Chemical Industries, Ltd. 2-azetidinone derivatives and process for their preparation
US4581170A (en) * 1984-08-03 1986-04-08 E. R. Squibb & Sons, Inc. N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones
JPH0649710B2 (ja) * 1984-08-06 1994-06-29 藤沢薬品工業株式会社 アゼチジノン誘導体およびその製造法
UY34585A (es) 2012-01-24 2013-09-02 Aicuris Gmbh & Co Kg Compuestos b-lactámicos sustituidos con amidina, su preparación y uso

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4337197A (en) * 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates

Also Published As

Publication number Publication date
FI833631A0 (fi) 1983-10-06
GR79704B (de) 1984-10-31
CA1253501A (en) 1989-05-02
KR840006337A (ko) 1984-11-29
FR2534253B1 (fr) 1985-07-26
HU190507B (en) 1986-09-29
PT77458A (en) 1983-11-01
FI833631A (fi) 1984-04-07
IE56600B1 (en) 1991-10-09
DE3336262A1 (de) 1984-04-12
SE8305509D0 (sv) 1983-10-06
ZA837491B (en) 1984-06-27
PT77458B (en) 1986-02-26
GB2129428B (en) 1986-03-19
KR900005132B1 (ko) 1990-07-20
SE8305509L (sv) 1984-04-07
AU1993983A (en) 1984-04-12
JPS5988462A (ja) 1984-05-22
DD222016A5 (de) 1985-05-08
GB2129428A (en) 1984-05-16
BE897883A (fr) 1984-03-30
NL8303410A (nl) 1984-05-01
CH658858A5 (fr) 1986-12-15
PH24175A (en) 1990-03-22
ES8504814A1 (es) 1985-04-16
GB8326626D0 (en) 1983-11-09
IE832354L (en) 1984-04-06
AU568312B2 (en) 1987-12-24
IL69917A (en) 1987-10-20
DK457983A (da) 1984-04-07
IL69917A0 (en) 1984-01-31
NO833626L (no) 1984-04-09
ES526282A0 (es) 1985-04-16
IT1171722B (it) 1987-06-10
FR2534253A1 (fr) 1984-04-13
NZ205642A (en) 1986-08-08
IT8323172A0 (it) 1983-10-06
SU1318146A3 (ru) 1987-06-15
DK457983D0 (da) 1983-10-04

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