KR840003618A - 2-시아노벤즈 이미다졸 유도체의 제조방법 - Google Patents

2-시아노벤즈 이미다졸 유도체의 제조방법 Download PDF

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KR840003618A
KR840003618A KR1019830000465A KR830000465A KR840003618A KR 840003618 A KR840003618 A KR 840003618A KR 1019830000465 A KR1019830000465 A KR 1019830000465A KR 830000465 A KR830000465 A KR 830000465A KR 840003618 A KR840003618 A KR 840003618A
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South Korea
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optionally substituted
groups
group
halogen atoms
lower alkyl
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KR1019830000465A
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KR900003393B1 (ko
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지로동 레이몽 (외 1)
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미쉘 쇼메뜨
롱-쁠랑 아그로시미
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A01N43/52—1,3-Diazoles; Hydrogenated 1,3-diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Agronomy & Crop Science (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Wood Science & Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Photoreceptors In Electrophotography (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Processing And Handling Of Plastics And Other Materials For Molding In General (AREA)
  • Protection Of Static Devices (AREA)
  • Treatment And Processing Of Natural Fur Or Leather (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

내용 없음

Description

2-시아노벤즈 이미다졸 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (3)

  1. 일반식(Ⅰ)의 2-시아노벤즈이미다졸과 일반식(Ⅱ)의 할라이드를 반응시킴을 특징으로 하여 일반식(Ⅲ)의 2-시아노벤즈이미다졸의 유도체를 제조하는 방법.
    상기 일반식에서 n은 0,1,2 또는 3의 정수를 나타내며; R은 할로겐원자 또는 하나 이상의 할로겐 원자에 의해 임의로 치환된 저급알킬 래디칼; 하나 이상의 할로겐원자에 의해 또는 페닐기에 의해 임의로 치환된 저급 알콕시기; 하나 이상의 할로겐원자에 의해 임으로 치환된 저급 알킬티오기; 저급 알케닐기; 저급 알키닐기; 하나 또는 둘의 같거나 서로 다른 저급 알킬이에 의해 임의로 치환된 아미노기; 니트로기; 시아노기; 시아네이토기; 티오시아네이토기; 이소티오시아네이토기; 저급 알킬술포닐기; 하나 또는 둘의 같거나 서로 다른 저급 알킬기에 의해 임의로 치환된 술파모일기; 저급 알킬술피닐기; 하나 이상의 할로겐원자에 의해 임의로 치환된 아실기; 2∼5 탄소원자를 함유한 알콕시카르보닐기를 나타내며, 만일 n이 2이상이면 치환체 R은 같거나 서로 다를 수 있다; R'는 하나 이상의 할로겐원자에 의해 임의로 치환된 저급 알킬 또는 시클로알킬기; 스스로 임의 치환된 하나 또는 둘의 같거나 서로 다른 저급 알킬기 의해 임의로 치환된 아미노기; 질소원자와 헤테로시클릭환을 형성하는 두 기에 의해 치환된 질소원자, 4∼6 환멤버 및 환에서 1∼3 헤테로원자를 함유하며 임의로 치환된 헤테로시클릭환 자체를 나타내며 "저급"은 6탄소원자 이하를 함유하는 유기기를 의미한다.
  2. 제1항에 있어서, 2-시아노벤즈이미다졸과 할라이드의 반응이 산수용체의 존재하 극성 비양자성 용매에서 수행되는 방법.
  3. 제1항에 있어서, 2-시아노벤즈이미다졸의 알칼리금속염 또는 암모늄염과 할라이드의 반응이 극성비양자성 용매에서 수행되는 반응.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019830000465A 1982-02-09 1983-02-07 2-시아노벤즈 이미다졸 유도체의 제조방법 KR900003393B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR02281 1982-02-09
FR82-02281 1982-02-09
FR8202281A FR2521141A1 (fr) 1982-02-09 1982-02-09 Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides

Publications (2)

Publication Number Publication Date
KR840003618A true KR840003618A (ko) 1984-09-15
KR900003393B1 KR900003393B1 (ko) 1990-05-18

Family

ID=9270908

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KR1019830000465A KR900003393B1 (ko) 1982-02-09 1983-02-07 2-시아노벤즈 이미다졸 유도체의 제조방법

Country Status (30)

Country Link
US (1) US4536502A (ko)
EP (1) EP0087375B1 (ko)
JP (1) JPS58148864A (ko)
KR (1) KR900003393B1 (ko)
AT (1) ATE15663T1 (ko)
AU (1) AU568291B2 (ko)
BG (3) BG40955A3 (ko)
BR (1) BR8300628A (ko)
CA (1) CA1229850A (ko)
CS (1) CS235308B2 (ko)
CU (1) CU21531A3 (ko)
DD (1) DD208753A5 (ko)
DE (1) DE3360804D1 (ko)
DK (1) DK52683A (ko)
ES (1) ES519099A0 (ko)
FR (1) FR2521141A1 (ko)
GB (1) GB2114567B (ko)
GR (1) GR78101B (ko)
HU (1) HU190441B (ko)
IL (1) IL67857A (ko)
MA (1) MA19706A1 (ko)
NZ (1) NZ203207A (ko)
OA (1) OA07319A (ko)
PH (2) PH19082A (ko)
PL (1) PL135987B1 (ko)
PT (1) PT76212B (ko)
RO (2) RO90226A (ko)
SU (1) SU1346043A3 (ko)
TR (1) TR21444A (ko)
ZA (1) ZA83798B (ko)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2559150B1 (fr) * 1984-02-06 1986-06-27 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides
FR2572401B1 (fr) * 1984-10-26 1986-12-26 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation et leur utilisation comme fongicides et acaricides
US4728741A (en) * 1985-01-08 1988-03-01 Smithkline Beckman Corporation 1-substituted-2-mercapto benzimidazole compounds and intermediates
GB8519920D0 (en) * 1985-08-08 1985-09-18 Fbc Ltd Fungicides
FR2594437A1 (fr) * 1986-02-19 1987-08-21 Rhone Poulenc Agrochimie Nouveaux derives du cyano-2 benzimidazole, leur preparation, les compositions les contenant et leur utilisation comme fongicide
FR2608898A1 (fr) * 1986-12-30 1988-07-01 Rhone Poulenc Agrochimie Associations fongicides a base de cyanobenzimidazole et d'un fongicide systemique
CA1339133C (en) * 1987-03-13 1997-07-29 Rikuo Nasu Imidazole compounds and biocidal composition comprising the same for controlling harmful organisms
FR2643264B1 (fr) * 1989-02-20 1991-04-26 Rhone Poulenc Sante Trifluoromethoxy-5 benzimidazolamine-2, procede pour sa preparation et medicaments la contenant
AU638614B2 (en) * 1990-11-20 1993-07-01 Sumitomo Chemical Company, Limited Benzimidazole derivative, a method for producing the same, its intermediate compounds and an agricultural and horticultural fungicide containing the benzimidazole derivative as an active ingredient
US5395952A (en) * 1991-06-03 1995-03-07 Sumitomo Chemical Company, Limited Benzimidazole derivatives agricultural and horticultural fungicides containing the same as an active ingredient and intermediate compounds thereof
NZ242756A (en) * 1991-06-03 1994-07-26 Sumitomo Chemical Co Benzimidazole derivatives having a fused ring which contains 1 or 2 o atoms and at least 1 -cf2- unit; use as fungicides; and precursors
DE4139950A1 (de) * 1991-12-04 1993-06-09 Bayer Ag, 5090 Leverkusen, De 2-cyanobenzimidazole, ein verfahren zu ihrer herstellung und ihre verwendung und neue vorprodukte
ES2087418T3 (es) * 1991-12-16 1996-07-16 Ciba Geigy Ag Derivados de acidos sulfonicos de benzimidazol como microbicidas.
US5472974A (en) * 1992-02-26 1995-12-05 Sumitomo Chemical Company, Limited Benzimidazole derivatives, agricultural and horticultural fungicides containing the same as an active ingredient and intermediate compounds thereof
BR9306708A (pt) * 1992-07-10 1998-12-08 Ciba Geigy Ag Microbicidas
JPH08500352A (ja) * 1992-08-25 1996-01-16 チバーガイギー アクチェンゲゼルシャフト 殺微生物剤としてのベンズイミダゾール誘導体
DE4237597A1 (de) * 1992-11-06 1994-05-11 Bayer Ag Substituierte Benzimidazole
DE4237617A1 (de) * 1992-11-06 1994-05-11 Bayer Ag Verwendung von substituierten Benzimidazolen
US5376657A (en) * 1992-12-10 1994-12-27 Ciba-Geigy Corporation Microbicides
TW242556B (ko) * 1993-02-05 1995-03-11 Ciba Geigy
DE19831985A1 (de) 1998-07-16 2000-01-20 Bayer Ag Substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen
DE19920551A1 (de) 1999-05-05 2000-11-09 Bayer Ag Substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen
DE10049468A1 (de) * 2000-10-06 2002-04-11 Bayer Ag N-Alkoxyalkyl-substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen
DE102004042958A1 (de) * 2004-09-02 2006-03-09 Bayer Healthcare Ag Neue antiparasitäre Kombination von Wirkstoffen
DE102005000746A1 (de) * 2005-01-05 2006-07-13 Bayer Healthcare Ag Bekämpfung der Histomoniasis
DE102009038950A1 (de) 2009-08-26 2011-03-03 Bayer Animal Health Gmbh Neue antiparasitäre Kombination von Wirkstoffen

Family Cites Families (14)

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Publication number Priority date Publication date Assignee Title
FR1450505A (fr) * 1965-04-24 1966-06-24 Chimetron Sarl Nouvelles cétones dérivées des benzimidazoles sulfonés et sulfamidés
AU413408B2 (en) * 1966-09-19 1971-05-19 2-cyanobenzimidazoles
DE2014293A1 (de) * 1969-03-29 1970-10-08 Fisons Ltd., Felixstowe, Suffolk (Grossbritannien) Substituierte Benzimidazole und Verfahren zu ihrer Herstellung und Verwendung
NL7013343A (ko) * 1969-09-26 1971-03-30
BE792402A (fr) * 1971-12-07 1973-06-07 Ciba Geigy Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent
BE795098A (fr) * 1972-02-09 1973-08-07 Bayer Ag Nouveaux 1-aminosulfonyl-2-amino-benzimidazoles, leur procede de preparation et leur application comme fongicides
DE2242785A1 (de) * 1972-08-31 1974-03-14 Bayer Ag 1-alkylsulfonyl-2-trifluormethylbenzimidazole, verfahren zu ihrer herstellung sowie ihre verwendung als ektoparasitenmittel
US4122184A (en) * 1973-09-14 1978-10-24 Eli Lilly And Company Benzimidazole insecticides
US4018790A (en) * 1975-05-08 1977-04-19 Eli Lilly And Company Substituted 1-sulfonylbenzimidazoles
US4174454A (en) * 1975-08-28 1979-11-13 Eli Lilly And Company Alkylidenylmethyl-substituted 1-sulfonylbenzimidazoles
PT65486B (en) * 1975-08-28 1978-03-24 Lilly Co Eli Process for the preparation of carbonil-substituted 1-sulfonylbenzimidazoles
US4230868A (en) * 1979-04-17 1980-10-28 Eli Lilly And Company α-Alkyl-α-hydroxybenzyl-substituted 1-sulfonylbenzimidazoles
US4289782A (en) * 1979-04-17 1981-09-15 Eli Lilly And Company Antiviral 1-sulfonylbenzimidazoles
US4338329A (en) * 1979-11-14 1982-07-06 Eli Lilly And Company Antiviral method employing 1-sulfonylbenzimidazoles

Also Published As

Publication number Publication date
GB2114567B (en) 1985-10-30
AU1117483A (en) 1983-08-18
TR21444A (tr) 1984-07-01
GR78101B (ko) 1984-09-26
CU21531A3 (en) 1987-06-09
FR2521141B1 (ko) 1984-03-16
NZ203207A (en) 1985-02-28
RO90232A (ro) 1986-12-10
EP0087375B1 (fr) 1985-09-18
DK52683D0 (da) 1983-02-08
ATE15663T1 (de) 1985-10-15
GB2114567A (en) 1983-08-24
GB8303340D0 (en) 1983-03-09
SU1346043A3 (ru) 1987-10-15
PL240471A1 (en) 1984-07-02
BG37831A3 (en) 1985-08-15
BG40955A3 (en) 1987-03-14
PL135987B1 (en) 1986-01-31
ZA83798B (en) 1983-10-26
JPS58148864A (ja) 1983-09-05
ES8406447A1 (es) 1984-03-01
DD208753A5 (de) 1984-04-11
CS235308B2 (en) 1985-05-15
BG37995A3 (en) 1985-09-16
CA1229850A (en) 1987-12-01
HU190441B (en) 1986-09-29
EP0087375A1 (fr) 1983-08-31
IL67857A0 (en) 1983-06-15
PT76212B (fr) 1986-01-27
DK52683A (da) 1983-08-10
PH20207A (en) 1986-10-20
FR2521141A1 (fr) 1983-08-12
PH19082A (en) 1985-12-19
AU568291B2 (en) 1987-12-24
BR8300628A (pt) 1983-11-08
MA19706A1 (fr) 1983-10-01
KR900003393B1 (ko) 1990-05-18
DE3360804D1 (en) 1985-10-24
IL67857A (en) 1987-08-31
US4536502A (en) 1985-08-20
ES519099A0 (es) 1984-03-01
PT76212A (fr) 1983-03-01
OA07319A (fr) 1984-08-31
RO90226A (ro) 1986-10-30

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