KR890016019A - 페닐 피리미디논 유도체 - Google Patents

페닐 피리미디논 유도체 Download PDF

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Publication number
KR890016019A
KR890016019A KR1019890005246A KR890005246A KR890016019A KR 890016019 A KR890016019 A KR 890016019A KR 1019890005246 A KR1019890005246 A KR 1019890005246A KR 890005246 A KR890005246 A KR 890005246A KR 890016019 A KR890016019 A KR 890016019A
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KR
South Korea
Prior art keywords
compound
formula
halogen
hydrogen
fluorine
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KR1019890005246A
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English (en)
Inventor
로버트 퍼라이오 트레보
조세프 타폴크제이 데이비드
존 휘틀 알랜
Original Assignee
존 린드레이 렝
임페리알 케미칼 인더스트리스 피엘씨
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Publication date
Priority claimed from GB888809552A external-priority patent/GB8809552D0/en
Priority claimed from GB898906329A external-priority patent/GB8906329D0/en
Application filed by 존 린드레이 렝, 임페리알 케미칼 인더스트리스 피엘씨 filed Critical 존 린드레이 렝
Publication of KR890016019A publication Critical patent/KR890016019A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C07D239/36—One oxygen atom as doubly bound oxygen atom or as unsubstituted hydroxy radical
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Farming Of Fish And Shellfish (AREA)

Abstract

내용 없음

Description

페닐 피리미디논 유도체
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (13)

  1. 다음 구조식(I) 화합물.
    식중, R1및R2는 독립적으로 할로겐 또는 니트로로부터 선택되고 ; R3및R|4는 독립적으로 할로겐 또는 수소로 부터 선택되며 ; R5는 수소, 할로겐 또는 시아노이고 ; R6는 할로겐 또는 할로알킬인데 ; 단, R1,R2,R3및 R4모두가 불소는 아님.
  2. 제 1항에 의해, 최소한 하나의 R1및R2가 플루오로, 클로로, 브로모 또는 요오도인 화합물.
  3. 제 2항에 있어서, R1및R2둘다가 클로로인 화합물.
  4. 제 2항에 있어서, R1및R2둘다가 플루오르인 화합물.
  5. 전기한 항의 어느 한 항에 있어서, R6가 트리플루오로메틸 또는 펜타플루오로에틸인 화합물.
  6. 전기한 항의 어느 한 항에 있어서, R5가 수소, 염소 또는 불소인 화합물.
  7. 제 1항에 있어서, 다음 구조식(IA)인 화합물.
    식중, R1'또는 R2'중의 하나는 할로이고 다른 하나는 할로겐 또는 니트로이며 ; R5'는 수소 또는 할로겐이고 ; R6'는 트리플루오로메틸 또는 펜타플루오로에틸임.
  8. 제 1 항에 정의된 바와같은 구조식(I) 화합물의 살충적 또는 살비적 효과량을 해충 또는 해충의 소재지에 사용하는 것으로 구성되는, 해충 또는 진드기 해충을 조절하거나 살충하는 방법.
  9. 희석제 또는 담체와 함께 구조식(I) 화합물로 구성된 살충 또는 살비 조성물.
  10. 다음 구조식(IV) 화합물.
    식중, R3,R4,R5및 R6는 제 1 항에 정의된 바와같고, R8및 R9는 아미노 또는 제 1 항에 정의된 바와같은 그룹 R1또는 R2인데 단, 최소한 하나의 R8또는 R9가 아미노임.
  11. 다음 구조식(IIA) 화합물.
    식중, R11는 염소, R12는 불소 및 R13는 요오드이거나 또는 R11는니트로, R12는 브로모 및 R13는 브로모이거나 또는 R11는 아미노, R12는 플루오로 및 R13는 클로로임.
  12. 다음 구조식(IIIA) 또는 (VA)의 피리미디논 화합물.
    식중, R13는 수소, 할로겐 또는 시아노이고, R14는 할로 또는 할로알킬인데, 단, (a) R13가 시아노일때, R14는 염소 이외의 것이고; (b) R13및 R14둘다가 할로는 아니며;(c) R13가 할로일때, R14는 모노플루오로메틸 이외의 것이고 ; (d) R13가 수소일때, R14는 할로 또는 할로메틸 그룹이 아님.
    식중, R10은 수소 또는 C1-4알킬이고 R15는 시아노이고, R16는 구조식(V)에 관해 정의된 바와같은 R6이거나 또는 R15는 수소 또는 불소이외의 할로겐이고 R16는 펜타플루오로에틸 또는 디플루오로메틸임.
  13. 다음 구조식(II) 화합물을
    식중, R1,R2,R3및 R4는 제 1 항에 정의된 바와같고, R7는 이탈그룹임.
    다음 구조식(III) 화합물과 반응시키고,
    식중, R5및 R6는 제 1 항에 정의된 바와같음
    그 후에 원한다면 하나 이상의 다음 단계, 즉 그룹 R5,R2,R3또는 R4를 이러한 다른 그룹으로 전환시키는 것을 행하는 것으로 구성되는, 제 1 항의 구조식(I) 화합물의 제조방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019890005246A 1988-04-22 1989-04-21 페닐 피리미디논 유도체 KR890016019A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB888809552A GB8809552D0 (en) 1988-04-22 1988-04-22 Novel compounds
GB8809552.6 1988-04-22
GB8906329.1 1989-03-22
GB898906329A GB8906329D0 (en) 1989-03-22 1989-03-22 Novel compounds

Publications (1)

Publication Number Publication Date
KR890016019A true KR890016019A (ko) 1989-11-28

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ID=26293803

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019890005246A KR890016019A (ko) 1988-04-22 1989-04-21 페닐 피리미디논 유도체

Country Status (17)

Country Link
US (1) US5077297A (ko)
EP (1) EP0338686B1 (ko)
JP (1) JPH026476A (ko)
KR (1) KR890016019A (ko)
CN (1) CN1037705A (ko)
AT (1) ATE107633T1 (ko)
AU (1) AU618799B2 (ko)
CS (1) CS274447B2 (ko)
DE (1) DE68916315T2 (ko)
GB (1) GB8906946D0 (ko)
HU (1) HU204973B (ko)
NZ (1) NZ228782A (ko)
PH (1) PH26786A (ko)
PL (1) PL158930B1 (ko)
RO (2) RO104617B1 (ko)
RU (1) RU1833137C (ko)
YU (1) YU82389A (ko)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5149810A (en) * 1988-04-22 1992-09-22 Imperial Chemical Industries Plc Pyrimidine compounds
GB8908638D0 (en) * 1989-04-17 1989-06-01 Ici Plc Novel compounds
CA2014533A1 (en) * 1989-04-24 1990-10-24 Lester S. Mills Process for the production of 4 - hydroxy -6- polyfluoroalkylpyrimidines
GB9022445D0 (en) * 1990-10-16 1990-11-28 Ici Plc Heterocyclic compounds
GB9022444D0 (en) * 1990-10-16 1990-11-28 Ici Plc Heterocyclic compounds
CA2094949A1 (en) * 1992-04-28 1993-10-29 Eiki Nagano Pyrimidone derivatives and their use
GB9306184D0 (en) * 1993-03-25 1993-05-19 Zeneca Ltd Heteroaromatic compounds
US6271392B1 (en) 1994-10-07 2001-08-07 Rhone-Poulenc Inc. Intermediates useful for the synthesis of 1-arylpyrrole pesticides
AU4398597A (en) * 1996-10-03 1998-04-24 Nissan Chemical Industries Ltd. Heterocycle-fused pyrimidinone derivatives and herbicides
US6165942A (en) * 1996-10-03 2000-12-26 Nissan Chemical Industries, Ltd. Heterocycle-fused pyrimidinone derivative and herbicidal composition
WO1999044997A1 (fr) * 1998-03-06 1999-09-10 Ube Industries, Ltd. 6-(α-FLUOROALKYL)-4-PYRIMIDONES ET LEUR PROCEDE DE PRODUCTION
AU2002337498B2 (en) * 2001-09-21 2006-08-10 Mitsubishi Pharma Corporation 3-substituted-4-pyrimidone derivatives
AU2002953128A0 (en) * 2002-12-05 2002-12-19 Osmose (Australia) Pty Ltd Surface treatment for wood and wood products
TWI455919B (zh) * 2008-04-09 2014-10-11 Du Pont 製備３－三氟甲基查耳酮（ｃｈａｌｃｏｎｅ）之方法

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3185689A (en) * 1965-05-25 Tolyl-x-(jh)-pyrimidones
CA888730A (en) * 1971-12-21 W. Lutz Albert 2,3,5-substituted-6-trifluoromethyl-1,3-diazin-4-ones and their use as herbicides
GB1035092A (en) * 1959-08-14 1966-07-06 Du Pont Improvements relating to herbicides and novel 3-substituted uracils
US3235358A (en) * 1962-09-06 1966-02-15 Du Pont Control of undesirable vegetation
IT635567A (ko) * 1959-08-14 1900-01-01
GB1035097A (en) * 1962-12-07 1966-07-06 Du Pont Improvements relating to herbicides
GB1035098A (en) * 1962-12-07 1966-07-06 Du Pont Improvements relating to herbicides
GB1035091A (en) * 1962-12-07 1966-07-06 Du Pont Improvements relating to herbicides
US3291592A (en) * 1964-04-20 1966-12-13 Du Pont Method for increasing sugar cane yield
US3869457A (en) * 1968-06-17 1975-03-04 American Cyanamid Co 2,3,5-substituted-6-trifluoromethyl-1,3-diazin-4-ones
IL32279A (en) * 1968-06-17 1973-01-30 American Cyanamid Co Halo substituted uracils and hydrouracils and preparation of same
US3580913A (en) * 1968-06-17 1971-05-25 American Cyanamid Co Process for preparing substituted-6-trifluoromethyluracils
US3823135A (en) * 1972-12-26 1974-07-09 Shell Oil Co Pyrimidone herbicides
US4147528A (en) * 1973-04-23 1979-04-03 Rohm And Haas Company 6-Oxopyrimidine plant growth regulators
IT1153066B (it) * 1982-11-18 1987-01-14 Mentedison S P A Derivati del pirimidin-4-one ad attivita' erbicida
JPS6183146A (ja) * 1984-09-28 1986-04-26 Nippon Soda Co Ltd ２，５−ジハロ−３−トリフルオロメチルアニリン及びその製造方法
US5022915A (en) * 1990-03-01 1991-06-11 Ici Americas Inc. Substituted 2,4-diarylpyrimidines and their use as herbicides

Also Published As

Publication number Publication date
HUT49792A (en) 1989-11-28
AU618799B2 (en) 1992-01-09
DE68916315T2 (de) 1994-10-06
CN1037705A (zh) 1989-12-06
HU204973B (en) 1992-03-30
CS247989A2 (en) 1990-06-13
US5077297A (en) 1991-12-31
EP0338686A3 (en) 1990-11-28
RO104617B1 (en) 1993-03-30
ATE107633T1 (de) 1994-07-15
PH26786A (en) 1992-10-13
EP0338686B1 (en) 1994-06-22
DE68916315D1 (de) 1994-07-28
AU3317989A (en) 1989-10-26
PL158930B1 (pl) 1992-10-30
NZ228782A (en) 1991-07-26
EP0338686A2 (en) 1989-10-25
GB8906946D0 (en) 1989-05-10
RO107525B1 (ro) 1993-12-30
YU82389A (en) 1991-02-28
CS274447B2 (en) 1991-04-11
JPH026476A (ja) 1990-01-10
RU1833137C (ru) 1993-08-07

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