BE897883A - Acide azetidinyl sulfonique et analogues a action therapeutique - Google Patents
Acide azetidinyl sulfonique et analogues a action therapeutiqueInfo
- Publication number
- BE897883A BE897883A BE0/211621A BE211621A BE897883A BE 897883 A BE897883 A BE 897883A BE 0/211621 A BE0/211621 A BE 0/211621A BE 211621 A BE211621 A BE 211621A BE 897883 A BE897883 A BE 897883A
- Authority
- BE
- Belgium
- Prior art keywords
- analogs
- sulfonic acid
- therapeutic action
- hydrogen atom
- azetidinyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Beta-lactames portant un substituant (R5,R6,O, C SO3H) en position 1 et un substituant acylamine en position 3. Ils répondant à la formule (I), dans laquelle R1 est un radical acyle, un atome d'hydrogène ou un groupement protecteur de la fonction amine, R2 est un atome d'hydrogène ou un radical méthoxy, R3, R4, R5, et R6 sont identiques ou différents et sont chacun, de préférence, un atome d'hydrogène ou un radical alkyle inférieur. Ces composés sont utilisables comme agents antibactériens.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US43317582A | 1982-10-06 | 1982-10-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE897883A true BE897883A (fr) | 1984-03-30 |
Family
ID=23719123
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/211621A BE897883A (fr) | 1982-10-06 | 1983-09-30 | Acide azetidinyl sulfonique et analogues a action therapeutique |
Country Status (27)
Country | Link |
---|---|
JP (1) | JPS5988462A (fr) |
KR (1) | KR900005132B1 (fr) |
AU (1) | AU568312B2 (fr) |
BE (1) | BE897883A (fr) |
CA (1) | CA1253501A (fr) |
CH (1) | CH658858A5 (fr) |
DD (1) | DD222016A5 (fr) |
DE (1) | DE3336262A1 (fr) |
DK (1) | DK457983A (fr) |
ES (1) | ES8504814A1 (fr) |
FI (1) | FI833631A (fr) |
FR (1) | FR2534253B1 (fr) |
GB (1) | GB2129428B (fr) |
GR (1) | GR79704B (fr) |
HU (1) | HU190507B (fr) |
IE (1) | IE56600B1 (fr) |
IL (1) | IL69917A (fr) |
IT (1) | IT1171722B (fr) |
LU (1) | LU85033A1 (fr) |
NL (1) | NL8303410A (fr) |
NO (1) | NO833626L (fr) |
NZ (1) | NZ205642A (fr) |
PH (1) | PH24175A (fr) |
PT (1) | PT77458B (fr) |
SE (1) | SE8305509L (fr) |
SU (1) | SU1318146A3 (fr) |
ZA (1) | ZA837491B (fr) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1985004876A1 (fr) * | 1984-04-24 | 1985-11-07 | Takeda Chemical Industries, Ltd. | Derives de 2-azetidinone et leur procede de preparation |
EP0135194A1 (fr) * | 1983-09-16 | 1985-03-27 | Takeda Chemical Industries, Ltd. | Azétidinones et leur préparation |
US4581170A (en) * | 1984-08-03 | 1986-04-08 | E. R. Squibb & Sons, Inc. | N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones |
EP0171064B1 (fr) * | 1984-08-06 | 1995-07-12 | Fujisawa Pharmaceutical Co., Ltd. | Dérivés de l'azétidinone et procédé pour leur préparation |
UY34585A (es) | 2012-01-24 | 2013-09-02 | Aicuris Gmbh & Co Kg | Compuestos b-lactámicos sustituidos con amidina, su preparación y uso |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4337197A (en) * | 1980-10-31 | 1982-06-29 | E. R. Squibb & Sons, Inc. | O-sulfated β-lactam hydroxamic acids and intermediates |
-
1983
- 1983-09-19 NZ NZ205642A patent/NZ205642A/en unknown
- 1983-09-22 GR GR72513A patent/GR79704B/el unknown
- 1983-09-30 BE BE0/211621A patent/BE897883A/fr not_active IP Right Cessation
- 1983-10-03 FR FR838315712A patent/FR2534253B1/fr not_active Expired
- 1983-10-04 DK DK457983A patent/DK457983A/da not_active Application Discontinuation
- 1983-10-05 GB GB08326626A patent/GB2129428B/en not_active Expired
- 1983-10-05 NL NL8303410A patent/NL8303410A/nl not_active Application Discontinuation
- 1983-10-05 JP JP58187674A patent/JPS5988462A/ja active Pending
- 1983-10-05 LU LU85033A patent/LU85033A1/fr unknown
- 1983-10-05 DE DE19833336262 patent/DE3336262A1/de not_active Withdrawn
- 1983-10-05 SU SU833652346A patent/SU1318146A3/ru active
- 1983-10-05 NO NO833626A patent/NO833626L/no unknown
- 1983-10-06 IT IT23172/83A patent/IT1171722B/it active
- 1983-10-06 IL IL69917A patent/IL69917A/xx unknown
- 1983-10-06 AU AU19939/83A patent/AU568312B2/en not_active Ceased
- 1983-10-06 FI FI833631A patent/FI833631A/fi not_active Application Discontinuation
- 1983-10-06 CH CH5452/83A patent/CH658858A5/fr not_active IP Right Cessation
- 1983-10-06 HU HU833460A patent/HU190507B/hu not_active IP Right Cessation
- 1983-10-06 KR KR1019830004744A patent/KR900005132B1/ko not_active IP Right Cessation
- 1983-10-06 IE IE2354/83A patent/IE56600B1/en not_active IP Right Cessation
- 1983-10-06 SE SE8305509A patent/SE8305509L/xx not_active Application Discontinuation
- 1983-10-06 ES ES526282A patent/ES8504814A1/es not_active Expired
- 1983-10-06 DD DD83255479A patent/DD222016A5/de not_active IP Right Cessation
- 1983-10-06 ZA ZA837491A patent/ZA837491B/xx unknown
- 1983-10-06 CA CA000438477A patent/CA1253501A/fr not_active Expired
- 1983-10-06 PT PT77458A patent/PT77458B/pt not_active IP Right Cessation
-
1985
- 1985-07-22 PH PH32549A patent/PH24175A/en unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
US4302465B1 (fr) | ||
FR2439790A1 (fr) | Phosphinylalcanoyl prolines a action therapeutique, et leurs procedes de preparation | |
FI823923L (fi) | Antifibrinolytiskt aktiva foereningar | |
BE905109A (fr) | Derives de distamycine et leur procede de fabrication. | |
MY101614A (en) | Improvements in or relating to benzothiophene derivatives as antiasthmatic agents | |
FR2449682A1 (fr) | Derives d'acide quinoleine-carboxylique et leur utilisation en tant qu'agents antimicrobiens | |
DE3477488D1 (en) | Polymethoxybenzyl piperazine derivatives, processes for their preparation and pharmaceutical compositions containing said derivatives | |
BE897883A (fr) | Acide azetidinyl sulfonique et analogues a action therapeutique | |
FR2387989A1 (fr) | Analogues des alcaloides de l'ergot | |
FR2456765A1 (fr) | Composes iminoisoindoliniques, leur procede de preparation et leur application comme pigments | |
FR2445330A1 (fr) | Derives du 11-bromo-14,15-dioxo-e-homo-eburnane leur preparation et leur utilisation comme medicament | |
DK67384D0 (da) | N-iminopyridiniumbetainderivater | |
FR2361351A1 (fr) | Intermediaires de preparation d'homologues de somatostatine | |
FR2447375A1 (fr) | Analogues de la prostaglandine e1 et compositions pharmaceutiques les contenant | |
FR2428045A1 (fr) | Derives silyles de naphtacenones utilisables notamment dans la synthese d'agents antitumeurs | |
FR2592648A1 (fr) | Composes polyfluoroalkylthio-methyliques, leurs procedes de preparation et leurs applications comme agents tensio-actifs ou precurseurs de ces derniers. | |
FR2411173A1 (fr) | Anthranilates de n-hydroxyalkyl-carboxamides et leur application comme reticulants | |
DK422183A (da) | Fremgangsmaade til fremstilling af 5-halogenvinyl-2'-deoxyuridinderivater | |
FR2446284A1 (fr) | Tetrahydro-benzo(c)quinoleine-9(8h)ones | |
FR2603284A1 (fr) | Derives d'acide 7-oxabicyclo(2.2.1.)heptane hydroxamique a action therapeutique | |
ES8304578A1 (es) | Procedimiento para preparar derivados de la ergolina. | |
FR2410640A1 (fr) | Derives de phenoxyalcanolamines, leur preparation et leurs utilisations therapeutiques | |
FR2424912A1 (fr) | Derives de l'imidazole utilisables notamment pour le traitement de l'hypertension | |
BE900718A (fr) | Nouveaux derives du carbapeneme, leur preparation et leur utilisation comme medicaments. | |
ES535903A0 (es) | Procedimiento de preparacion de derivados de nitrosoureas |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: E.R. SQUIBB & SONS INC. Effective date: 19930930 |