KR840004712A - 벤조퀴논 유도체의 제조방법 - Google Patents

벤조퀴논 유도체의 제조방법 Download PDF

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KR840004712A
KR840004712A KR1019830001533A KR830001533A KR840004712A KR 840004712 A KR840004712 A KR 840004712A KR 1019830001533 A KR1019830001533 A KR 1019830001533A KR 830001533 A KR830001533 A KR 830001533A KR 840004712 A KR840004712 A KR 840004712A
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신지 데라오 (외 2)
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구라바야시 이꾸시로
다께다야꾸 힝고오교 가부시끼 가이샤
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Abstract

내용 없음

Description

벤조퀴논 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (3)

  1. 하기 일반식(Ⅱ)의 화합물을 산화시킴을 특징으로 하는 하기 일반식(Ⅰ)의 화합물의 제조방법.
    [상기 식에서, R1및 R2는 같거나 다르며 각각 메틸 또는 메톡시이고 ; n은 0∼21의 정수이고 ; m은 0 또는 1이고 ; Z는 식의 기(여기서, R3및 R4는 동일 또는 상이하며 각각은 수소원자 또는 임의로 치환될 수 있는 알킬기이거나, 또는 R3및 R4는 인접한 질소 원자와 함께 모르폴리노기를 형성함), 식 -COR5의 기(여기서, R5는 α-아미노산 잔기 또는 치환되거나 치환되지 않은 글루코사민 잔기), 식
    의 기(여기서, R6는 탄소 원자수 1∼3의 2가의 탄화수소기), 식의 기(여기서, R6는 전기 정의한 바와 같음), 식 -(CH=CH)1-COR7의 기(여기서, 1은 1∼4의 정수이고 R7은 히드록시, 메톡시 또는 메틸임)이고 ; X는 수소 또는 임의로 보호될 수 있는 히드록시기이며 ; Y는 임의로 보호될 수 있는 히드록시기임].
  2. 하기 일반식(Ⅲ)의 화합물 또는 그의 반응성 유도체를 α-아미노산 또는 치환되거나 치환되지 않은 글루코사민과 항께 카르복실기에서 반응시킴을 특징으로 하는 하기 일반식(Ia)의 화합물의 제조방법.
    (상기 식에서, R1및 R2는 같거나 다르며 각각 메틸 또는 메톡시이고 ; n은 0∼21의 정수이며 ; R5는 α-아미노산 잔기 또는 치환되거나 치환되지 않은 글루코사민 잔기임).
  3. 하기 일반식(Ⅸ)의 화합물을 포름산 존재하 하기 일반식(Ⅷ)의 화합물과 반응시킴을 특징으로 하는 하기 일반식(Ⅰ-b)의 화합물의 제조방법.
    (상기 식에서, R1및 R2는 같거나 다르며 각각 메틸 또는 메톡시이고 ; n은 0∼21의 정수이고, m은 0 또는 1이고 ; R3및 R4는 같거나 다르며 각각 수소 또는 임의로 치환될 수 있는 알킬기이거나, 또는 R3및 R4는 인접한 질소 원자와 함께 모르폴리노기를 형성함).
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019830001533A 1982-04-13 1983-04-13 벤조퀴논 유도체의 제조방법 KR900008110B1 (ko)

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JP57062224A JPS58177934A (ja) 1982-04-13 1982-04-13 ベンゾキノン誘導体
JP62224 1982-04-13

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US (4) US4526719A (ko)
EP (1) EP0092136B1 (ko)
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AT (1) ATE15182T1 (ko)
CA (1) CA1242708A (ko)
DE (1) DE3360655D1 (ko)
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US4751303A (en) 1988-06-14
US4943645A (en) 1990-07-24
EP0092136B1 (en) 1985-08-28
US4874752A (en) 1989-10-17
CA1242708A (en) 1988-10-04
EP0092136A1 (en) 1983-10-26
DE3360655D1 (en) 1985-10-03
HU195767B (en) 1988-07-28
JPH038327B2 (ko) 1991-02-05
KR900008110B1 (ko) 1990-10-31

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