BE897883A - AZETIDINYL SULFONIC ACID AND THERAPEUTIC ACTION ANALOGS - Google Patents
AZETIDINYL SULFONIC ACID AND THERAPEUTIC ACTION ANALOGSInfo
- Publication number
- BE897883A BE897883A BE0/211621A BE211621A BE897883A BE 897883 A BE897883 A BE 897883A BE 0/211621 A BE0/211621 A BE 0/211621A BE 211621 A BE211621 A BE 211621A BE 897883 A BE897883 A BE 897883A
- Authority
- BE
- Belgium
- Prior art keywords
- analogs
- sulfonic acid
- therapeutic action
- hydrogen atom
- azetidinyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Beta-lactames portant un substituant (R5,R6,O, C SO3H) en position 1 et un substituant acylamine en position 3. Ils répondant à la formule (I), dans laquelle R1 est un radical acyle, un atome d'hydrogène ou un groupement protecteur de la fonction amine, R2 est un atome d'hydrogène ou un radical méthoxy, R3, R4, R5, et R6 sont identiques ou différents et sont chacun, de préférence, un atome d'hydrogène ou un radical alkyle inférieur. Ces composés sont utilisables comme agents antibactériens.Beta-lactams carrying a substituent (R5, R6, O, C SO3H) in position 1 and an acylamine substituent in position 3. They correspond to formula (I), in which R1 is an acyl radical, a hydrogen atom or a protecting group for the amine function, R2 is a hydrogen atom or a methoxy radical, R3, R4, R5, and R6 are identical or different and are each, preferably, a hydrogen atom or a lower alkyl radical. These compounds can be used as antibacterial agents.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43317582A | 1982-10-06 | 1982-10-06 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE897883A true BE897883A (en) | 1984-03-30 |
Family
ID=23719123
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/211621A BE897883A (en) | 1982-10-06 | 1983-09-30 | AZETIDINYL SULFONIC ACID AND THERAPEUTIC ACTION ANALOGS |
Country Status (27)
| Country | Link |
|---|---|
| JP (1) | JPS5988462A (en) |
| KR (1) | KR900005132B1 (en) |
| AU (1) | AU568312B2 (en) |
| BE (1) | BE897883A (en) |
| CA (1) | CA1253501A (en) |
| CH (1) | CH658858A5 (en) |
| DD (1) | DD222016A5 (en) |
| DE (1) | DE3336262A1 (en) |
| DK (1) | DK457983A (en) |
| ES (1) | ES8504814A1 (en) |
| FI (1) | FI833631A (en) |
| FR (1) | FR2534253B1 (en) |
| GB (1) | GB2129428B (en) |
| GR (1) | GR79704B (en) |
| HU (1) | HU190507B (en) |
| IE (1) | IE56600B1 (en) |
| IL (1) | IL69917A (en) |
| IT (1) | IT1171722B (en) |
| LU (1) | LU85033A1 (en) |
| NL (1) | NL8303410A (en) |
| NO (1) | NO833626L (en) |
| NZ (1) | NZ205642A (en) |
| PH (1) | PH24175A (en) |
| PT (1) | PT77458B (en) |
| SE (1) | SE8305509L (en) |
| SU (1) | SU1318146A3 (en) |
| ZA (1) | ZA837491B (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1985004876A1 (en) * | 1984-04-24 | 1985-11-07 | Takeda Chemical Industries, Ltd. | 2-azetidinone derivatives and process for their preparation |
| EP0135194A1 (en) * | 1983-09-16 | 1985-03-27 | Takeda Chemical Industries, Ltd. | Azetidinones and their production |
| US4581170A (en) * | 1984-08-03 | 1986-04-08 | E. R. Squibb & Sons, Inc. | N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones |
| DE3588039T2 (en) * | 1984-08-06 | 1995-11-16 | Fujisawa Pharmaceutical Co | Azetidinone derivatives and process for their preparation. |
| UY34585A (en) | 2012-01-24 | 2013-09-02 | Aicuris Gmbh & Co Kg | B-LACTAMIC COMPOUNDS REPLACED WITH AMIDINE, ITS PREPARATION AND USE |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4337197A (en) * | 1980-10-31 | 1982-06-29 | E. R. Squibb & Sons, Inc. | O-sulfated β-lactam hydroxamic acids and intermediates |
-
1983
- 1983-09-19 NZ NZ205642A patent/NZ205642A/en unknown
- 1983-09-22 GR GR72513A patent/GR79704B/el unknown
- 1983-09-30 BE BE0/211621A patent/BE897883A/en not_active IP Right Cessation
- 1983-10-03 FR FR838315712A patent/FR2534253B1/en not_active Expired
- 1983-10-04 DK DK457983A patent/DK457983A/en not_active Application Discontinuation
- 1983-10-05 NO NO833626A patent/NO833626L/en unknown
- 1983-10-05 NL NL8303410A patent/NL8303410A/en not_active Application Discontinuation
- 1983-10-05 JP JP58187674A patent/JPS5988462A/en active Pending
- 1983-10-05 LU LU85033A patent/LU85033A1/en unknown
- 1983-10-05 GB GB08326626A patent/GB2129428B/en not_active Expired
- 1983-10-05 SU SU833652346A patent/SU1318146A3/en active
- 1983-10-05 DE DE19833336262 patent/DE3336262A1/en not_active Withdrawn
- 1983-10-06 CH CH5452/83A patent/CH658858A5/en not_active IP Right Cessation
- 1983-10-06 CA CA000438477A patent/CA1253501A/en not_active Expired
- 1983-10-06 ZA ZA837491A patent/ZA837491B/en unknown
- 1983-10-06 IE IE2354/83A patent/IE56600B1/en not_active IP Right Cessation
- 1983-10-06 PT PT77458A patent/PT77458B/en not_active IP Right Cessation
- 1983-10-06 HU HU833460A patent/HU190507B/en not_active IP Right Cessation
- 1983-10-06 SE SE8305509A patent/SE8305509L/en not_active Application Discontinuation
- 1983-10-06 DD DD83255479A patent/DD222016A5/en not_active IP Right Cessation
- 1983-10-06 IT IT23172/83A patent/IT1171722B/en active
- 1983-10-06 ES ES526282A patent/ES8504814A1/en not_active Expired
- 1983-10-06 FI FI833631A patent/FI833631A/en not_active Application Discontinuation
- 1983-10-06 KR KR1019830004744A patent/KR900005132B1/en not_active IP Right Cessation
- 1983-10-06 IL IL69917A patent/IL69917A/en unknown
- 1983-10-06 AU AU19939/83A patent/AU568312B2/en not_active Ceased
-
1985
- 1985-07-22 PH PH32549A patent/PH24175A/en unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: E.R. SQUIBB & SONS INC. Effective date: 19930930 |