KR910016699A - 헤테로사이클릭아세토니트릴 및 그의 살균성 용도 - Google Patents

헤테로사이클릭아세토니트릴 및 그의 살균성 용도 Download PDF

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KR910016699A
KR910016699A KR1019910003852A KR910003852A KR910016699A KR 910016699 A KR910016699 A KR 910016699A KR 1019910003852 A KR1019910003852 A KR 1019910003852A KR 910003852 A KR910003852 A KR 910003852A KR 910016699 A KR910016699 A KR 910016699A
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phenyl
compound
het
integer
alkyl
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하워드 쉐이버 스티븐
하워드 레이놀즈 찰스
마이클 스자팩스 에드워드
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원본미기재
롬 앤드 하스 캄파니
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/26—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/57—Nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D241/12—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

내용 없음

Description

헤테로사이클릭아세토니트릴 및 그의 살균성 용도
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (12)

  1. 하기 일반식의 화합물, 및 그의 작물학적으로 허용되는 거울상 이성체, 산부가염 및 금속 착화합물:
    상기식에서, Ar1은 할로겐, 니트로, 시아노, (C1-C12)알킬, (C1-C12)할로알킬, (C3-C8)사이클로알킬, (C5-C8)사이클로알케닐, (C2-C12)알케닐, (C2-C12)알키닐, (C1-C12)알콕시, (C1-C12)할로알콕시,(C1-C12) 알킬티오, (C1-C12)알킬설피닐, (C1-C12)알킬설포닐, 페닐, 페녹시, 펜(C1-C12)알킬, 펜(C2-C12)알케닐, 펜(C2-C12)알키닐 및 (C5-C12)사이클로알킬(C1-C6)알킬로 이루어진 그룹중에서 독립적으로 선택되는 3개 이하의 치환체로 임의로 치환된 C6내지 C10아틸 그룹으로 선택되고; Ar2는 치환체가 Ar1에 대해 상기 열거한 치환체중에서 독립적으로 선택되는, 임의로 치환된(C6-C10)아릴 그룹이거나, 또는, Ar2는 티오페닐 또는 푸라닐일수 있으며; Het는 3 내지 5 개의 탄소 원자 및 1 내지 3개의 질소원자로 이루어지는 6-원 헤테로사이클릭 고리이고 ; n은 정수 2 또는 3이나 ; 단, Het가 피라지닐이고 n이 2인 경우에는, Ar1및 Ar2는 둘다 페닐일 수 없다.
  2. 제2항에 있어서, Ar1및 Ar2가 페닐, 또는 메틸, 할로메틸, 할로겐 및 알콕시로 이루어진 그룹중에서 선택되는 2개 이항의 치환체로 치환된 페닐로부터 독립적으로 선택되고, Het가 4 또는 5개의 탄소원자 및 1 또는 2개의 질소 원자로 이루어진 6원 헤테로사이클릭 고리이며, n이 정수 2 또는 3인 화합물.
  3. 제1항에 있어서, Ar1이 페닐 또는 2- 또는 4-할로치환된 페닐이고, Ar2가 페닐 또는 3- 또는 4-할로치환된 페닐이며, Het가 피라지닐, 3-피리딜 또는 5-피리미딜이고, n이 정수 2인 화합물.
  4. 제1항에 있어서, Ar1이 2-또는 4-클로로-, 2-또는 4-플루오르페닐이고, Ar2가 4-클로로-또는 4-플루오로페닐이며, Het가 3-피리딜 또는 5-피리미딜이며, n이 정수 2인 화합물.
  5. 살균 효과량의 제1항의 화합물 및 작물학적으로 허용되는 불활성 담체를 포함하는 살균성 조성물.
  6. 살균 효과량의 제2항의 화합물 및 작물학적으로 허용되는 불활성 담체를 포함하는 살균성 조성물.
  7. 살균 효과량의 제3항의 화합물 및 작물학적으로 허용되는 불활성 담체를 포함하는 살균성 조성물.
  8. 살균 효과량의 제4항의 화합물 및 작물학적으로 허용되는 불활성 담체를 포함하는 살균성 조성물.
  9. 균류 또는 상기 균류의 서식지에 살균 효과량의 하기 일반식의 화합물 및 그의 작물학적으로 허용되는 거울 상이성체, 산 부가염 및 금속 착화합물을 접촉시킴을 포함하는 균류의 방제 방법:
    상기식에서, Ar1은 할로겐, 니트로, 시아노, (C1-C12)알킬, (C1-C12)할로알킬, (C3-C8)사이클로알킬, (C5-C8)사이클로알케닐, (C2-C12)알케닐, (C2-C12)알키닐, (C1-C12)알콕시, (C1-C12)할로알콕시,(C1-C12) 알킬티오, (C1-C12)알킬설피닐, (C1-C12)알킬설포닐, 페녹시, 페닐, 펜(C1-C12)알킬, 펜(C2-C12)알케닐, 펜(C2-C12)알키닐 및 (C5-C6)사이클로알킬(C1-C6)알킬로 이루어진 그룹중에서 독립적으로 선택되는 3개 이하의 치환체로 임의로 치환된 C6내지 C10아틸 그룹으로 선택되고; Ar2는 치환체가 Ar1에 대해 상기 열거한 치환체중에서 독립적으로 선택되는, 임의로 치환된(C6-C10)아릴 그룹이거나, 또는, Ar2는 티옵닐 또는 푸라닐일수 있으며; Het는 3 내지 5개의 탄소원자 및 1 내지 3개의 질소원자로 이루어지는 6-원 헤테로사이클릭고리이고; n은 정수 2 또는 3이다.
  10. 제9항에 있어서, Ar1및 Ar2가 페닐, 또는 메틸, 할로메틸, 할로겐 및 알콕시로 이루어진 그룹중에서 선택되는 2개 이하의 치환체로 치환된 페닐로부터 독립적으로 선택되고, Het가 4 또는 5개의 탄소원자 및 1 또는 2개의 질소 원자로 이루어진 6원 헤테로사이클릭 고리이며, n이 정수 2 또는 3인 방법.
  11. 제9항에 있어서, Ar1이 페닐 또는 2-또는 4-할로치환된 페닐이고, Ar2가 페닐 또는 3-또는 4-할로치환된 페닐이며, Het가 피라지닐, 3-피리딜 또는 5-피리미딜이고, n이 정수 2인 방법.
  12. 제9항에 있어서, Ar1이 2-또는 4-클로로-, 또는 2-또는 4-플루오로페닐이고, Ar2가 4-클로로-또는 4-플루오로페닐이며, Het가 3-피리딜 또는 5-피리미딜이며, n이 정수 2인 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019910003852A 1990-03-12 1991-03-11 헤테로사이클릭아세토니트릴 및 그의 살균성 용도 KR910016699A (ko)

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US (2) US5397793A (ko)
EP (1) EP0451948B1 (ko)
JP (1) JP3034971B2 (ko)
KR (1) KR910016699A (ko)
AR (1) AR248399A1 (ko)
AT (1) ATE116297T1 (ko)
AU (1) AU648065B2 (ko)
BR (1) BR9100962A (ko)
CA (1) CA2037162A1 (ko)
DE (1) DE69106199T2 (ko)
ES (1) ES2069198T3 (ko)
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US5484787A (en) 1996-01-16
ES2069198T3 (es) 1995-05-01
AR248399A1 (es) 1995-08-18
CA2037162A1 (en) 1991-09-13
DE69106199D1 (de) 1995-02-09
EP0451948B1 (en) 1994-12-28
BR9100962A (pt) 1991-11-05
DE69106199T2 (de) 1995-05-11
NZ237307A (en) 1993-12-23
JPH04217666A (ja) 1992-08-07
US5397793A (en) 1995-03-14
EP0451948A1 (en) 1991-10-16
AU648065B2 (en) 1994-04-14
ATE116297T1 (de) 1995-01-15
JP3034971B2 (ja) 2000-04-17
AU7280891A (en) 1991-09-12

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