SE8305509D0 - ACETIDINYL SULPHONIC ACID AND ANALOGS - Google Patents

ACETIDINYL SULPHONIC ACID AND ANALOGS

Info

Publication number
SE8305509D0
SE8305509D0 SE8305509A SE8305509A SE8305509D0 SE 8305509 D0 SE8305509 D0 SE 8305509D0 SE 8305509 A SE8305509 A SE 8305509A SE 8305509 A SE8305509 A SE 8305509A SE 8305509 D0 SE8305509 D0 SE 8305509D0
Authority
SE
Sweden
Prior art keywords
acetidinyl
analogs
sulphonic acid
image
hydrogen atoms
Prior art date
Application number
SE8305509A
Other languages
Swedish (sv)
Other versions
SE8305509L (en
Inventor
W A Slusarchyk
D R Kronenthal
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of SE8305509D0 publication Critical patent/SE8305509D0/en
Publication of SE8305509L publication Critical patent/SE8305509L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Abstract

Antibiotic activity is exhibited by beta -lactams having an <IMAGE> substituent in the 1-position and an acylamino substituent in the 3- position, R<5> and R<6> being hydrogen atoms at various defined substituents or R<5> and R<6> together completing a ring. The corresponding 3-amino compounds may be produced as intermediates. The compounds may be of the formula:- <IMAGE> or salts or esters thereof, R1 being hydrogen or acyl and R2, R3 and R4 being hydrogen atoms or substituents.
SE8305509A 1982-10-06 1983-10-06 ACETIDINYL SULPHONIC ACID AND ANALOGS SE8305509L (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US43317582A 1982-10-06 1982-10-06

Publications (2)

Publication Number Publication Date
SE8305509D0 true SE8305509D0 (en) 1983-10-06
SE8305509L SE8305509L (en) 1984-04-07

Family

ID=23719123

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8305509A SE8305509L (en) 1982-10-06 1983-10-06 ACETIDINYL SULPHONIC ACID AND ANALOGS

Country Status (27)

Country Link
JP (1) JPS5988462A (en)
KR (1) KR900005132B1 (en)
AU (1) AU568312B2 (en)
BE (1) BE897883A (en)
CA (1) CA1253501A (en)
CH (1) CH658858A5 (en)
DD (1) DD222016A5 (en)
DE (1) DE3336262A1 (en)
DK (1) DK457983A (en)
ES (1) ES8504814A1 (en)
FI (1) FI833631A (en)
FR (1) FR2534253B1 (en)
GB (1) GB2129428B (en)
GR (1) GR79704B (en)
HU (1) HU190507B (en)
IE (1) IE56600B1 (en)
IL (1) IL69917A (en)
IT (1) IT1171722B (en)
LU (1) LU85033A1 (en)
NL (1) NL8303410A (en)
NO (1) NO833626L (en)
NZ (1) NZ205642A (en)
PH (1) PH24175A (en)
PT (1) PT77458B (en)
SE (1) SE8305509L (en)
SU (1) SU1318146A3 (en)
ZA (1) ZA837491B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985004876A1 (en) * 1984-04-24 1985-11-07 Takeda Chemical Industries, Ltd. 2-azetidinone derivatives and process for their preparation
EP0135194A1 (en) * 1983-09-16 1985-03-27 Takeda Chemical Industries, Ltd. Azetidinones and their production
US4581170A (en) * 1984-08-03 1986-04-08 E. R. Squibb & Sons, Inc. N-hydroxyl protecting groups and process and intermediates for the preparation of 3-acylamino-1-hydroxy-2-azetidinones
DE3588039T2 (en) * 1984-08-06 1995-11-16 Fujisawa Pharmaceutical Co Azetidinone derivatives and process for their preparation.
UY34585A (en) 2012-01-24 2013-09-02 Aicuris Gmbh & Co Kg B-LACTAMIC COMPOUNDS REPLACED WITH AMIDINE, ITS PREPARATION AND USE

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4337197A (en) * 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates

Also Published As

Publication number Publication date
FI833631A0 (en) 1983-10-06
NO833626L (en) 1984-04-09
IL69917A (en) 1987-10-20
AU568312B2 (en) 1987-12-24
GB8326626D0 (en) 1983-11-09
LU85033A1 (en) 1984-05-10
GR79704B (en) 1984-10-31
KR840006337A (en) 1984-11-29
AU1993983A (en) 1984-04-12
IL69917A0 (en) 1984-01-31
IE832354L (en) 1984-04-06
IT8323172A0 (en) 1983-10-06
PH24175A (en) 1990-03-22
BE897883A (en) 1984-03-30
JPS5988462A (en) 1984-05-22
FR2534253A1 (en) 1984-04-13
NZ205642A (en) 1986-08-08
DK457983A (en) 1984-04-07
CH658858A5 (en) 1986-12-15
FI833631A (en) 1984-04-07
PT77458A (en) 1983-11-01
GB2129428B (en) 1986-03-19
HU190507B (en) 1986-09-29
KR900005132B1 (en) 1990-07-20
DE3336262A1 (en) 1984-04-12
DD222016A5 (en) 1985-05-08
GB2129428A (en) 1984-05-16
NL8303410A (en) 1984-05-01
PT77458B (en) 1986-02-26
DK457983D0 (en) 1983-10-04
SE8305509L (en) 1984-04-07
ES526282A0 (en) 1985-04-16
ES8504814A1 (en) 1985-04-16
CA1253501A (en) 1989-05-02
ZA837491B (en) 1984-06-27
IT1171722B (en) 1987-06-10
IE56600B1 (en) 1991-10-09
FR2534253B1 (en) 1985-07-26
SU1318146A3 (en) 1987-06-15

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Effective date: 19870402