KR930703353A - 황체화 호르몬 방출 호르몬(lhrh)길항제 - Google Patents

황체화 호르몬 방출 호르몬(lhrh)길항제

Info

Publication number
KR930703353A
KR930703353A KR1019930701418A KR930701418A KR930703353A KR 930703353 A KR930703353 A KR 930703353A KR 1019930701418 A KR1019930701418 A KR 1019930701418A KR 930701418 A KR930701418 A KR 930701418A KR 930703353 A KR930703353 A KR 930703353A
Authority
KR
South Korea
Prior art keywords
hormone
parent compound
lhrh
antagonist
dala
Prior art date
Application number
KR1019930701418A
Other languages
English (en)
Other versions
KR100244624B1 (ko
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of KR930703353A publication Critical patent/KR930703353A/ko
Application granted granted Critical
Publication of KR100244624B1 publication Critical patent/KR100244624B1/ko

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/23Luteinising hormone-releasing hormone [LHRH]; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Endocrinology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
KR1019930701418A 1990-11-10 1991-11-08 황체 형성 호르몬 방출 호르몬(lhrh) 길항제 및 이를 함유하는 약제학적 조성물 KR100244624B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN90108955A CN1036343C (zh) 1990-11-10 1990-11-10 新促黄体生成素释放激素拮抗类似物的制备方法
CN90108955.9 1990-11-10
PCT/EP1991/002110 WO1992008733A1 (en) 1990-11-10 1991-11-08 Lhrh-antagonists

Publications (2)

Publication Number Publication Date
KR930703353A true KR930703353A (ko) 1993-11-29
KR100244624B1 KR100244624B1 (ko) 2000-02-15

Family

ID=4881223

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019930701418A KR100244624B1 (ko) 1990-11-10 1991-11-08 황체 형성 호르몬 방출 호르몬(lhrh) 길항제 및 이를 함유하는 약제학적 조성물

Country Status (29)

Country Link
EP (1) EP0564466B1 (ko)
KR (1) KR100244624B1 (ko)
CN (1) CN1036343C (ko)
AT (1) ATE149520T1 (ko)
AU (1) AU662496B2 (ko)
CA (1) CA2095932C (ko)
CZ (1) CZ284168B6 (ko)
DE (1) DE69125024T2 (ko)
DK (1) DK0564466T3 (ko)
EE (1) EE03141B1 (ko)
ES (1) ES2100965T3 (ko)
FI (1) FI933156A (ko)
GR (1) GR3023389T3 (ko)
HR (1) HRP920585B1 (ko)
IE (1) IE913915A1 (ko)
LT (1) LT3971B (ko)
LV (1) LV10106B (ko)
NO (1) NO931697L (ko)
NZ (1) NZ240505A (ko)
PH (1) PH31178A (ko)
PL (1) PL170564B1 (ko)
PT (1) PT99458B (ko)
RU (1) RU2123499C1 (ko)
SI (1) SI9111779B (ko)
SK (1) SK281319B6 (ko)
UA (1) UA41300C2 (ko)
WO (1) WO1992008733A1 (ko)
YU (1) YU48831B (ko)
ZA (1) ZA918847B (ko)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2164096T3 (es) * 1992-12-18 2002-02-16 Abbott Lab Antagonistas de lhrh que comprenden restos de aminoacilo modificados en posicion 5 y 6.
US6828415B2 (en) 1993-02-19 2004-12-07 Zentaris Gmbh Oligopeptide lyophilisate, their preparation and use
DE4305225A1 (de) * 1993-02-19 1994-08-25 Asta Medica Ag Neues Herstellverfahren für Cetrorelix Lyophilisat
DE4338015A1 (de) * 1993-11-08 1995-05-11 Asta Medica Ag Verwendung von D-glucopyranuronsäuren und deren Derivaten zum Einbau in pharmakologisch wirksame Peptide und deren Salze
US5843901A (en) * 1995-06-07 1998-12-01 Advanced Research & Technology Institute LHRH antagonist peptides
US5968547A (en) 1997-02-24 1999-10-19 Euro-Celtique, S.A. Method of providing sustained analgesia with buprenorphine
CN101037472B (zh) * 2006-03-14 2013-03-27 中国人民解放军军事医学科学院毒物药物研究所 具有低组胺释放作用的促黄体生成素释放激素拮抗剂
CN102675418B (zh) * 2011-03-15 2016-04-20 中国人民解放军军事医学科学院毒物药物研究所 Lhrh拮抗剂衍生物、其制备方法及用途
CN103524599B (zh) * 2012-07-05 2016-04-20 中国人民解放军军事医学科学院毒物药物研究所 环肽lhrh拮抗剂衍生物及其药物用途
CN104418936B (zh) * 2013-08-20 2018-06-05 中国人民解放军军事医学科学院毒物药物研究所 Lhrh拮抗剂衍生物及其药物用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4801577A (en) * 1987-02-05 1989-01-31 Syntex (U.S.A.) Inc. Nonapeptide and decapeptide analogs of LHRH useful as LHRH antagonists
US4851385A (en) * 1987-07-15 1989-07-25 Indiana University Foundation LHRH antagonist analogs having low histamine-release activity

Also Published As

Publication number Publication date
SK281319B6 (sk) 2001-02-12
EP0564466B1 (en) 1997-03-05
FI933156A0 (fi) 1993-07-09
CA2095932A1 (en) 1992-05-11
LV10106B (en) 1995-04-20
PL170564B1 (pl) 1996-12-31
DE69125024T2 (de) 1997-07-17
CA2095932C (en) 2003-02-25
EE03141B1 (et) 1998-12-15
SK45393A3 (en) 1993-10-06
CN1036343C (zh) 1997-11-05
RU2123499C1 (ru) 1998-12-20
ES2100965T3 (es) 1997-07-01
IE913915A1 (en) 1992-05-20
GR3023389T3 (en) 1997-08-29
EP0564466A1 (en) 1993-10-13
FI933156A (fi) 1993-07-09
YU177991A (sh) 1994-06-24
NZ240505A (en) 1993-04-28
DE69125024D1 (de) 1997-04-10
ZA918847B (en) 1992-08-26
WO1992008733A1 (en) 1992-05-29
LV10106A (lv) 1994-05-10
HRP920585B1 (en) 2000-08-31
KR100244624B1 (ko) 2000-02-15
SI9111779B (en) 2001-12-31
AU8861291A (en) 1992-06-11
CN1061605A (zh) 1992-06-03
CZ284168B6 (cs) 1998-09-16
PT99458B (pt) 1999-02-26
DK0564466T3 (da) 1997-08-25
NO931697L (no) 1993-07-07
PH31178A (en) 1998-03-20
YU48831B (sh) 2002-03-18
SI9111779A (en) 1997-04-30
ATE149520T1 (de) 1997-03-15
LTIP1513A (en) 1995-06-26
HRP920585A2 (en) 1997-04-30
AU662496B2 (en) 1995-09-07
CZ84893A3 (en) 1994-02-16
PT99458A (pt) 1992-10-30
UA41300C2 (uk) 2001-09-17
PL295427A1 (en) 1993-09-06
NO931697D0 (no) 1993-05-10
LT3971B (en) 1996-05-27

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