LU73993A1 - - Google Patents

Info

Publication number
LU73993A1
LU73993A1 LU73993A LU73993A LU73993A1 LU 73993 A1 LU73993 A1 LU 73993A1 LU 73993 A LU73993 A LU 73993A LU 73993 A LU73993 A LU 73993A LU 73993 A1 LU73993 A1 LU 73993A1
Authority
LU
Luxembourg
Application number
LU73993A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of LU73993A1 publication Critical patent/LU73993A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
LU73993A 1974-12-13 1975-12-11 LU73993A1 (https=)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
LU73993A1 true LU73993A1 (https=) 1976-11-11

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
LU73993A LU73993A1 (https=) 1974-12-13 1975-12-11

Country Status (27)

Country Link
US (1) US4051252A (https=)
JP (1) JPS5182266A (https=)
AT (1) AT343653B (https=)
BE (1) BE836528A (https=)
CA (1) CA1059523A (https=)
CH (1) CH622250A5 (https=)
CS (1) CS189731B2 (https=)
DD (1) DD125484A5 (https=)
DE (1) DE2458965C3 (https=)
DK (1) DK137082C (https=)
ES (1) ES443429A1 (https=)
FI (1) FI753493A7 (https=)
FR (1) FR2293928A1 (https=)
GB (1) GB1490306A (https=)
HK (1) HK52580A (https=)
HU (1) HU173557B (https=)
IE (1) IE42208B1 (https=)
IL (1) IL48642A (https=)
KE (1) KE3078A (https=)
LU (1) LU73993A1 (https=)
NL (1) NL7514521A (https=)
NO (1) NO145382C (https=)
PL (1) PL99858B1 (https=)
SE (1) SE419645B (https=)
SU (1) SU604487A3 (https=)
YU (1) YU315275A (https=)
ZA (1) ZA757777B (https=)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
ZA200301701B (en) * 2000-09-15 2004-03-01 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002022605A1 (en) 2000-09-15 2002-03-21 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6989385B2 (en) 2000-12-21 2006-01-24 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
BR0212841A (pt) 2001-09-26 2004-08-03 Pharmacia Italia Spa Derivado ativo de aminoindazole como inibidores de cinase, processo para sua preparação e composições farmacêuticas que os contém
WO2003066629A2 (en) * 2002-02-06 2003-08-14 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
US20040009981A1 (en) 2002-03-15 2004-01-15 David Bebbington Compositions useful as inhibitors of protein kinases
MXPA04011417A (es) 2002-05-17 2005-02-14 Pharmacia Italia Spa Derivados de aminoindazol activos como inhibidores de cinasa, procedimiento para su preparacion y composiciones farmaceuticas que los comprenden.
MY141867A (en) 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
CN1319968C (zh) 2002-08-02 2007-06-06 沃泰克斯药物股份有限公司 用作gsk-3的抑制剂的吡唑组合物
WO2004041285A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
US7601718B2 (en) 2003-02-06 2009-10-13 Vertex Pharmaceuticals Incorporated Compositions useful as inhibitors of protein kinases
US7592340B2 (en) * 2003-12-04 2009-09-22 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
ATE542814T1 (de) 2005-08-18 2012-02-15 Vertex Pharma Pyrazinkinaseinhibitoren
MX2008005814A (es) * 2005-11-03 2008-10-15 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasa.
ES2385404T3 (es) * 2006-04-14 2012-07-24 Abbott Laboratories Procedimiento para la preparación de ureas de indazolilo que inhiben los receptores vaniloides de subtipo 1 (VR1)
CA2668429A1 (en) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
ES2347721T3 (es) 2006-12-19 2010-11-03 Vertex Pharmaceuticals, Inc. Aminopirimidinas utiles como inhibidores de proteina quinasas.
AU2008226457B2 (en) 2007-03-09 2014-03-20 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
EP2137183B1 (en) 2007-03-09 2011-09-28 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
EP2134709A1 (en) 2007-03-09 2009-12-23 Vertex Pharmaceuticals, Inc. Aminopyridines useful as inhibitors of protein kinases
NZ580343A (en) 2007-04-13 2012-03-30 Vertex Pharma Aminopyrimidines useful as kinase inhibitors
JP5389785B2 (ja) 2007-05-02 2014-01-15 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害剤として有用なチアゾールおよびピラゾール
MX2009011811A (es) * 2007-05-02 2010-01-14 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasa.
CA2694381A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
EP2164842A2 (en) * 2007-05-24 2010-03-24 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
NZ582879A (en) * 2007-07-31 2012-03-30 Vertex Pharma Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
MX2011002312A (es) * 2008-09-03 2011-04-26 Vertex Pharma Co-cristales y formulaciones farmaceuticas que comprenden los mismos.
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
WO2014017936A2 (en) 2012-07-24 2014-01-30 Bial- Portela & Ca, S.A. Urea compounds and their use as enzyme inhibitors
JP2015528013A (ja) * 2012-07-27 2015-09-24 ビアル−ポルテラ エ コンパニア,ソシエダッド アノニマ 置換ウレア化合物の合成方法
AU2014293731B2 (en) 2013-07-24 2018-03-08 Bial - Portela & Ca, S.A. Imidazolecarboxamides and their use as FAAH inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3277100A (en) * 1963-05-31 1966-10-04 Du Pont Novel substituted pyrazoles
NL6707299A (https=) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
AT343653B (de) 1978-06-12
IE42208L (en) 1976-06-13
SU604487A3 (ru) 1978-04-25
AU8717075A (en) 1977-06-09
NO145382C (no) 1982-03-10
ATA939775A (de) 1977-10-15
DD125484A5 (https=) 1977-04-20
IL48642A0 (en) 1976-02-29
FR2293928A1 (fr) 1976-07-09
HK52580A (en) 1980-09-26
YU315275A (en) 1982-02-28
CA1059523A (en) 1979-07-31
DE2458965A1 (de) 1976-06-16
GB1490306A (en) 1977-11-02
FI753493A7 (https=) 1976-06-14
SE7513990L (sv) 1976-06-14
NL7514521A (nl) 1976-06-15
DE2458965C3 (de) 1979-10-11
SE419645B (sv) 1981-08-17
ES443429A1 (es) 1977-04-16
NO754024L (https=) 1976-06-15
CH622250A5 (https=) 1981-03-31
FR2293928B1 (https=) 1979-09-21
DK137082B (da) 1978-01-16
DE2458965B2 (de) 1979-02-22
JPS5182266A (en) 1976-07-19
US4051252A (en) 1977-09-27
PL99858B1 (pl) 1978-08-31
IL48642A (en) 1979-12-30
DK137082C (da) 1978-06-19
NO145382B (no) 1981-11-30
DK567275A (da) 1976-06-14
IE42208B1 (en) 1980-06-18
ZA757777B (en) 1976-11-24
KE3078A (en) 1980-10-03
CS189731B2 (en) 1979-04-30
BE836528A (fr) 1976-06-11
HU173557B (hu) 1979-06-28

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